Microwave-assisted synthesis, molecular docking, and biological evaluation of 2-arylidene-2H-furo[2,3-f]chromen-3(7H)-ones as antioxidant and antimicrobial agents

2017 ◽  
Vol 26 (8) ◽  
pp. 1735-1746 ◽  
Author(s):  
Dongamanti Ashok ◽  
Kavitha Rangu ◽  
Srinivas Gundu ◽  
Arunapriya Lakkadi ◽  
Parthasarathy Tigulla
Keyword(s):  
Molecular Docking ◽  
Antimicrobial Agents ◽  
Biological Evaluation ◽  
Microwave Assisted Synthesis ◽  
Microwave Assisted

Thiazole fused thiosemicarbazones: Microwave-assisted synthesis, biological evaluation and molecular docking study

2019 ◽  
Vol 1179 ◽  
pp. 401-410 ◽  
Author(s):  
Neelam P. Prajapati ◽  
Kinjal D. Patel ◽  
Rajesh H. Vekariya ◽  
Hitesh D. Patel ◽  
Dhanaji P. Rajani
Keyword(s):  
Molecular Docking ◽  
Docking Study ◽  
Biological Evaluation ◽  
Microwave Assisted Synthesis ◽  
Molecular Docking Study ◽  
Microwave Assisted

scholarly journals Microwave-assisted synthesis, biological evaluation and molecular docking studies of new coumarin-based 1,2,3-triazoles

RSC Advances ◽  
2020 ◽  
Vol 10 (20) ◽  
pp. 11615-11623 ◽  
Author(s):  
Ravinder Dharavath ◽  
Nalaparaju Nagaraju ◽  
M. Ram Reddy ◽  
D. Ashok ◽  
M. Sarasija ◽  
...  
Keyword(s):  
Molecular Docking ◽  
Click Reaction ◽  
Docking Studies ◽  
Biological Evaluation ◽  
Microwave Assisted Synthesis ◽  
Terminal Alkynes ◽  
Triazole Derivatives ◽  
Molecular Docking Studies ◽  
Microwave Assisted ◽  
Highly Efficient

Coumarin-based 1,4-disubstituted 1,2,3-triazole derivatives were synthesized using a highly efficient, eco-friendly protocol via a copper(i)-catalyzed click reaction between various substituted arylazides and terminal alkynes.

Microwave assisted synthesis and biological evaluation of a series of 1,5-benzothiazepines as potential cytotoxic and antimicrobial agents

2014 ◽  
Vol 5 (1) ◽  
pp. 138-143 ◽  
Author(s):  
Subhash Yenupuri ◽  
Agastyaraju V. L. N. Satyanarayana Hariharan ◽  
Bharat Kumar Bugata ◽  
Divakara Laxman Somayajulu Nori
Keyword(s):  
Antimicrobial Agents ◽  
Biological Evaluation ◽  
Microwave Assisted Synthesis ◽  
Microwave Assisted ◽  
Synthesis And Biological Evaluation

Microwave assisted synthesis, biological evaluation, and molecular docking of novel chroman scaffolds incorporating spirochromanone framework

2016 ◽  
Vol 25 (12) ◽  
pp. 2882-2894 ◽  
Author(s):  
Dongamanti Ashok ◽  
Devulapally Mohan Gandhi ◽  
Aamate Vikas Kumar ◽  
Gundu Srinivas ◽  
Malladi Srinivas Reddy ◽  
...  
Keyword(s):  
Molecular Docking ◽  
Biological Evaluation ◽  
Microwave Assisted Synthesis ◽  
Microwave Assisted

4-Thiazolidinone derivatives as potent antimicrobial agents: microwave-assisted synthesis, biological evaluation and docking studies

MedChemComm ◽  
2015 ◽  
Vol 6 (2) ◽  
pp. 319-326 ◽  
Author(s):  
Eleni Pitta ◽  
Evangelia Tsolaki ◽  
Athina Geronikaki ◽  
Jovana Petrović ◽  
Jasmina Glamočlija ◽  
...  
Keyword(s):  
Reverse Transcriptase ◽  
Inhibitory Activity ◽  
Antimicrobial Agents ◽  
Docking Studies ◽  
Biological Evaluation ◽  
Microwave Assisted Synthesis ◽  
Microwave Assisted ◽  
Hiv 1

A series of ten thiazolidin-4-one derivatives was synthesized and evaluated for their antibacterial, antifungal and HIV-1 reverse transcriptase (RT) inhibitory activity.

Microwave assisted synthesis of novel Pyrazole derivatives and their biological evaluation as anti-bacterial agents

2020 ◽  
Vol 23 ◽  
Author(s):  
Hadis Khodadad ◽  
Farhad Hatamjafari ◽  
Khalil Pourshamsian ◽  
Babak Sadeghi
Keyword(s):  
Antibacterial Activity ◽  
Aromatic Aldehydes ◽  
Catalytic Amount ◽  
Antibacterial Activities ◽  
Structural Features ◽  
Biological Evaluation ◽  
Aureus Strain ◽  
Microwave Assisted Synthesis ◽  
Pyrazole Derivatives ◽  
Microwave Assisted

Aim and Objective: Microwave-assisted condensation of acetophenone 1 and aromatic aldehydes 2 gave chalcone analogs 3, which were cyclized to pyrazole derivatives 6a-f via the reaction with hydrazine hydrate and oxalic acid in the presence of the catalytic amount of acetic acid in ethanol. Materials and Methods: The structural features of the synthesized compounds were characterized by melting point, FT-IR, 1H, 13C NMR and elemental analysis. Results: The antibacterial activities of the synthesized pyrazoles was evaluated against three gram-positive bacteria such as Enterococcus durans, Staphylococcus aureus, Bacillus subtilis and two gram-negative bacteria such as Escherichia coli and Salmonella typhimurium. Conclusion: All the synthesized pyrazoles showed relatively high antibacterial activity against S. aureus strain and none of them demonstrated antibacterial activity against E. coli.

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