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New small molecule inhibitors of histone methyl transferase DOT1L with a nitrile as a non-traditional replacement for heavy halogen atoms
Bioorganic & Medicinal Chemistry Letters
◽
10.1016/j.bmcl.2016.07.041
◽
2016
◽
Vol 26
(18)
◽
pp. 4518-4522
◽
Cited By ~ 8
Author(s):
Sophie S. Spurr
◽
Elliott D. Bayle
◽
Wenyu Yu
◽
Fengling Li
◽
Wolfram Tempel
◽
...
Keyword(s):
Small Molecule
◽
Small Molecule Inhibitors
◽
Methyl Transferase
◽
Halogen Atoms
◽
Histone Methyl Transferase
Download Full-text
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From molecular diagnostics to molecular targeted therapy with natural product small molecule inhibitors in oral squamous cell carcinoma
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◽
10.1055/s-2007-986722
◽
2007
◽
Vol 73
(09)
◽
Cited By ~ 1
Author(s):
VB Konkimalla
◽
VL Suhas
◽
NR Chandra
◽
E Gebhart
◽
T Efferth
Keyword(s):
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◽
Targeted Therapy
◽
Oral Squamous Cell Carcinoma
◽
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◽
Natural Product
◽
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◽
Small Molecule
◽
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◽
Molecular Targeted Therapy
◽
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Faculty Opinions recommendation of Nanomolar small molecule inhibitors for alphav(beta)6, alphav(beta)5, and alphav(beta)3 integrins.
Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature
◽
10.3410/f.1004750.54854
◽
2002
◽
Author(s):
Carol Otey
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Faculty Opinions recommendation of Identification of small molecule inhibitors of anthrax lethal factor.
Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature
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10.3410/f.1016978.201559
◽
2004
◽
Author(s):
Kristina Downing
Keyword(s):
Small Molecule
◽
Small Molecule Inhibitors
◽
Lethal Factor
◽
Anthrax Lethal Factor
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Faculty Opinions recommendation of Harnessing chaperones to generate small-molecule inhibitors of amyloid beta aggregation.
Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature
◽
10.3410/f.1017973.285766
◽
2005
◽
Author(s):
George Perry
Keyword(s):
Small Molecule
◽
Amyloid Beta
◽
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Faculty Opinions recommendation of High-affinity small molecule inhibitors of T cell costimulation: compounds for immunotherapy.
Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature
◽
10.3410/f.1023153.264839
◽
2005
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Author(s):
Robert Kelley
Keyword(s):
T Cell
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Small Molecule
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Small Molecule Inhibitors
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High Affinity
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Faculty Opinions recommendation of Novel small molecule inhibitors of 3-phosphoinositide-dependent kinase-1.
Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature
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10.3410/f.1024840.292879
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2005
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Author(s):
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Keyword(s):
Small Molecule
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Faculty Opinions recommendation of Identification of new small molecule inhibitors of cystic fibrosis transmembrane conductance regulator protein: in vitro and in vivo studies.
Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature
◽
10.3410/f.1069767.522696
◽
2007
◽
Author(s):
Kim Barrett
Keyword(s):
Cystic Fibrosis
◽
Small Molecule
◽
Small Molecule Inhibitors
◽
In Vivo Studies
◽
Transmembrane Conductance Regulator
◽
Transmembrane Conductance
◽
Regulator Protein
◽
Cystic Fibrosis Transmembrane
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Faculty Opinions recommendation of SIRT1 regulates the histone methyl-transferase SUV39H1 during heterochromatin formation.
Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature
◽
10.3410/f.1096033.552028
◽
2007
◽
Author(s):
Andrew D Sharrocks
Keyword(s):
Methyl Transferase
◽
Heterochromatin Formation
◽
Histone Methyl Transferase
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Faculty Opinions recommendation of Discovery and characterization of small molecule inhibitors of the BET family bromodomains.
Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature
◽
10.3410/f.13411091.14784061
◽
2011
◽
Author(s):
Martin Stahl
Keyword(s):
Small Molecule
◽
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Faculty Opinions recommendation of Rational design of small-molecule inhibitors of the LEDGF/p75-integrase interaction and HIV replication.
Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature
◽
10.3410/f.3462958.3157056
◽
2010
◽
Author(s):
Jim Maher
Keyword(s):
Small Molecule
◽
Rational Design
◽
Small Molecule Inhibitors
◽
Hiv Replication
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