Characterization and development of a peptide substrate-based phosphate transfer assay for the human vascular endothelial growth factor receptor-2 tyrosine kinase

Genshi Zhao; Robert B. Peery; Jonathan M. Yingling

doi:10.1016/j.ab.2006.10.038

Characterization and development of a peptide substrate-based phosphate transfer assay for the human vascular endothelial growth factor receptor-2 tyrosine kinase

Analytical Biochemistry ◽

10.1016/j.ab.2006.10.038 ◽

2007 ◽

Vol 360 (2) ◽

pp. 196-206 ◽

Cited By ~ 4

Author(s):

Genshi Zhao ◽

Robert B. Peery ◽

Jonathan M. Yingling

Keyword(s):

Vascular Endothelial Growth Factor ◽

Growth Factor ◽

Tyrosine Kinase ◽

Growth Factor Receptor ◽

Vascular Endothelial ◽

Peptide Substrate ◽

Endothelial Growth Factor

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Treatment of Mid-Pregnant Mice with KRN633, an Inhibitor of Vascular Endothelial Growth Factor Receptor Tyrosine Kinase, Induces Abnormal Retinal Vascular Patterning in Their Newborn Pups

Birth Defects Research Part B Developmental and Reproductive Toxicology ◽

10.1002/bdrb.21112 ◽

2014 ◽

Vol 101 (4) ◽

pp. 293-299 ◽

Cited By ~ 4

Author(s):

Akane Morita ◽

Tsutomu Nakahara ◽

Naomichi Abe ◽

Yuki Kurauchi ◽

Asami Mori ◽

...

Keyword(s):

Vascular Endothelial Growth Factor ◽

Growth Factor ◽

Tyrosine Kinase ◽

Receptor Tyrosine Kinase ◽

Growth Factor Receptor ◽

Vascular Endothelial ◽

Vascular Patterning ◽

Pregnant Mice ◽

Endothelial Growth Factor

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Everolimus zur Behandlung des metastasierten Nierenzellkarzinoms nach Versagen der ersten VEGFr-TKI(Vascular Endothelial Growth Factor Receptor-Tyrosine Kinase Inhibitor)-Therapie: Ergebnisse einer Interimsanalyse einer nichtinterventionellen Studie

Karger Kompass Onkologie ◽

10.1159/000356898 ◽

2014 ◽

Vol 1 (1) ◽

pp. 28-29

Keyword(s):

Vascular Endothelial Growth Factor ◽

Growth Factor ◽

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitor ◽

Receptor Tyrosine Kinase ◽

Kinase Inhibitor ◽

Growth Factor Receptor ◽

Vascular Endothelial ◽

Receptor Tyrosine Kinase Inhibitor ◽

Endothelial Growth Factor

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The Tyrosine Kinase Inhibitor Cediranib Blocks Ligand-Induced Vascular Endothelial Growth Factor Receptor-3 Activity and Lymphangiogenesis

Cancer Research ◽

10.1158/0008-5472.can-07-5809 ◽

2008 ◽

Vol 68 (12) ◽

pp. 4754-4762 ◽

Cited By ~ 86

Author(s):

Caroline A. Heckman ◽

Tanja Holopainen ◽

Maria Wirzenius ◽

Salla Keskitalo ◽

Michael Jeltsch ◽

...

Keyword(s):

Vascular Endothelial Growth Factor ◽

Growth Factor ◽

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitor ◽

Kinase Inhibitor ◽

Growth Factor Receptor ◽

Vascular Endothelial ◽

Endothelial Growth Factor

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The role of vascular endothelial growth factor receptor 1 tyrosine kinase signaling in bleomycin-induced pulmonary fibrosis

Biomedicine & Pharmacotherapy ◽

10.1016/j.biopha.2019.109067 ◽

2019 ◽

Vol 117 ◽

pp. 109067 ◽

Cited By ~ 1

Author(s):

Hideki Amano ◽

Yoshio Mastui ◽

Yoshiya Ito ◽

Yusaku Shibata ◽

Tomohiro Betto ◽

...

Keyword(s):

Vascular Endothelial Growth Factor ◽

Growth Factor ◽

Pulmonary Fibrosis ◽

Tyrosine Kinase ◽

Growth Factor Receptor ◽

Vascular Endothelial ◽

Kinase Signaling ◽

Tyrosine Kinase Signaling ◽

Endothelial Growth Factor

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Evaluation of a Series of Naphthamides as Potent, Orally Active Vascular Endothelial Growth Factor Receptor-2 Tyrosine Kinase Inhibitors¶

Journal of Medicinal Chemistry ◽

10.1021/jm701098w ◽

2008 ◽

Vol 51 (6) ◽

pp. 1668-1680 ◽

Cited By ~ 22

Author(s):

Matthew M. Weiss ◽

Jean-Christophe Harmange ◽

Anthony J. Polverino ◽

David Bauer ◽

Loren Berry ◽

...

