Solid-phase synthesis and thermal denaturation study of cyclic PNAs targeting the HIV-1 TAR RNA loop

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2007.07.030 ◽

2007 ◽

Vol 17 (21) ◽

pp. 6026-6030 ◽

Author(s):

Gregory Upert ◽

Mohamed Mehiri ◽

Audrey Di Giorgio ◽

Roger Condom ◽

Nadia Patino

Keyword(s):

Thermal Denaturation ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Phase Synthesis ◽

Thermal Denaturation Study ◽

Tar Rna ◽

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Solid Phase Synthesis of Novel Pyrrolidinedione Analogs as Potent HIV-1 Integrase Inhibitors

Journal of Combinatorial Chemistry ◽

10.1021/cc9001026 ◽

2010 ◽

Vol 12 (1) ◽

pp. 84-90 ◽

Author(s):

Annapurna Pendri ◽

Timothy L. Troyer ◽

Michael J. Sofia ◽

Michael A. Walker ◽

B. Narasimhulu Naidu ◽

...

Keyword(s):

Solid Phase Synthesis ◽

Solid Phase ◽

Integrase Inhibitors ◽

Phase Synthesis ◽

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Solid-Phase Synthesis, Thermal Denaturation Studies, Nuclease Resistance, and Cellular Uptake of (Oligodeoxyribonucleoside)methylborane Phosphine–DNA Chimeras

Journal of the American Chemical Society ◽

10.1021/ja201314q ◽

2011 ◽

Vol 133 (25) ◽

pp. 9844-9854 ◽

Author(s):

Heera Krishna ◽

Marvin H. Caruthers

Keyword(s):

Cellular Uptake ◽

Thermal Denaturation ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Phase Synthesis ◽

Nuclease Resistance

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ChemInform Abstract: A New Method for the Solid Phase Synthesis of Hydroxyethylamine Peptide Bond Isosters: Synthesis of an HIV-1 Protease Inhibitor and of a β-Casomorphin-5 Analogue.

10.1002/chin.199408279 ◽

2010 ◽

Vol 25 (8) ◽

pp. no-no

Author(s):

D. TOURWE ◽

J. PIRON ◽

P. DEFREYN ◽

G. VAN BINST

Keyword(s):

Protease Inhibitor ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Peptide Bond ◽

Phase Synthesis ◽

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Solid-Phase Synthesis of the Alkenyldiarylmethane (ADAM) Series of Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors

The Journal of Organic Chemistry ◽

10.1021/jo0100291 ◽

2001 ◽

Vol 66 (18) ◽

pp. 5958-5964 ◽

Author(s):

Guozhang Xu ◽

Tracy L. Loftus ◽

Heather Wargo ◽

Jim A. Turpin ◽

Robert W. Buckheit, ◽

...

Keyword(s):

Reverse Transcriptase ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Reverse Transcriptase Inhibitors ◽

Phase Synthesis ◽

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Diversity-oriented solid-phase synthesis and biological evaluation of oligonucleotide hairpins as HIV-1 RT RNase H inhibitors

Nucleic Acids Research ◽

10.1093/nar/gkh948 ◽

2004 ◽

Vol 32 (21) ◽

pp. 6164-6175 ◽

Author(s):

Rami N. Hannoush ◽

Kyung-Lyum Min ◽

Masad J. Damha

Keyword(s):

Solid Phase Synthesis ◽

Solid Phase ◽

Biological Evaluation ◽

Rnase H ◽

Phase Synthesis ◽

Synthesis And Biological Evaluation ◽

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Research on anti-HIV-1 agents. Part 2: Solid-phase synthesis, biological evaluation and molecular modeling studies of 2,5,6-trisubstituted-4(3H)-pyrimidinones targeting HIV-1 reverse transcriptase

Tetrahedron ◽

10.1016/s0040-4020(01)00815-8 ◽

2001 ◽

Vol 57 (39) ◽

pp. 8357-8367 ◽

Author(s):

Maurizio Botta ◽

Federico Corelli ◽

Giovanni Maga ◽

Fabrizio Manetti ◽

Michela Renzulli ◽

...

Keyword(s):

Molecular Modeling ◽

Reverse Transcriptase ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Biological Evaluation ◽

Phase Synthesis ◽

Modeling Studies ◽

Molecular Modeling Studies ◽

Anti Hiv ◽

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Solid-phase synthesis of 5′-O-β,γ-methylenetriphosphate derivatives of nucleosides and evaluation of their inhibitory activity against HIV-1 reverse transcriptase

Tetrahedron Letters ◽

10.1016/j.tetlet.2010.04.005 ◽

2010 ◽

Vol 51 (22) ◽

pp. 3010-3013 ◽

Author(s):

Yousef Ahmadibeni ◽

Chandravanu Dash ◽

Stuart F.J. Le Grice ◽

Keykavous Parang

Keyword(s):

Reverse Transcriptase ◽

Inhibitory Activity ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Phase Synthesis ◽

Derivatives Of ◽

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Solid-Phase synthesis of diamine and polyamine amino acid derivatives as HIV-1 tat-TAR binding inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/s0968-0896(02)00305-x ◽

2003 ◽

Vol 11 (1) ◽

pp. 87-94 ◽

Author(s):

G Jimenez Bueno ◽

T Klimkait ◽

I.H Gilbert ◽

C Simons

Keyword(s):

Solid Phase Synthesis ◽

Solid Phase ◽

Amino Acid Derivatives ◽

Phase Synthesis ◽

Hiv 1 ◽

Binding Inhibitors

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SOLID-PHASE SYNTHESIS OF A PEPTIDE COMPRISING THE 605-611 DISULFIDE LOOP OF GP41, TRANSMEMBRANE GLYCOPROTEIN OF HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 (HIV-1)

Organic Preparations and Procedures International ◽

10.1080/00304949509458472 ◽

1995 ◽

Vol 27 (3) ◽

pp. 375-377

Author(s):

G. G. Gevorkian ◽

M. Viveros ◽

F. Zamudio ◽

C. Larralde

Keyword(s):

Human Immunodeficiency Virus ◽

Human Immunodeficiency Virus Type ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Phase Synthesis ◽

Transmembrane Glycoprotein ◽

Immunodeficiency Virus ◽

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Solid-phase synthesis and evaluation of TAR RNA targeted β-carboline–nucleoside conjugates

Organic & Biomolecular Chemistry ◽

10.1039/b809598a ◽

2008 ◽

Vol 6 (20) ◽

pp. 3741 ◽

Author(s):

Peng Zhao ◽

Hong-Wei Jin ◽

Zhen-Jun Yang ◽

Liang-Ren Zhang ◽

Li-He Zhang

Keyword(s):

Solid Phase Synthesis ◽

Solid Phase ◽

Phase Synthesis ◽

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