Structure–activity relationship of boronic acid derivatives of tyropeptin: Proteasome inhibitors

2010 ◽  
Vol 20 (19) ◽  
pp. 5839-5842 ◽  
Author(s):  
Takumi Watanabe ◽  
Hikaru Abe ◽  
Isao Momose ◽  
Yoshikazu Takahashi ◽  
Daishiro Ikeda ◽  
...  
Keyword(s):  
Boronic Acid ◽  
Proteasome Inhibitors ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity ◽  
Boronic Acid Derivatives ◽  
Relationship Of ◽  
Derivatives Of

scholarly journals From in vitro to in cellulo: structure–activity relationship of (2-nitrophenyl)methanol derivatives as inhibitors of PqsD in Pseudomonas aeruginosa

2014 ◽  
Vol 12 (32) ◽  
pp. 6094-6104 ◽  
Author(s):  
Michael P. Storz ◽  
Giuseppe Allegretta ◽  
Benjamin Kirsch ◽  
Martin Empting ◽  
Rolf W. Hartmann
Keyword(s):  
Pseudomonas Aeruginosa ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Relationship Of ◽  
Derivatives Of

More than 60 derivatives of (2-nitrophenyl)methanol were synthesized and evaluated regarding their potency to inhibit PqsD. In vitro and in cellulo structure–activity relationships were derived.

scholarly journals An Overview of Bioactive Alkaloid, Semi-Synthetic Analogs, Mechanism of Action and Structure-Activity Relationship of Piperine as Antioxidant

2021 ◽  
Vol 33 (9) ◽  
pp. 2244-2250
Author(s):  
Sagar Joshi ◽  
Salahuddin ◽  
Rajnish Kumar ◽  
Divya Sharma
Keyword(s):  
Antioxidant Activity ◽  
Mechanism Of Action ◽  
Structure Activity Relationship ◽  
Black Pepper ◽  
Activity Relationship ◽  
Pharmacological Activities ◽  
Structure Activity ◽  
Natural Alkaloid ◽  
Relationship Of ◽  
Derivatives Of

Piperine, a natural alkaloid obtained from black pepper exhibit a variety of pharmacological activities like antioxidant activity and in this article, the mechanism of the antioxidant, structure-activity relationship of piperine as an antioxidant and various schemes of derivatives of piperine as antioxidants were discussed.

Synthesis and structure–activity relationship of amidine derivatives of 3,4-ethylenedioxythiophene as novel antibacterial agents

2015 ◽  
Vol 90 ◽  
pp. 68-81 ◽  
Author(s):  
Ivana Stolić ◽  
Hana Čipčić Paljetak ◽  
Mihaela Perić ◽  
Mario Matijašić ◽  
Višnja Stepanić ◽  
...  
Keyword(s):  
Antibacterial Agents ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of ◽  
Derivatives Of
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