Structure-Activity Relationship and Characterization of Novel Influenza Inhibitors

Biophysical Journal ◽

10.1016/j.bpj.2017.11.2322 ◽

2018 ◽

Vol 114 (3) ◽

pp. 419a

Author(s):

Gregory Mohl ◽

Nathan Liddle ◽

David Michaelis ◽

David Busath

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity

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Microscale characterization of the structure–activity relationship of a heparin-binding glycopeptide using affinity capillary electrophoresis and immobilized enzymes

Journal of Chromatography A ◽

10.1016/s0021-9673(99)00452-5 ◽

1999 ◽

Vol 853 (1-2) ◽

pp. 189-195 ◽

Author(s):

Niels H.H Heegaard

Keyword(s):

Capillary Electrophoresis ◽

Immobilized Enzymes ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Heparin Binding ◽

Affinity Capillary Electrophoresis ◽

Structure Activity ◽

Relationship Of

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nSynthesis and characterization of 1-amidino-O-alkylureas metal complexes as α- glucosidase Inhibitors: Structure-activity relationship, molecular docking, and kinetic studies

Journal of Molecular Structure ◽

10.1016/j.molstruc.2021.131726 ◽

2021 ◽

pp. 131726

Author(s):

Firouz Matloubi Moghaddam ◽

Maryam Daneshfar ◽

Zahra Daneshfar ◽

Aida Iraji ◽

Atefe Samandari-Najafabad ◽

...

Keyword(s):

Molecular Docking ◽

Metal Complexes ◽

Kinetic Studies ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity ◽

Glucosidase Inhibitors

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Characterization of the Human and Mouse Sphingosine 1-Phosphate Receptor, S1P5(Edg-8): Structure−Activity Relationship of Sphingosine1-Phosphate Receptors†

Biochemistry ◽

10.1021/bi011606i ◽

2001 ◽

Vol 40 (46) ◽

pp. 14053-14060 ◽

Author(s):

Dong-Soon Im ◽

Jeremy Clemens ◽

Timothy L. Macdonald ◽

Kevin R. Lynch

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity ◽

Sphingosine 1 Phosphate ◽

Relationship Of ◽

Human And Mouse

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Synthesis and Characterization of Neurotensin Analogues for Structure/Activity Relationship Studies. Acetyl-neurotensin-(8-13) Is the Shortest Analogue with Full Binding and Pharmacological Activities

European Journal of Biochemistry ◽

10.1111/j.1432-1033.1982.tb05913.x ◽

1982 ◽

Vol 124 (1) ◽

pp. 117-125 ◽

Author(s):

Claude GRANIER ◽

Jurphaas RIETSCHOTEN ◽

Patrick KITABGI ◽

Claudine POUSTIS ◽

Pierre FREYCHET

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Synthesis And Characterization ◽

Pharmacological Activities ◽

Structure Activity ◽

Neurotensin Analogues

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Design, Structure–Activity Relationship, and in Vivo Characterization of the Development Candidate NVP-HSP990

Journal of Medicinal Chemistry ◽

10.1021/jm501107q ◽

2014 ◽

Vol 57 (21) ◽

pp. 9124-9129 ◽

Author(s):

Christopher M. McBride ◽

Barry Levine ◽

Yi Xia ◽

Cornelia Bellamacina ◽

Timothy Machajewski ◽

...

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity ◽

Design Structure ◽

In Vivo Characterization

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Structure-Activity Relationship of Toxic-Shock-Syndrome Toxin-1: Derivation and Characterization of Immunologically and Biologically Active Fragments

The Journal of Infectious Diseases ◽

10.1093/infdis/158.6.1287 ◽

1988 ◽

Vol 158 (6) ◽

pp. 1287-1295 ◽

Author(s):

C. Edwin ◽

J. Parsonnet ◽

E. H. Kass

Keyword(s):

Toxic Shock Syndrome ◽

Structure Activity Relationship ◽

Biologically Active ◽

Activity Relationship ◽

Toxic Shock ◽

Structure Activity ◽

Toxic Shock Syndrome Toxin ◽

Active Fragments ◽

Relationship Of

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Further characterization of β3-adrenoceptors in the guinea pig gastric fundus: stereoselectivity, β-adrenoceptor alkylation, and structure-activity relationship

Canadian Journal of Physiology and Pharmacology ◽

10.1139/cjpp-79-12-985 ◽

2001 ◽

Vol 79 (12) ◽

pp. 985-995 ◽

Author(s):

Takahiro Horinouchi ◽

Katsuo Koike

Keyword(s):

Structure Activity Relationship ◽

Gastric Fundus ◽

Activity Relationship ◽

Structure Activity

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Characterization of antioxidant, α-glucosidase and tyrosinase inhibitors from the rhizomes of Potentilla anserina L. and their structure–activity relationship

Food Chemistry ◽

10.1016/j.foodchem.2020.127714 ◽

2021 ◽

Vol 336 ◽

pp. 127714 ◽

Author(s):

Dan Yang ◽

Lei Wang ◽

Jianxiu Zhai ◽

Na Han ◽

Zhihui Liu ◽

...

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity ◽

Potentilla Anserina ◽

Tyrosinase Inhibitors

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Synthesis and characterization of photoaffinity labelling reagents towards the Hsp90 C-terminal domain

Organic & Biomolecular Chemistry ◽

10.1039/c6ob02097f ◽

2017 ◽

Vol 15 (7) ◽

pp. 1597-1605 ◽

Author(s):

Binto Simon ◽

Xuexia Huang ◽

Huangxian Ju ◽

Guoxuan Sun ◽

Min Yang

Keyword(s):

Binding Pocket ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Synthesis And Characterization ◽

Photoaffinity Labelling ◽

Terminal Domain ◽

Structure Activity

The synthesis of diazirine type photoaffinity labelling reagents to probe the Hsp90 C-terminal domain binding pocket and the structure–activity relationship. The structure illustrates probe positions only.

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Structure-activity relationship studies and pharmacological characterization of N5-heteroarylalkyl-substituted-2-(2-furanyl)thiazolo[5,4-d]pyrimidine-5,7-diamine-based derivatives as inverse agonists at human A2A adenosine receptor

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2018.06.020 ◽

2018 ◽

Vol 155 ◽

pp. 552-561 ◽

Author(s):

Flavia Varano ◽

Daniela Catarzi ◽

Fabrizio Vincenzi ◽

Matteo Falsini ◽

Silvia Pasquini ◽

...

Keyword(s):

Adenosine Receptor ◽

Structure Activity Relationship ◽

Activity Relationship ◽

A2a Adenosine Receptor ◽

Pharmacological Characterization ◽

Inverse Agonists ◽

Structure Activity

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