Design, synthesis and biological activity of novel substituted pyrazole amide derivatives targeting EcR/USP receptor

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Jin Xie ◽  
Yong-Qiang Li ◽  
De-Kai Yuan ◽  
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Liming Hu ◽  
Zhipeng Li ◽  
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MedChemComm ◽  
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The design, synthesis, characterization and biological evaluation of new ferrocenyl and ruthenocenyl derivatives of the antimalarial mefloquine is described.


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