Equine metabolism of the selective androgen receptor modulator AC‐262536 in vitro and in urine, plasma and hair following oral administration

Identification of Selected in vitro-Generated Phase-I Metabolites of the Steroidal Selective Androgen Receptor Modulator MK-0773 for Doping Control Purposes

European Journal of Mass Spectrometry ◽

10.1255/ejms.1415 ◽

2016 ◽

Vol 22 (2) ◽

pp. 49-59 ◽

Cited By ~ 11

Author(s):

Andreas Lagojda ◽

Dirk Kuehne ◽

Oliver Krug ◽

Andreas Thomas ◽

Tina Wigger ◽

...

Keyword(s):

Androgen Receptor ◽

Phase I ◽

Doping Control ◽

Investigation of the metabolism of the selective androgen receptor modulator LGD‐4033 in equine urine, plasma and hair following oral administration

Drug Testing and Analysis ◽

10.1002/dta.2719 ◽

2020 ◽

Vol 12 (2) ◽

pp. 247-260 ◽

Cited By ~ 5

Author(s):

Charlotte Cutler ◽

Marjaana Viljanto ◽

Pamela Hincks ◽

Jocelyn Habershon‐Butcher ◽

Tessa Muir ◽

...

Keyword(s):

Androgen Receptor ◽

Oral Administration ◽

CHARACTERIZATION OF THE IN VITRO METABOLISM OF SELECTIVE ANDROGEN RECEPTOR MODULATOR USING HUMAN, RAT, AND DOG LIVER ENZYME PREPARATIONS

Drug Metabolism and Disposition ◽

10.1124/dmd.105.007112 ◽

2005 ◽

Vol 34 (2) ◽

pp. 243-253 ◽

Cited By ~ 25

Author(s):

Wenqing Gao ◽

Zengru Wu ◽

Casey E. Bohl ◽

Jun Yang ◽

Duane D. Miller ◽

...

Keyword(s):

Androgen Receptor ◽

Liver Enzyme ◽

In Vitro Metabolism ◽

Enzyme Preparations ◽

Receptor Modulator ◽

Dog Liver

Detection of the selective androgen receptor modulator GSK2881078 and metabolites in urine and hair after single oral administration

Drug Testing and Analysis ◽

10.1002/dta.2943 ◽

2020 ◽

Author(s):

Alina Rading ◽

Patricia Anielski ◽

Detlef Thieme ◽

Annekathrin Martina Keiler

Keyword(s):

Androgen Receptor ◽

Oral Administration ◽

Receptor Modulator ◽

Single Oral Administration

A selective androgen receptor modulator with minimal prostate hypertrophic activity enhances lean body mass in male rats and stimulates sexual behavior in female rats

Endocrine ◽

10.1007/s12020-007-9005-2 ◽

2007 ◽

Vol 32 (1) ◽

pp. 41-51 ◽

Cited By ~ 25

Author(s):

George F. Allan ◽

Pamela Tannenbaum ◽

Tifanie Sbriscia ◽

Olivia Linton ◽

Muh-Tsann Lai ◽

...

Keyword(s):

Sexual Behavior ◽

Androgen Receptor ◽

Lean Body Mass ◽

Body Mass ◽

Female Rats ◽

Male Rats ◽

Improving selective androgen receptor modulator discovery and preclinical evaluation

Expert Opinion on Drug Discovery ◽

10.1517/17460440903206957 ◽

2009 ◽

Vol 4 (9) ◽

pp. 981-993 ◽

Cited By ~ 9

Author(s):

Jeremy Orion Jones

Keyword(s):

Androgen Receptor ◽

Preclinical Evaluation ◽

Safety and Tolerability of LGD-4033, a Novel Non-Steroidal Oral Selective Androgen Receptor Modulator (SARM), in Healthy Men

10.1210/endo-meetings.2011.part3.p27.p3-207 ◽

2011 ◽

pp. P3-207-P3-207

Author(s):

Shehzad Basaria ◽

Lauren Collins ◽

Melinda Sheffield-Moore ◽

Edgar L Dillon ◽

Katie Orwoll ◽

...

Keyword(s):

Androgen Receptor ◽

Healthy Men ◽

Selective Androgen Receptor Modulator

Encyclopedia of Molecular Pharmacology ◽

10.1007/978-3-540-38918-7_6689 ◽

2008 ◽

pp. 1112-1112

Keyword(s):

Androgen Receptor ◽

Selective Androgen Receptor Modulator S42 Suppresses Prostate Cancer Cell Proliferation

Endocrinology ◽

10.1210/en.2018-00099 ◽

2018 ◽

Vol 159 (4) ◽

pp. 1774-1792 ◽

Cited By ~ 3

Author(s):

Takako Kawanami ◽

Tomoko Tanaka ◽

Yuriko Hamaguchi ◽

Takashi Nomiyama ◽

Hajime Nawata ◽

...

Keyword(s):

Prostate Cancer ◽

Cell Proliferation ◽

Androgen Receptor ◽

Cancer Cell ◽

Prostate Cancer Cell ◽

Cancer Cell Proliferation ◽

Pharmacokinetic drug interactions of the selective androgen receptor modulator GTx-024(Enobosarm) with itraconazole, rifampin, probenecid, celecoxib and rosuvastatin

Investigational New Drugs ◽

10.1007/s10637-016-0353-8 ◽

2016 ◽

Vol 34 (4) ◽

pp. 458-467 ◽

Cited By ~ 8

Author(s):

Christopher C. Coss ◽

Amanda Jones ◽

James T. Dalton

Keyword(s):

Androgen Receptor ◽

Drug Interactions ◽

Receptor Modulator ◽

Pharmacokinetic Drug