Eosinophils adhesion assay as a tool for phenotypic drug screening - The pharmacology of 1,3,5 – Triazine and 1H-indole like derivatives against the human histamine H4 receptor

2021 ◽  
Vol 890 ◽  
pp. 173611
Author(s):  
Marek Grosicki ◽  
Maristella Adami ◽  
Cristina Micheloni ◽  
Monika Głuch-Lutwin ◽  
Agata Siwek ◽  
...  
Keyword(s):  
Drug Screening ◽  
Adhesion Assay ◽  
Histamine H4 Receptor ◽  
H4 Receptor ◽  
Human Histamine

Discovery of Novel Human Histamine H4 Receptor Ligands by Large-Scale Structure-Based Virtual Screening

2008 ◽  
Vol 51 (11) ◽  
pp. 3145-3153 ◽  
Author(s):  
Róbert Kiss ◽  
Béla Kiss ◽  
Árpád Könczöl ◽  
Ferenc Szalai ◽  
Ivett Jelinek ◽  
...  
Keyword(s):  
Virtual Screening ◽  
Large Scale ◽  
Large Scale Structure ◽  
Scale Structure ◽  
Receptor Ligands ◽  
Histamine H4 Receptor ◽  
H4 Receptor ◽  
Human Histamine

Binding mode analysis and enrichment studies on homology models of the human histamine H4 receptor

2008 ◽  
Vol 43 (5) ◽  
pp. 1059-1070 ◽  
Author(s):  
Róbert Kiss ◽  
Béla Noszál ◽  
Ákos Rácz ◽  
András Falus ◽  
Dániel Erős ◽  
...  
Keyword(s):  
Binding Mode ◽  
Mode Analysis ◽  
Histamine H4 Receptor ◽  
H4 Receptor ◽  
Human Histamine ◽  
Homology Models

In Silico Characterization of Ligand Binding Modes in the Human Histamine H4 Receptor and their Impact on Receptor Activation

ChemBioChem ◽  
2010 ◽  
Vol 11 (13) ◽  
pp. 1850-1855 ◽  
Author(s):  
Tim Werner ◽  
Kerstin Sander ◽  
Yusuf Tanrikulu ◽  
Tim Kottke ◽  
Ewgenij Proschak ◽  
...  
Keyword(s):  
Ligand Binding ◽  
In Silico ◽  
Receptor Activation ◽  
Binding Modes ◽  
Histamine H4 Receptor ◽  
H4 Receptor ◽  
In Silico Characterization ◽  
Human Histamine

Genetic variations within the promotor region of the human histamine H4 receptor gene in psoriasis patients

2016 ◽  
Vol 114 ◽  
pp. 121-127 ◽  
Author(s):  
Susanne Mommert ◽  
Lisanne Ratz ◽  
Kira Herwig ◽  
Maren Rost ◽  
Ralf Gutzmer ◽  
...  
Keyword(s):  
Receptor Gene ◽  
Genetic Variations ◽  
Histamine H4 Receptor ◽  
Promotor Region ◽  
H4 Receptor ◽  
Human Histamine

Identification of 2-arylbenzimidazoles as potent human histamine H4 receptor ligands

2006 ◽  
Vol 16 (23) ◽  
pp. 6043-6048 ◽  
Author(s):  
Alice Lee-Dutra ◽  
Kristen L. Arienti ◽  
Daniel J. Buzard ◽  
Michael D. Hack ◽  
Haripada Khatuya ◽  
...  
Keyword(s):  
Receptor Ligands ◽  
Histamine H4 Receptor ◽  
H4 Receptor ◽  
Human Histamine

Electrophysiology-based analysis of human histamine H4 receptor pharmacology using GIRK channel coupling in Xenopus oocytes

2008 ◽  
Vol 591 (1-3) ◽  
pp. 52-58 ◽  
Author(s):  
Kristoffer Sahlholm ◽  
Johanna Nilsson ◽  
Daniel Marcellino ◽  
Kjell Fuxe ◽  
Peter Århem
Keyword(s):  
Xenopus Oocytes ◽  
Channel Coupling ◽  
Histamine H4 Receptor ◽  
Girk Channel ◽  
Receptor Pharmacology ◽  
H4 Receptor ◽  
Human Histamine
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