Preclinical Evaluation of theEffects of Trazpiroben (TAK-906), a Novel, Potent Dopamine D2/D3 Receptor Antagonist for the Management of Gastroparesis

Effect of dopamine D2/D3 receptor antagonist sulpiride on amphetamine-induced changes in striatal extracellular dopamine

10.1016/s0014-2999(01)00936-0 ◽

2001 ◽

Vol 418 (3) ◽

pp. 201-206 ◽

Cited By ~ 15

Author(s):

Jason N Jaworski ◽

Rueben A Gonzales ◽

Patrick K Randall

Keyword(s):

Receptor Antagonist ◽

D3 Receptor ◽

Extracellular Dopamine ◽

Dopamine D2 ◽

Induced Changes

The Dopamine D2/D3 Receptor Antagonist APD421 in Combination with Ondansetron Effectively Prevents Acute Cisplatin-Induced Nausea and Vomiting (CINV)

Annals of Oncology ◽

10.1016/s0923-7534(20)34118-1 ◽

2012 ◽

Vol 23 ◽

pp. ix507 ◽

Cited By ~ 1

Author(s):

J. Herrstedt ◽

Y. Summers ◽

G. Daugaard ◽

T.B. Christensen ◽

K. Holmskov ◽

...

Keyword(s):

Receptor Antagonist ◽

Nausea And Vomiting ◽

D3 Receptor ◽

Blonanserin, an Antipsychotic and Dopamine D2/D3 Receptor Antagonist, and Ameliorated Alcohol Dependence

Clinical Neuropharmacology ◽

10.1097/wnf.0b013e318280028a ◽

2013 ◽

Vol 36 (2) ◽

pp. 68-69 ◽

Cited By ~ 3

Author(s):

Manabu Takaki ◽

Hiroshi Ujike

Keyword(s):

Alcohol Dependence ◽

Receptor Antagonist ◽

D3 Receptor ◽

F15063, a potential antipsychotic with dopamine D2/D3 receptor antagonist and 5-HT1A receptor agonist properties: Influence on immediate-early gene expression in rat prefrontal cortex and striatum

10.1016/j.ejphar.2009.08.019 ◽

2009 ◽

Vol 620 (1-3) ◽

pp. 27-35 ◽

Cited By ~ 19

Author(s):

Liesbeth A. Bruins Slot ◽

Fabrice Lestienne ◽

Catherine Grevoz-Barret ◽

Adrian Newman-Tancredi ◽

Didier Cussac

Keyword(s):

Gene Expression ◽

Prefrontal Cortex ◽

Receptor Antagonist ◽

Receptor Agonist ◽

Immediate Early Gene ◽

Early Gene ◽

Immediate Early ◽

D3 Receptor ◽

Early Gene Expression ◽

F15063, a potential antipsychotic with dopamine D2/D3 receptor antagonist, 5-HT1A receptor agonist and dopamine D4 receptor partial agonist properties: Influence on neuronal firing and neurotransmitter release

10.1016/j.ejphar.2009.02.001 ◽

2009 ◽

Vol 607 (1-3) ◽

pp. 74-83 ◽

Cited By ~ 7

Author(s):

Marie-Bernadette Assié ◽

Ouissame Mnie-Filali ◽

Véronique Ravailhe ◽

Christelle Benas ◽

Marc Marien ◽

...

Keyword(s):

Receptor Antagonist ◽

Neurotransmitter Release ◽

Receptor Agonist ◽

Partial Agonist ◽

Neuronal Firing ◽

D3 Receptor ◽

Dopamine D4 Receptor ◽

Dopamine D2 ◽

D4 Receptor

Su1764 TAK-906, A NOVEL DOPAMINE D2/D3 RECEPTOR ANTAGONIST FOR THE TREATMENT OF GASTROPARESIS

Gastroenterology ◽

10.1016/s0016-5085(20)32292-7 ◽

2020 ◽

Vol 158 (6) ◽

pp. S-638-S-639

Author(s):

Roger Whiting ◽

Agnes Choppin ◽

Gary Luehr

Keyword(s):

Receptor Antagonist ◽

D3 Receptor ◽

The MCH1 receptor antagonist SNAP 94847 induces sensitivity to dopamine D2/D3 receptor agonists in rats and mice

10.1016/j.ejphar.2008.10.051 ◽

2009 ◽

Vol 602 (1) ◽

pp. 66-72 ◽

Cited By ~ 16

Author(s):

Douglas A. Marsteller ◽

Christophe P.G. Gerald ◽

Ron Kong ◽

Manuel Cajina ◽

Douglas A. Craig ◽

...

Keyword(s):

Receptor Antagonist ◽

D3 Receptor ◽

Receptor Agonists ◽

Dopamine D2 ◽

Rats And Mice

Decreased Dopamine D2/D3-Receptor Binding in the Temporal Lobe and the Bilateral Basal Ganglia in patients with Temporal Lobe Epilepsy

Klinische Neurophysiologie ◽

10.1055/s-0032-1301572 ◽

2012 ◽

Vol 43 (01) ◽

Author(s):

VE Bernedo Paredes ◽

H Schwartz ◽

M Gartenschläger ◽

HG Buchholz ◽

...

Keyword(s):

Basal Ganglia ◽

Temporal Lobe Epilepsy ◽

Temporal Lobe ◽

Receptor Binding ◽

D3 Receptor ◽

Dopamine D3 Receptor Antagonist SB-277011A Influences Cell Firing in the Rat Ventral Tegmental Area, Parallel Role with the Cannabinoid System in Addiction and Neuropsychiatry Disorders?

The Open Neuropsychopharmacology Journal ◽

10.2174/1876523800902020086 ◽

2009 ◽

Vol 2 (2) ◽

pp. 86-92

Author(s):

Francesca Formenti ◽

Viviana Sonntag ◽

Francesco Congestri ◽

Francesco Crespi

Keyword(s):

Receptor Antagonist ◽

Ventral Tegmental Area ◽

Dopamine D3 Receptor ◽

D3 Receptor ◽

Cannabinoid System ◽

Dopamine D3 ◽

Cell Firing ◽

Ventral Tegmental

Increased Dopamine D2/D3 Receptor Binding After Recovery from Anorexia Nervosa Measured by Positron Emission Tomography and [11C]Raclopride

Biological Psychiatry ◽

10.1016/j.biopsych.2005.05.003 ◽

2005 ◽

Vol 58 (11) ◽

pp. 908-912 ◽

Cited By ~ 219

Author(s):

Guido K. Frank ◽

Ursula F. Bailer ◽

Shannan E. Henry ◽

Wayne Drevets ◽

Carolyn C. Meltzer ◽

...

Keyword(s):

Positron Emission Tomography ◽

Anorexia Nervosa ◽

Receptor Binding ◽

Emission Tomography ◽

D3 Receptor ◽

Dopamine D2 ◽

Positron Emission