Synthesis, biological evaluation and structure–activity relationship of 2-styrylquinazolones as anti-tubercular agents

2016 ◽  
Vol 26 (11) ◽  
pp. 2663-2669 ◽  
Author(s):  
Pradeep S. Jadhavar ◽  
Tejas M. Dhameliya ◽  
Maulikkumar D. Vaja ◽  
Dinesh Kumar ◽  
Jonnalagadda Padma Sridevi ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of

scholarly journals Synthesis, Biological Evaluation, and Structure-activity Relationship of Clonazepam, Meclonazepam, and 1,4-Benzodiazepine Compounds with Schistosomicidal Activity

2012 ◽  
Vol 79 (6) ◽  
pp. 943-949 ◽  
Author(s):  
Carla M. S. Menezes ◽  
Gildardo Rivera ◽  
Marina A. Alves ◽  
Daniel N. do Amaral ◽  
Jean Pierre B. Thibaut ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of

In vitro biological evaluation and consideration about structure-activity relationship of silver(I) aminoacidate complexes

2020 ◽  
Vol 210 ◽  
pp. 111170
Author(s):  
Gabriela Kuzderová ◽  
Michaela Rendošová ◽  
Róbert Gyepes ◽  
Miroslav Almáši ◽  
Danica Sabolová ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of

Synthesis and Antineoplastic Activity of Quinoline Derivatives

2008 ◽  
Vol 61 (7) ◽  
pp. 531 ◽  
Author(s):  
Qiang Zhou ◽  
Jing Hou ◽  
Huamin Li ◽  
Li Cui ◽  
Han Jia ◽  
...  
Keyword(s):  
Cytotoxic Activity ◽  
Cell Lines ◽  
Cancer Cell ◽  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Antineoplastic Activity ◽  
Activity Relationship ◽  
Quinoline Derivatives ◽  
Structure Activity ◽  
Relationship Of

Designed as a new series of molecules that contain the quinoline substructure, several 11H-indolo[3.2-c]quinoline derivatives were synthesized and subjected to biological evaluation. Several compounds were found to exhibit cytotoxic activity against the growth of colon (HTC-8), liver (BEL-7402), gastric (BCG-823), pulmonary gland (A549), and ovary (A2780) cancer cell lines. The structure–activity relationship of these compounds is discussed.

scholarly journals The synthesis, biological evaluation and structure–activity relationship of 2-phenylaminomethylene-cyclohexane-1,3-diones as specific anti-tuberculosis agents

MedChemComm ◽  
2017 ◽  
Vol 8 (11) ◽  
pp. 2133-2141 ◽  
Author(s):  
Muzafar Ahmad Rather ◽  
Ali Mohd Lone ◽  
Bisma Teli ◽  
Zubair Shanib Bhat ◽  
Paramjeet Singh ◽  
...  
Keyword(s):  
Mycobacterium Tuberculosis ◽  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of

Synthetic interventions on previously identified hits; structure39was identified as the best lead againstMycobacterium tuberculosisH37Rv and was evaluated further.

scholarly journals Discovery, Biological Evaluation, and Structure−Activity Relationship of Amidine Based Sphingosine Kinase Inhibitors

2010 ◽  
Vol 53 (7) ◽  
pp. 2766-2778 ◽  
Author(s):  
Thomas P. Mathews ◽  
Andrew J. Kennedy ◽  
Yugesh Kharel ◽  
Perry C. Kennedy ◽  
Oana Nicoara ◽  
...  
Keyword(s):  
Kinase Inhibitors ◽  
Sphingosine Kinase ◽  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of

scholarly journals Biological evaluation and structure activity relationship of 9-methyl-1-phenyl-9H-pyrido[3,4-b]indole derivatives as anti-leishmanial agents

2019 ◽  
Vol 84 ◽  
pp. 98-105 ◽  
Author(s):  
Penta Ashok ◽  
Subhash Chander ◽  
Terry K. Smith ◽  
Rajnish Prakash Singh ◽  
Prabhat Nath Jha ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Activity Relationship ◽  
Indole Derivatives ◽  
Structure Activity ◽  
Relationship Of
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