Synthesis and herbicidal activity of pyrimidyl‐1,2,4‐triazole derivatives containing aryl sulfonyl moiety

Author(s):  
Lingyun Yang ◽  
Yi Sun ◽  
Zhifeng Lu ◽  
Jingru Liang ◽  
Tao Wang ◽  
...  
1977 ◽  
Vol 8 (47) ◽  
pp. no-no
Author(s):  
V. MESSORI ◽  
L. BALDI ◽  
G. BIANCHETTI

2019 ◽  
Vol 56 (3) ◽  
pp. 968-971 ◽  
Author(s):  
Jin‐Xia Mu ◽  
Zhi‐Wen Zhai ◽  
Cheng‐Xia Tan ◽  
Jian‐Quan Weng ◽  
Hong‐Ke Wu ◽  
...  

2011 ◽  
Vol 4 (8) ◽  
pp. 685-688
Author(s):  
H.Ighachane H.Ighachane ◽  
◽  
H.El ayadi H.El ayadi ◽  
My.H.Sedra My.H.Sedra ◽  
H.B.Lazrek H.B.Lazrek

2001 ◽  
Vol 26 (4) ◽  
pp. 383-384 ◽  
Author(s):  
Akemi HOSOKAWA ◽  
Osamu IKEDA ◽  
Chizuko SASAKI ◽  
Yasuko T. OSANO ◽  
Tetsuo JIKIHARA

2018 ◽  
Author(s):  
Yiming Zhao ◽  
Huy van Nguyen ◽  
Louise Male ◽  
Philip Craven ◽  
Benjamin R. Buckley ◽  
...  

<div>Twelve 1,5-disubtituted and fourteen 5-substituted 1,2,3-triazole derivatives bearing diaryl or dialkyl phosphines at the 5-position were synthesised and used as ligands for palladium-catalysed Suzuki-Miyaura cross-coupling reactions. Bulky substrates were tested, and lead-like product formation was demonstrated. The online tool SambVca 2.0 was used to assess steric parameters of ligands and preliminary buried volume determination using XRD obtained data in a small number of cases proved to be informative. Two modelling approaches were compared for the determination of</div><div>the buried volume of ligands where XRD data was not available. An approach with imposed steric restrictions was found to be superior in leading to buried volume determinations that closely correlate with observed reaction conversions. The online tool LLAMA was used to determine lead-likeness of potential Suzuki-Miyaura cross-coupling products, from which ten of the most lead-like were successfully synthesised. Thus, confirming these readily accessible triazole-containing phosphines as highly suitable ligands for reaction screening and optimisation in drug discovery campaigns.</div>


HortScience ◽  
1998 ◽  
Vol 33 (3) ◽  
pp. 484e-485
Author(s):  
Patrick C. Wilson ◽  
Ted Whitwell ◽  
Steven J. Klaine

This research focuses on the potential use of Canna hybrida `King Humbert' for removing simazine from contaminated water generated at golf courses and ornamental nurseries. Because of simazine's herbicidal activity, it is important for levels in solution not to exceed plant tolerance levels. Tolerance levels for C. hybrida were determined by dosing plants for 7 d with 0, 0.01, 0.03, 0.1, 0.3, 1.0, or 3.0 mg simazine/L nutrient media. Measurements of 7-d fresh mass production and photosynthetic efficiency (Fv/Fm) were taken. Simazine uptake and distribution within the plant was determined by dosing plants with 2.03 mCi 14C-simazine (0.243 mg/L) for 1, 3, 5, or 7 d. Plant tissues were analyzed by combustion and liquid scintillation counting. Fresh mass production was reduced 66% and 78% for plants exposed to 1.0 and 3.0 mg/L, respectively. Likewise, photosynthetic efficiency was reduced to 66% and 40% of the controls at the same respective concentrations. Plant uptake of simazine accounted for 13%, 34%, 48%, and 65% of the original simazine in the dosing solution after 1-, 3-, 5-, and 7-d exposure, respectively. This simazine was distributed primarily between roots and leaves.


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