New 3‐(1 H ‐benzo[ d ]imidazol‐2‐yl)quinolin‐2(1 H )‐one‐based triazole derivatives: Design, synthesis, and biological evaluation as antiproliferative and apoptosis‐inducing agents

2021 ◽  
Author(s):  
Nikhil B. Gaikwad ◽  
Sapana Bansode ◽  
Shankar Biradar ◽  
Mayuri Ban ◽  
Nanduri Srinivas ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Design Synthesis ◽  
Triazole Derivatives ◽  
Apoptosis Inducing Agents ◽  
Synthesis And Biological Evaluation

Design, Synthesis, and Biological Evaluation of New Indole-Acrylamide-1,2,3-Triazole Derivatives as Potential α-Glucosidase Inhibitors

2020 ◽  
pp. 1-9
Author(s):  
Seyed Esmaeil Sadat-Ebrahimi ◽  
Hiva Babania ◽  
Maryam Mohammadi-Khanaposhtani ◽  
Mohammad Sadegh Asgari ◽  
Somayeh Mojtabavi ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Design Synthesis ◽  
Triazole Derivatives ◽  
Glucosidase Inhibitors ◽  
Synthesis And Biological Evaluation

scholarly journals Design, synthesis and biological evaluation of tacrine-1,2,3-triazole derivatives as potent cholinesterase inhibitors

MedChemComm ◽  
2018 ◽  
Vol 9 (1) ◽  
pp. 149-159 ◽  
Author(s):  
Gaochan Wu ◽  
Yun Gao ◽  
Dongwei Kang ◽  
Boshi Huang ◽  
Zhipeng Huo ◽  
...  
Keyword(s):  
Cholinesterase Inhibitors ◽  
Biological Evaluation ◽  
Dipolar Cycloaddition ◽  
Design Synthesis ◽  
Triazole Derivatives ◽  
Design And Synthesis ◽  
Cuaac Reaction ◽  
Synthesis And Biological Evaluation

We report herein the design and synthesis of a series of 11 novel tacrine-1,2,3-triazole derivatives via a Cu(i)-catalyzed alkyne–azide 1,3-dipolar cycloaddition (CuAAC) reaction.

Design synthesis and biological evaluation of 3-substituted triazole derivatives

2011 ◽  
Vol 22 (5) ◽  
pp. 519-522 ◽  
Author(s):  
Bao Gang Wang ◽  
Shi Chong Yu ◽  
Xiao Yun Chai ◽  
Yong Zheng Yan ◽  
Hong Gang Hu ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Design Synthesis ◽  
Triazole Derivatives ◽  
Synthesis And Biological Evaluation

A library of 1,2,3-triazole-substituted oleanolic acid derivatives as anticancer agents: design, synthesis, and biological evaluation

2015 ◽  
Vol 13 (5) ◽  
pp. 1507-1514 ◽  
Author(s):  
Gaofei Wei ◽  
Weijing Luan ◽  
Shuai Wang ◽  
Shanshan Cui ◽  
Fengran Li ◽  
...  
Keyword(s):  
Oleanolic Acid ◽  
Anticancer Agents ◽  
Cycloaddition Reaction ◽  
Biological Evaluation ◽  
Dipolar Cycloaddition ◽  
Design Synthesis ◽  
Triazole Derivatives ◽  
Synthesis And Biological Evaluation

A series of novel oleanolic acid coupled 1,2,3-triazole derivatives have been designed and synthesized by employing a Cu(i) catalyzed Huisgen 1,3-dipolar cycloaddition reaction.

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