Design, synthesis and biological evaluation of novel 2-methylpyrimidine-4-ylamine derivatives as inhibitors of Escherichia coli pyruvate dehydrogenase complex E1

2012 ◽  
Vol 20 (5) ◽  
pp. 1665-1670 ◽  
Author(s):  
Junbo He ◽  
Lingling Feng ◽  
Jing Li ◽  
Ruijuan Tao ◽  
Fang Wang ◽  
...  
RSC Advances ◽  
2016 ◽  
Vol 6 (6) ◽  
pp. 4310-4320 ◽  
Author(s):  
Haifeng He ◽  
Jiangtao Feng ◽  
Junbo He ◽  
Qin Xia ◽  
Yanliang Ren ◽  
...  

Optimal binding mode of novel E. coli PDHc E1 inhibitor 9d.


Biochemistry ◽  
2017 ◽  
Vol 56 (49) ◽  
pp. 6491-6502 ◽  
Author(s):  
Yuan Zhou ◽  
Jiangtao Feng ◽  
Hongwu He ◽  
Leifeng Hou ◽  
Wen Jiang ◽  
...  

Sign in / Sign up

Export Citation Format

Share Document