Activation and Drug Design of a Muscarinic G-Protein Coupled Receptor

Biophysical Journal ◽

10.1016/j.bpj.2014.11.547 ◽

2015 ◽

Vol 108 (2) ◽

pp. 95a

Author(s):

Yinglong Miao ◽

J. Andrew McCammon

Keyword(s):

Drug Design ◽

G Protein ◽

G Protein Coupled Receptor ◽

G Protein Coupled

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Protein expression and purification of G-protein coupled receptor kinase 6 (GRK6), toward structure-based drug design and discovery for multiple myeloma

Protein Expression and Purification ◽

10.1016/j.pep.2021.105890 ◽

2021 ◽

pp. 105890

Author(s):

Tien L. Olson ◽

Shangji Zhang ◽

Dillon Labban ◽

Emily Kaschner ◽

Manuel Aceves ◽

...

Keyword(s):

Multiple Myeloma ◽

Drug Design ◽

Protein Expression ◽

G Protein ◽

Receptor Kinase ◽

Expression And Purification ◽

G Protein Coupled Receptor ◽

Structure Based Drug Design ◽

Protein Expression And Purification ◽

G Protein Coupled

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From G Protein-coupled Receptor Structure Resolution to Rational Drug Design

Journal of Biological Chemistry ◽

10.1074/jbc.r115.668251 ◽

2015 ◽

Vol 290 (32) ◽

pp. 19489-19495 ◽

Author(s):

Ali Jazayeri ◽

Joao M. Dias ◽

Fiona H. Marshall

Keyword(s):

Drug Design ◽

G Protein ◽

Rational Drug Design ◽

G Protein Coupled Receptor ◽

Receptor Structure ◽

Rational Drug ◽

G Protein Coupled

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Computational methods in drug design: Modeling G protein-coupled receptor monomers, dimers, and oligomers

The AAPS Journal ◽

10.1007/bf02854903 ◽

2006 ◽

Vol 8 (2) ◽

pp. E322-E336 ◽

Author(s):

Patricia H. Reggio

Keyword(s):

Drug Design ◽

G Protein ◽

Computational Methods ◽

G Protein Coupled Receptor ◽

G Protein Coupled

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Toward Deciphering the Code to Aminergic G Protein-Coupled Receptor Drug Design

Chemistry & Biology ◽

10.1016/j.chembiol.2008.03.004 ◽

2008 ◽

Vol 15 (4) ◽

pp. 343-353 ◽

Author(s):

Edwin S. Tan ◽

Eli S. Groban ◽

Matthew P. Jacobson ◽

Thomas S. Scanlan

Keyword(s):

Drug Design ◽

G Protein ◽

G Protein Coupled Receptor ◽

G Protein Coupled

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What is the potential of G protein-coupled receptor allosteric sites in drug design?

Future Medicinal Chemistry ◽

10.4155/fmc.14.32 ◽

2014 ◽

Vol 6 (7) ◽

pp. 729-732 ◽

Author(s):

Stephen L Garland

Keyword(s):

Drug Design ◽

G Protein ◽

G Protein Coupled Receptor ◽

Allosteric Sites ◽

G Protein Coupled

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Definition of the G Protein-Coupled Receptor Transmembrane Bundle Binding Pocket and Calculation of Receptor Similarities for Drug Design

Journal of Medicinal Chemistry ◽

10.1021/jm900319e ◽

2009 ◽

Vol 52 (14) ◽

pp. 4429-4442 ◽

Author(s):

David E. Gloriam ◽

Steven M. Foord ◽

Frank E. Blaney ◽

Stephen L. Garland

Keyword(s):

Drug Design ◽

G Protein ◽

Binding Pocket ◽

G Protein Coupled Receptor ◽

Definition Of ◽

G Protein Coupled

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Dynamics and flexibility of G-protein-coupled receptor conformations and their relevance to drug design

Drug Discovery Today ◽

10.1016/j.drudis.2010.08.018 ◽

2010 ◽

Vol 15 (21-22) ◽

pp. 951-957 ◽

Author(s):

Nagarajan Vaidehi

Keyword(s):

Drug Design ◽

G Protein ◽

G Protein Coupled Receptor ◽

G Protein Coupled

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Computational Methods in Drug Design: Modeling G Protein-Coupled Receptor Monomers, Dimers, and Oligomers

Drug Addiction ◽

10.1007/978-0-387-76678-2_3 ◽

2008 ◽

pp. 41-68

Author(s):

Patricia H. Reggio

Keyword(s):

Drug Design ◽

G Protein ◽

Computational Methods ◽

G Protein Coupled Receptor ◽

G Protein Coupled

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Author response for "Estrogen receptor alpha, g‐protein coupled receptor 1, and aromatase: developmental, sex, and region‐specific differences across the rat caudate‐putamen, nucleus accumbens core and shell"

10.1002/cne.24978/v4/response1 ◽

2020 ◽

Author(s):

Amanda A. Krentzel ◽

Jaime A. Willett ◽

Ashlyn G. Johnson ◽

John Meitzen

Keyword(s):

Estrogen Receptor ◽

Nucleus Accumbens ◽

G Protein ◽

Estrogen Receptor Alpha ◽

Author Response ◽

G Protein Coupled Receptor ◽

Nucleus Accumbens Core ◽

Caudate Putamen ◽

Receptor Alpha ◽

G Protein Coupled

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Author response for "Estrogen receptor alpha, g‐protein coupled receptor 1, and aromatase: developmental, sex, and region‐specific differences across the rat caudate‐putamen, nucleus accumbens core and shell"

10.1002/cne.24978/v3/response1 ◽

2020 ◽

Author(s):

Amanda A. Krentzel ◽

Jaime A. Willett ◽

Ashlyn G. Johnson ◽

John Meitzen

Keyword(s):

Estrogen Receptor ◽

Nucleus Accumbens ◽

G Protein ◽

Estrogen Receptor Alpha ◽

Author Response ◽

G Protein Coupled Receptor ◽

Nucleus Accumbens Core ◽

Caudate Putamen ◽

Receptor Alpha ◽

G Protein Coupled

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