Design, synthesis, and biological evaluation of fluoronitrophenyl substituted folate analogues as potential inhibitors of GAR transformylase and AICAR transformylase

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(00)00271-7 ◽

2000 ◽

Vol 10 (13) ◽

pp. 1471-1475 ◽

Author(s):

Dale L. Boger ◽

Thomas H. Marsilje ◽

René A. Castro ◽

Michael P. Hedrick ◽

Qing Jin ◽

...

Keyword(s):

Biological Evaluation ◽

Design Synthesis ◽

Potential Inhibitors ◽

Synthesis And Biological Evaluation

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Design, synthesis, and biological evaluation of pyrimidine derivatives as potential inhibitors of human calcium/calmodulin-dependent protein kinase IV

Chemical Biology & Drug Design ◽

10.1111/cbdd.12898 ◽

2016 ◽

Vol 89 (5) ◽

pp. 741-754 ◽

Author(s):

Ehtesham Jameel ◽

Huma Naz ◽

Parvez Khan ◽

Mohd. Tarique ◽

Jitendra Kumar ◽

...

Keyword(s):

Protein Kinase ◽

Biological Evaluation ◽

Pyrimidine Derivatives ◽

Dependent Protein Kinase ◽

Design Synthesis ◽

Calcium Calmodulin Dependent ◽

Dependent Protein ◽

Potential Inhibitors ◽

Synthesis And Biological Evaluation

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Rational design, synthesis, and biological evaluation of rigid pyrrolidone analogues as potential inhibitors of prostate cancer cell growth

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(01)00097-x ◽

2001 ◽

Vol 11 (8) ◽

pp. 955-959 ◽

Author(s):

Lixin Qiao ◽

Lian-Yun Zhao ◽

Suo-Bao Rong ◽

Xiong-Wu Wu ◽

Shaomeng Wang ◽

...

Keyword(s):

Prostate Cancer ◽

Cell Growth ◽

Cancer Cell ◽

Rational Design ◽

Prostate Cancer Cell ◽

Biological Evaluation ◽

Cancer Cell Growth ◽

Design Synthesis ◽

Potential Inhibitors ◽

Synthesis And Biological Evaluation

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Design, Synthesis and Biological Evaluation of Substituted Guanidine Indole Derivatives as Potential Inhibitors of HIV-1 Tat-TAR Interaction

Medicinal Chemistry ◽

10.2174/1573406410666140306151815 ◽

2013 ◽

Vol 10 (7) ◽

pp. 738-746 ◽

Author(s):

Jun Wang ◽

Yan Wang ◽

Zhenyu Li ◽

Peng Zhan ◽

Rujun Bai ◽

...

Keyword(s):

Biological Evaluation ◽

Indole Derivatives ◽

Design Synthesis ◽

Potential Inhibitors ◽

Synthesis And Biological Evaluation ◽

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ChemInform Abstract: Rational Design, Synthesis, and Biological Evaluation of Rigid Pyrrolidone Analogues as Potential Inhibitors of Prostate Cancer Cell Growth.

10.1002/chin.200132119 ◽

2010 ◽

Vol 32 (32) ◽

pp. no-no

Author(s):

Alan P. Kozikowski ◽

et al. et al.

Keyword(s):

Prostate Cancer ◽

Cell Growth ◽

Cancer Cell ◽

Rational Design ◽

Prostate Cancer Cell ◽

Biological Evaluation ◽

Cancer Cell Growth ◽

Design Synthesis ◽

Potential Inhibitors ◽

Synthesis And Biological Evaluation

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Design, synthesis and biological evaluation of novel 2-(5-aryl-1H-imidazol-1-yl) derivatives as potential inhibitors of the HIV-1 Vpu and host BST-2 protein interaction

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2020.112111 ◽

2020 ◽

Vol 190 ◽

pp. 112111 ◽

Author(s):

Thompho J. Rashamuse ◽

Zikhona Njengele ◽

E. Mabel Coyanis ◽

Yasien Sayed ◽

Salerwe Mosebi ◽

...

Keyword(s):

Protein Interaction ◽

Biological Evaluation ◽

Design Synthesis ◽

Potential Inhibitors ◽

Synthesis And Biological Evaluation ◽

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Design, synthesis and biological evaluation of novel bouchardatine analogs as potential inhibitors of adipogenesis/lipogenesis in 3T3-L1 adipocytes

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2018.01.089 ◽

2018 ◽

Vol 147 ◽

pp. 90-101 ◽

Author(s):

Lin Gao ◽

Zhao Xu ◽

Yong Rao ◽

Yu-Ting Lu ◽

Yu-Tao Hu ◽

...

Keyword(s):

Biological Evaluation ◽

Design Synthesis ◽

Potential Inhibitors ◽

Synthesis And Biological Evaluation

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1,3,4-Oxadiazoline derivatives as novel potential inhibitors targeting chitin biosynthesis: Design, synthesis and biological evaluation

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2008.11.095 ◽

2009 ◽

Vol 19 (2) ◽

pp. 332-335 ◽

Author(s):

Shaoyong Ke ◽

Fengyi Liu ◽

Ni Wang ◽

Qing Yang ◽

Xuhong Qian

Keyword(s):

Biological Evaluation ◽

Design Synthesis ◽

Potential Inhibitors ◽

Synthesis And Biological Evaluation

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Design, synthesis, and biological evaluation of simplified α-Keto heterocycle, trifluoromethyl ketone, and formyl substituted folate analogues as potential inhibitors of GAR transformylase and AICAR transformylase

Bioorganic & Medicinal Chemistry ◽

10.1016/s0968-0896(03)00456-5 ◽

2003 ◽

Vol 11 (20) ◽

pp. 4487-4501 ◽

Author(s):

Thomas H Marsilje ◽

Michael P Hedrick ◽

Joel Desharnais ◽

Ali Tavassoli ◽

Yan Zhang ◽

...

Keyword(s):

Biological Evaluation ◽

Design Synthesis ◽

Potential Inhibitors ◽

Synthesis And Biological Evaluation

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Design, synthesis and biological evaluation of novel carbamates as potential inhibitors of acetylcholinesterase and butyrylcholinesterase

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2020.115324 ◽

2020 ◽

Vol 28 (5) ◽

pp. 115324 ◽

Author(s):

Jie Wu ◽

Marco Pistolozzi ◽

Siyu Liu ◽

Wen Tan

Keyword(s):

Biological Evaluation ◽

Design Synthesis ◽

Potential Inhibitors ◽

Synthesis And Biological Evaluation

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Design, Synthesis and Biological Evaluation of some Chalcone Derivatives as Potential Pancreatic Lipase Inhibitors

10.3390/ecsoc-17-b024 ◽

2013 ◽

Author(s):

Dao Tran

Keyword(s):

Pancreatic Lipase ◽

Biological Evaluation ◽

Design Synthesis ◽

Chalcone Derivatives ◽

Pancreatic Lipase Inhibitors ◽

Synthesis And Biological Evaluation

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