An in vivo Positron Emission Tomography Study of Adenosine 2A Receptor Occupancy by Preladenant using 11C-SCH442416 in Healthy Subjects

Igor Grachev; Miroslava Doder; David Brooks; Rainer Hinz

doi:10.17229/jdit.2014-0712-002

An in vivo Positron Emission Tomography Study of Adenosine 2A Receptor Occupancy by Preladenant using 11C-SCH442416 in Healthy Subjects

Journal of Diagnostic Imaging in Therapy ◽

10.17229/jdit.2014-0712-002 ◽

2014 ◽

Vol 1 (1) ◽

pp. 20-48 ◽

Cited By ~ 2

Author(s):

Igor Grachev ◽

Miroslava Doder ◽

David Brooks ◽

Rainer Hinz

Keyword(s):

Positron Emission Tomography ◽

Healthy Subjects ◽

Receptor Occupancy ◽

Emission Tomography ◽

Positron Emission Tomography Study ◽

Positron Emission ◽

Adenosine 2A Receptor

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Dopamine D2 receptor occupancy by perospirone: a positron emission tomography study in patients with schizophrenia and healthy subjects

Psychopharmacology ◽

10.1007/s00213-010-1783-1 ◽

2010 ◽

Vol 209 (4) ◽

pp. 285-290 ◽

Cited By ~ 7

Author(s):

Ryosuke Arakawa ◽

Hiroshi Ito ◽

Akihiro Takano ◽

Masaki Okumura ◽

Hidehiko Takahashi ◽

...

Keyword(s):

Positron Emission Tomography ◽

Healthy Subjects ◽

Dopamine D2 Receptor ◽

D2 Receptor ◽

Receptor Occupancy ◽

Emission Tomography ◽

Positron Emission Tomography Study ◽

Dopamine D2 ◽

Dopamine D2 Receptor Occupancy ◽

Positron Emission

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In Vivo Serotonin 5HT2A Receptor Binding and Personality Traits in Healthy Subjects: A Positron Emission Tomography Study

NeuroImage ◽

10.1006/nimg.2002.1239 ◽

2002 ◽

Vol 17 (3) ◽

pp. 1470-1478 ◽

Cited By ~ 69

Author(s):

F.M. Moresco ◽

M. Dieci ◽

A. Vita ◽

C. Messa ◽

C. Gobbo ◽

...

Keyword(s):

Positron Emission Tomography ◽

Personality Traits ◽

Receptor Binding ◽

Healthy Subjects ◽

Emission Tomography ◽

Positron Emission Tomography Study ◽

5Ht2a Receptor ◽

Positron Emission

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Faculty Opinions recommendation of D₂-receptor occupancy measurement of JNJ-37822681, a novel fast off-rate D₂-receptor antagonist, in healthy subjects using positron emission tomography: single dose versus steady state and dose selection.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.717953114.793458670 ◽

2012 ◽

Author(s):

John Davis

Keyword(s):

Positron Emission Tomography ◽

Single Dose ◽

Steady State ◽

Receptor Antagonist ◽

Healthy Subjects ◽

Receptor Occupancy ◽

Emission Tomography ◽

Dose Selection ◽

Positron Emission

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Significant effects of cholinesterase inhibitors on tau pathology in the Alzheimer's disease continuum: An in vivo positron emission tomography study

International Journal of Geriatric Psychiatry ◽

10.1002/gps.5522 ◽

2021 ◽

Author(s):

Fumihiko Yasuno ◽

Hiroyuki Minami

Keyword(s):

Alzheimer’S Disease ◽

Alzheimer's Disease ◽

Positron Emission Tomography ◽

Cholinesterase Inhibitors ◽

Emission Tomography ◽

Positron Emission Tomography Study ◽

Tau Pathology ◽

Positron Emission

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Correction to: An open-label, positron emission tomography study of the striatal D2/D3 receptor occupancy and pharmacokinetics of single-dose oral brexpiprazole in healthy participants

European Journal of Clinical Pharmacology ◽

10.1007/s00228-020-03071-z ◽

2021 ◽

Author(s):

Dean F. Wong ◽

Arash Raoufinia ◽

Patricia Bricmont ◽

James R. Brašić ◽

Robert D. McQuade ◽

...