Keyword(s):

Vascular Endothelial Growth Factor ◽

Growth Factor ◽

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitors ◽

Kinase Inhibitors ◽

Growth Factor Receptor ◽

Vascular Endothelial ◽

Endothelial Growth Factor ◽

Orally Active

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PTK787/ZK222584, a tyrosine kinase inhibitor of vascular endothelial growth factor receptor, reduces uptake of the contrast agent GdDOTA by murine orthotopic B16/BL6 melanoma tumours and inhibits their growth in vivo

NMR in Biomedicine ◽

10.1002/nbm.961 ◽

2005 ◽

Vol 18 (5) ◽

pp. 308-321 ◽

Cited By ~ 44

Author(s):

Markus Rudin ◽

Paul M. J. McSheehy ◽

Peter R. Allegrini ◽

Martin Rausch ◽

Diana Baumann ◽

...

Keyword(s):

Vascular Endothelial Growth Factor ◽

Growth Factor ◽

Tyrosine Kinase ◽

Contrast Agent ◽

Tyrosine Kinase Inhibitor ◽

Kinase Inhibitor ◽

Growth Factor Receptor ◽

Vascular Endothelial ◽

Endothelial Growth Factor

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Hepatotoxicity of vascular endothelial growth factor receptor tyrosine kinase inhibitors: clinical practice and evidence

Drugs & Therapy Perspectives ◽

10.1007/s40267-017-0416-8 ◽

2017 ◽

Vol 33 (8) ◽

pp. 395-402

Author(s):

Bulent Cetin ◽

Irem Bilgetekin ◽

Mustafa Cengiz ◽

Ahmet Ozet

Keyword(s):

Vascular Endothelial Growth Factor ◽

Clinical Practice ◽

Growth Factor ◽

Tyrosine Kinase ◽

Receptor Tyrosine Kinase ◽

Kinase Inhibitors ◽

Growth Factor Receptor ◽

Vascular Endothelial ◽

Endothelial Growth Factor ◽

Receptor Tyrosine Kinase Inhibitors

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Inhibition of choroidal neovascularization by blocking vascular endothelial growth factor receptor tyrosine kinase

Japanese Journal of Ophthalmology ◽

10.1007/s10384-007-0506-6 ◽

2008 ◽

Vol 52 (2) ◽

pp. 91-98 ◽

Cited By ~ 25

Author(s):

Junko Kami ◽

Kimimasa Muranaka ◽

Yasuo Yanagi ◽

Ryo Obata ◽

Yasuhiro Tamaki ◽

...

Keyword(s):

Vascular Endothelial Growth Factor ◽

Growth Factor ◽

Tyrosine Kinase ◽

Choroidal Neovascularization ◽

Receptor Tyrosine Kinase ◽

Growth Factor Receptor ◽

Vascular Endothelial ◽

Endothelial Growth Factor

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Inhibition of Chronic and Acute Skin Inflammation by Treatment with a Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitor

American Journal Of Pathology ◽

10.2353/ajpath.2008.071074 ◽

2008 ◽

Vol 173 (1) ◽

pp. 265-277 ◽

Cited By ~ 59

Author(s):

Cornelia Halin ◽

Hermann Fahrngruber ◽

Josef G. Meingassner ◽

Guido Bold ◽

Amanda Littlewood-Evans ◽

...

Keyword(s):

Vascular Endothelial Growth Factor ◽

Growth Factor ◽

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitor ◽

Receptor Tyrosine Kinase ◽

Kinase Inhibitor ◽

Growth Factor Receptor ◽

Skin Inflammation ◽

Vascular Endothelial ◽

Endothelial Growth Factor

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Naphthamides as Novel and Potent Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitors: Design, Synthesis, and Evaluation¶

Journal of Medicinal Chemistry ◽

10.1021/jm701097z ◽

2008 ◽

Vol 51 (6) ◽

pp. 1649-1667 ◽

Cited By ~ 43

Author(s):

Jean-Christophe Harmange ◽

Matthew M. Weiss ◽

Julie Germain ◽

Anthony J. Polverino ◽

George Borg ◽

...

Keyword(s):

Vascular Endothelial Growth Factor ◽

Growth Factor ◽

Tyrosine Kinase ◽

Receptor Tyrosine Kinase ◽

Kinase Inhibitors ◽

Growth Factor Receptor ◽

Vascular Endothelial ◽

Design Synthesis ◽

Endothelial Growth Factor ◽

Receptor Tyrosine Kinase Inhibitors

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