scholarly journals Thyrotropin-releasing hormone receptors (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database

2019 ◽  
Vol 2019 (4) ◽  
Author(s):  
Anthony P. Davenport ◽  
Marvin Gershengorn ◽  
Rebecca Hills
Keyword(s):  
Hormone Receptors ◽  
Thyrotropin Releasing Hormone ◽  
Releasing Hormone ◽  
Kd Values ◽  
Trh Analogues ◽  
Trh Receptors

Thyrotropin-releasing hormone (TRH) receptors (provisional nomenclature as recommended by NC-IUPHAR [13]) are activated by the endogenous tripeptide TRH (pGlu-His-ProNH2). TRH and TRH analogues fail to distinguish TRH1 and TRH2 receptors [28]. [3H]TRH (human, mouse, rat) is able to label both TRH1 and TRH2 receptors with Kd values of 13 and 9 nM respectively. Synthesis and biology of ring-modified L-Histidine containing TRH analogues has been reported [22].

Studies on the transport of thyrotropin-releasing hormone (TRH) analogues in Caco-2 cell monolayers

2003 ◽  
Vol 55 (5) ◽  
pp. 603-608 ◽  
Author(s):  
Akihiko Urayama ◽  
Shizuo Yamada ◽  
Yoshiharu Deguchi ◽  
Yuki Ohmori ◽  
Ryohei Kimura
Keyword(s):  
Thyrotropin Releasing Hormone ◽  
Releasing Hormone ◽  
Cell Monolayers ◽  
Trh Analogues

Synthesis and biology of new thyrotropin-Releasing hormone (TRH) analogues

2002 ◽  
Vol 10 (1) ◽  
pp. 189-194 ◽  
Author(s):  
Rahul Jain ◽  
Jatinder Singh ◽  
Jeffery H Perlman ◽  
Marvin C Gershengorn
Keyword(s):  
Thyrotropin Releasing Hormone ◽  
Releasing Hormone ◽  
Trh Analogues
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