Keyword(s):

Positron Emission Tomography ◽

Single Dose ◽

Receptor Occupancy ◽

Emission Tomography ◽

Positron Emission Tomography Study ◽

D3 Receptor ◽

Open Label ◽

Positron Emission ◽

Dose Oral ◽

Healthy Participants

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Positron emission tomography study of in vivo dopamine release using L-[11C]DOPA

Neuroscience Research Supplements ◽

10.1016/s0921-8696(06)80372-5 ◽

1991 ◽

Vol 14 ◽

pp. S128

Author(s):

Yasuyoshi Watanabe ◽

Per Hartvig ◽

Joakim Tedroff ◽

Peter Bjurling ◽

Hirotaka Onoe ◽

...

Keyword(s):

Positron Emission Tomography ◽

Dopamine Release ◽

Emission Tomography ◽

Positron Emission Tomography Study ◽

Positron Emission

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5-Hydroxytryptamine1A Receptor Occupancy by Novel Full Antagonist 2-[4-[4-(7-Chloro-2,3-dihydro-1,4-benzdioxyn-5-yl)-1-piperazinyl]butyl]-1,2-benzisothiazol-3-(2H)-one-1,1-dioxide: A [11C][O-methyl-3H]-N-(2-(4-(2-methoxyphenyl)-1-piperazinyl)ethyl)-N-(2-pyridinyl)cyclohexanecarboxamide Trihydrochloride (WAY-100635) Positron Emission Tomography Study in Humans

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.301.3.1144 ◽

2002 ◽

Vol 301 (3) ◽

pp. 1144-1150 ◽

Cited By ~ 37

Author(s):

Eugenii A. Rabiner ◽

Martin R. Wilkins ◽

Federico Turkheimer ◽

Roger N. Gunn ◽

Joanna Udo de Haes ◽

...

Keyword(s):

Positron Emission Tomography ◽

Receptor Occupancy ◽

Emission Tomography ◽

Positron Emission Tomography Study ◽

Positron Emission ◽

Way 100635

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A Positron Emission Tomography Study of Quetiapine in Schizophrenia: A Preliminary Finding of an Antipsychotic Effect With Only Transiently High Dopamine D2 Receptor Occupancy

Archives of General Psychiatry ◽

10.1001/archpsyc.57.6.553 ◽

2000 ◽

Vol 57 (6) ◽

pp. 553-559 ◽

Cited By ~ 253

Author(s):

S. Kapur

Keyword(s):

Positron Emission Tomography ◽

Dopamine D2 Receptor ◽

D2 Receptor ◽

Preliminary Finding ◽

Receptor Occupancy ◽

Emission Tomography ◽

Positron Emission Tomography Study ◽

Dopamine D2 Receptor Occupancy ◽

Antipsychotic Effect ◽

Positron Emission

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Central Benzodiazepine Receptors: Quantitative Positron Emission Tomography Study in Healthy Subjects and Anxious Patients

New Concepts in Anxiety ◽

10.1007/978-1-349-11847-2_15 ◽

1991 ◽

pp. 203-210

Author(s):

P. Abadie ◽

J. C. Bisserbe ◽

J. P. Boulenger ◽

J. M. Travere ◽

L. Barre ◽

...

Keyword(s):

Positron Emission Tomography ◽

Healthy Subjects ◽

Benzodiazepine Receptors ◽

Emission Tomography ◽

Positron Emission Tomography Study ◽

Positron Emission ◽

Central Benzodiazepine Receptors

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Brain histamine H1 receptor occupancy of orally administered antihistamines measured by positron emission tomography with 11C-doxepin in a placebo-controlled crossover study design in healthy subjects: a comparison of olopatadine and ketotifen

British Journal of Clinical Pharmacology ◽

10.1111/j.1365-2125.2005.02514.x ◽

2006 ◽

Vol 61 (1) ◽

pp. 16-26 ◽

Cited By ~ 49

Author(s):

Manabu Tashiro ◽

Hideki Mochizuki ◽

Yumiko Sakurada ◽

Kenji Ishii ◽

Keiichi Oda ◽

...

Keyword(s):

Positron Emission Tomography ◽

Crossover Study ◽

Study Design ◽

Healthy Subjects ◽

Receptor Occupancy ◽

Emission Tomography ◽

H1 Receptor ◽

Brain Histamine ◽

Positron Emission ◽

Histamine H1 Receptor Occupancy

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