Synthesis, biological evaluation and structure–activity relationship of new GABA uptake inhibitors, derivatives of 4-aminobutanamides

2014 ◽  
Vol 83 ◽  
pp. 256-273 ◽  
Author(s):  
Paula Kowalczyk ◽  
Kinga Sałat ◽  
Georg C. Höfner ◽  
Marta Mucha ◽  
Anna Rapacz ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Activity Relationship ◽  
Gaba Uptake ◽  
Structure Activity ◽  
Uptake Inhibitors ◽  
Relationship Of ◽  
Derivatives Of ◽  
Gaba Uptake Inhibitors

Structure activity relationship of selective GABA uptake inhibitors

2015 ◽  
Vol 23 (10) ◽  
pp. 2480-2488 ◽  
Author(s):  
Stine B. Vogensen ◽  
Lars Jørgensen ◽  
Karsten K. Madsen ◽  
Andreas Jurik ◽  
Nrupa Borkar ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Gaba Uptake ◽  
Structure Activity ◽  
Uptake Inhibitors ◽  
Relationship Of ◽  
Gaba Uptake Inhibitors

scholarly journals Synthesis, Biological Evaluation, and Structure-activity Relationship of Clonazepam, Meclonazepam, and 1,4-Benzodiazepine Compounds with Schistosomicidal Activity

2012 ◽  
Vol 79 (6) ◽  
pp. 943-949 ◽  
Author(s):  
Carla M. S. Menezes ◽  
Gildardo Rivera ◽  
Marina A. Alves ◽  
Daniel N. do Amaral ◽  
Jean Pierre B. Thibaut ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of

scholarly journals From in vitro to in cellulo: structure–activity relationship of (2-nitrophenyl)methanol derivatives as inhibitors of PqsD in Pseudomonas aeruginosa

2014 ◽  
Vol 12 (32) ◽  
pp. 6094-6104 ◽  
Author(s):  
Michael P. Storz ◽  
Giuseppe Allegretta ◽  
Benjamin Kirsch ◽  
Martin Empting ◽  
Rolf W. Hartmann
Keyword(s):  
Pseudomonas Aeruginosa ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Relationship Of ◽  
Derivatives Of

More than 60 derivatives of (2-nitrophenyl)methanol were synthesized and evaluated regarding their potency to inhibit PqsD. In vitro and in cellulo structure–activity relationships were derived.

Structure–activity relationship of boronic acid derivatives of tyropeptin: Proteasome inhibitors

2010 ◽  
Vol 20 (19) ◽  
pp. 5839-5842 ◽  
Author(s):  
Takumi Watanabe ◽  
Hikaru Abe ◽  
Isao Momose ◽  
Yoshikazu Takahashi ◽  
Daishiro Ikeda ◽  
...  
Keyword(s):  
Boronic Acid ◽  
Proteasome Inhibitors ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity ◽  
Boronic Acid Derivatives ◽  
Relationship Of ◽  
Derivatives Of

Synthesis, biological evaluation and structure–activity relationship of 2-styrylquinazolones as anti-tubercular agents

2016 ◽  
Vol 26 (11) ◽  
pp. 2663-2669 ◽  
Author(s):  
Pradeep S. Jadhavar ◽  
Tejas M. Dhameliya ◽  
Maulikkumar D. Vaja ◽  
Dinesh Kumar ◽  
Jonnalagadda Padma Sridevi ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of
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