scholarly journals Synthesis, Characterization and Biological Evaluation of Some Benzothiazole Derivatives as Potential Antimicrobial Agent.

2016 ◽  
Vol 11 (05) ◽  
pp. 105-112
Author(s):  
Ashok G. Awale
Keyword(s):  
Antimicrobial Agent ◽  
Biological Evaluation ◽  
Benzothiazole Derivatives

Purification and Biological Evaluation of Some Bioactive Metabolomics as Antimicrobial Agent

2013 ◽  
Vol 10 (5) ◽  
pp. 437-443
Author(s):  
Ramar Perumal Samy ◽  
Gautam Sethi ◽  
Vincent T.K Chow
Keyword(s):  
Antimicrobial Agent ◽  
Biological Evaluation

Synthesis and biological evaluation of benzothiazole derivatives as potent antitumor agents

2005 ◽  
Vol 15 (14) ◽  
pp. 3328-3332 ◽  
Author(s):  
Masao Yoshida ◽  
Ichiro Hayakawa ◽  
Noriyuki Hayashi ◽  
Toshinori Agatsuma ◽  
Youko Oda ◽  
...  
Keyword(s):  
Antitumor Agents ◽  
Biological Evaluation ◽  
Benzothiazole Derivatives ◽  
Synthesis And Biological Evaluation

scholarly journals Identification and biological evaluation of novel benzothiazole derivatives bearing a pyridine-semicarbazone moiety as apoptosis inducers via activation of procaspase-3 to caspase-3

MedChemComm ◽  
2019 ◽  
Vol 10 (3) ◽  
pp. 465-477 ◽  
Author(s):  
Junjie Ma ◽  
Xin Ni ◽  
Yali Gao ◽  
Kun Huang ◽  
Jiaan Liu ◽  
...  
Keyword(s):  
Caspase 3 ◽  
Biological Evaluation ◽  
Benzothiazole Derivatives

A series of benzothiazole derivatives bearing a pyridine-semicarbazone moiety were identified as apoptosis inducers via activation of procaspase-3 to caspase-3.

scholarly journals Synthesis, spectral studies and biological activity of 2, 3-disubstituted imidazo [2, 1-b] benzothiazole derivatives

2018 ◽  
Vol 6 (01) ◽  
pp. 01-08
Author(s):  
Yashveer Singh ◽  
Baljeet Kaur ◽  
Amandeep Kaur ◽  
Vivek Kumar Gupta ◽  
Monika Gupta
Keyword(s):  
Antimicrobial Activity ◽  
Catalytic Domain ◽  
Biological Evaluation ◽  
Spectral Studies ◽  
Thiazole Ring ◽  
Standard Drug ◽  
Atp Binding Site ◽  
Benzothiazole Derivatives ◽  
Antibacterial And Antifungal ◽  
Synthesis And Biological Evaluation

Benzothiazole is a heterocyclic compound formed by the fusion of benzene and thiazole ring. The moiety had been reported to act via competing with ATP binding site at the catalytic domain of tyrosine kinase. The present work involves the synthesis and biological evaluation of 4, 5 disubstituted imidazo [2, 1-b] benzothiazole derivatives. The antimicrobial activity of the synthesized derivatives was carried out against Gram + ve bacteria Staphylococcus aureus (MTCC 3160) and Gram –ve bacteria Bordetella bronchiseptica (MTCC 6838), Pseudomonas aeruginosa (T11) and fungal strains Candida albicans (MTCC 1637). Ciprofloxacin and Fluconazole were used as standard drug for antibacterial and antifungal activity respectively. The compounds 6a1, 6a2, 6a3, 6b1 and 8a1 exhibited good antimicrobial activity against all the strains. The derivative 8a1 was further screened for anticancer activity against MCF-7 cell line using Doxorubicin as standard. The structures of the synthesized compounds were established by IR and NMR spectral studies.

scholarly journals Design, Recombinant Fusion Expression and Biological Evaluation of Vasoactive Intestinal Peptide Analogue as Novel Antimicrobial Agent

Molecules ◽  
2017 ◽  
Vol 22 (11) ◽  
pp. 1963 ◽  
Author(s):  
Chunlan Xu ◽  
Yu Guo ◽  
Xiangjin Qiao ◽  
Xiaoya Shang ◽  
Weining Niu ◽  
...  
Keyword(s):  
Antimicrobial Agent ◽  
Vasoactive Intestinal Peptide ◽  
Biological Evaluation ◽  
Fusion Expression ◽  
Peptide Analogue

Mannich bases and novel benzothiazole derivatives of imidazo[2,1-b][1,3,4]thiadiazoles and their biological evaluation

2006 ◽  
Vol 27 (6) ◽  
pp. 553-569 ◽  
Author(s):  
Vinayak S. Hegde ◽  
Gundurao D. Kolavi ◽  
Ravi S. Lamani ◽  
Imtiyaz Ahmed M. Khazi
Keyword(s):  
Mannich Bases ◽  
Biological Evaluation ◽  
Benzothiazole Derivatives ◽  
Derivatives Of
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