A high‐throughput fluorescence polarization assay for the determination of Kd for soluble epoxide hydrolase inhibitors

Soluble Epoxide Hydrolase Inhibitors ◽

Fluorescence Polarization Assay

Rapid Determination of Soluble Epoxide Hydrolase Inhibitors in Rat Hepatic Microsomes by High-Performance Liquid Chromatography with Electrospray Tandem Mass Spectrometry

Analytical Biochemistry ◽

10.1006/abio.2001.5423 ◽

2001 ◽

Vol 299 (2) ◽

pp. 227-234 ◽

Cited By ~ 9

Author(s):

Takaho Watanabe ◽

Bruce D. Hammock

Keyword(s):

Mass Spectrometry ◽

High Performance ◽

Epoxide Hydrolase ◽

Rapid Determination ◽

Tandem Mass ◽

Electrospray Tandem Mass Spectrometry ◽

Hepatic Microsomes ◽

Faculty Opinions recommendation of Enhancement of antinociception by coadministration of nonsteroidal anti-inflammatory drugs and soluble epoxide hydrolase inhibitors.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1046256.496189 ◽

2006 ◽

Author(s):

Deanna Kroetz

Keyword(s):

Epoxide Hydrolase ◽

Soluble Epoxide Hydrolase Inhibitors ◽

Inflammatory Drugs ◽

Anti Inflammatory

Development of a high-throughput screen for soluble epoxide hydrolase inhibition

Analytical Biochemistry ◽

10.1016/j.ab.2006.04.045 ◽

2006 ◽

Vol 355 (1) ◽

pp. 71-80 ◽

Cited By ~ 52

Author(s):

Nicola M. Wolf ◽

Christophe Morisseau ◽

Paul D. Jones ◽

Bertold Hock ◽

Bruce D. Hammock

Keyword(s):

High Throughput ◽

Epoxide Hydrolase ◽

High Throughput Screen

Synthesis and Properties of N-[R-Adamantan-1(2)-yl]-N′-(2-fluorophenyl)ureas—Target-Oriented Soluble Epoxide Hydrolase Inhibitors

Russian Journal of Organic Chemistry ◽

10.1134/s1070428018090063 ◽

2018 ◽

Vol 54 (9) ◽

pp. 1307-1312 ◽

Cited By ~ 3

Author(s):

V. V. Burmistrov ◽

G. M. Butov

Keyword(s):

Epoxide Hydrolase ◽

Dietary soluble epoxide hydrolase inhibitors effect on hepatic gene expression of lipid metabolism in hamsters

The FASEB Journal ◽

10.1096/fasebj.22.1_supplement.479.53 ◽

2008 ◽

Vol 22 (S1) ◽

Author(s):

Glenn Bartley ◽

Hsing‐Ju Tsai ◽

Yun‐Jeong Hong ◽

Bruce Hammock ◽

Wallace Yokoyama

Keyword(s):

Gene Expression ◽

Lipid Metabolism ◽

Epoxide Hydrolase ◽

Hepatic Gene Expression ◽

Identifying Simultaneous Matrix Metalloproteinases/Soluble Epoxide Hydrolase Inhibitors

The FASEB Journal ◽

10.1096/fasebj.29.1_supplement.781.1 ◽

2015 ◽

Vol 29 (S1) ◽

Author(s):

Ahmed El‐Sherbeni ◽

Rabia Bhatti ◽

Ayman El‐Kadi

Keyword(s):

Matrix Metalloproteinases ◽

Epoxide Hydrolase ◽

Synthesis and properties of 1-(R-adamant-1-yl)-3-(1-propionylpiperidin-4-yl)ureas and 4-({4-[3-(R-adamant-1-yl)ureido]cyclohexyl}oxy)benzoic acids, efficient target-oriented human soluble epoxide hydrolase inhibitors

Russian Chemical Bulletin ◽

10.1007/s11172-017-1961-y ◽

2017 ◽

Vol 66 (10) ◽

pp. 1876-1880 ◽

Cited By ~ 5

Author(s):

G. M. Butov ◽

V. V. Burmistrov ◽

D. V. Danilov

Keyword(s):

Epoxide Hydrolase ◽

Benzoic Acids ◽

In vitro and in silico investigation of anthocyanin derivatives as soluble epoxide hydrolase inhibitors

International Journal of Biological Macromolecules ◽

10.1016/j.ijbiomac.2018.02.061 ◽

2018 ◽

Vol 112 ◽

pp. 961-967 ◽

Cited By ~ 5

Author(s):

Jang Hoon Kim ◽

In Sook Cho ◽

Jaihyuk Ryu ◽

Ji Sun Lee ◽

Jong Seong Kang ◽

...

Keyword(s):

In Silico ◽

Epoxide Hydrolase ◽

Discovery of Novel Soluble Epoxide Hydrolase Inhibitors as Potent Vasodilators

Scientific Reports ◽

10.1038/s41598-018-32449-4 ◽

2018 ◽

Vol 8 (1) ◽

Cited By ~ 7

Author(s):

Neetika Tripathi ◽

Sarvesh Paliwal ◽

Swapnil Sharma ◽

Kanika Verma ◽

Ritika Gururani ◽

...

Keyword(s):

Epoxide Hydrolase ◽

Optimization of a high-throughput fluorescence polarization assay for STAT5B DNA binding domain-targeting inhibitors

Journal of Pharmaceutical and Biomedical Analysis ◽

10.1016/j.jpba.2020.113182 ◽

2020 ◽

Vol 184 ◽

pp. 113182 ◽

Cited By ~ 1

Author(s):

Pimyupa Manaswiyoungkul ◽

Fettah Erdogan ◽

Olasunkanmi O. Olaoye ◽

Aaron D. Cabral ◽

Elvin D. de Araujo ◽

...

Keyword(s):

Dna Binding ◽

High Throughput ◽

Fluorescence Polarization ◽

Binding Domain ◽

Dna Binding Domain ◽

Fluorescence Polarization Assay