Sustainable chemistry, synthesis and structure-activity relationship studies of biologically important small molecules

Mapping Intimacies ◽

10.31274/etd-180810-3391 ◽

2013 ◽

Author(s):

Gerald R. Pollock, III

Keyword(s):

Small Molecules ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Sustainable Chemistry ◽

Structure Activity

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TLR2 Agonistic Small Molecules: Detailed Structure–Activity Relationship, Applications, and Future Prospects

Journal of Medicinal Chemistry ◽

10.1021/acs.jmedchem.0c01627 ◽

2020 ◽

Author(s):

Arshpreet Kaur ◽

Deepender Kaushik ◽

Sakshi Piplani ◽

Surinder K. Mehta ◽

Nikolai Petrovsky ◽

...

Keyword(s):

Small Molecules ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Future Prospects ◽

Detailed Structure ◽

Structure Activity

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Ensemble learning-based quantitative structure-activity relationship platform predicts binding behavior of RNA-targeted small molecules

10.33774/chemrxiv-2021-czl9p ◽

2021 ◽

Author(s):

Zhengguo Cai ◽

Martina Zafferani ◽

Amanda Hargrove

Keyword(s):

Small Molecules ◽

Ensemble Learning ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Binding Behavior ◽

Structure Activity

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Structure‐activity relationship and mode of action studies highlight 1‐(4‐biphenylylmethyl)‐1H‐imidazole derived small molecules as potent CYP121 inhibitors

ChemMedChem ◽

10.1002/cmdc.202100283 ◽

2021 ◽

Author(s):

Sebastian Adam ◽

Isabell Walter ◽

Rolf Hartmann ◽

Andreas Kany ◽

Jesko Köhnke ◽

...

Keyword(s):

Small Molecules ◽

Mode Of Action ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity

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Evaluating Molecular Properties Involved in Transport of Small Molecules in Stratum Corneum: A Quantitative Structure-Activity Relationship for Skin Permeability

Molecules ◽

10.3390/molecules23040911 ◽

2018 ◽

Vol 23 (4) ◽

pp. 911 ◽

Author(s):

Chen-Peng Chen ◽

Chan-Cheng Chen ◽

Chia-Wen Huang ◽

Yen-Ching Chang

Keyword(s):

Stratum Corneum ◽

Small Molecules ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Molecular Properties ◽

Activity Relationship ◽

Skin Permeability ◽

Quantitative Structure ◽

Structure Activity

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Structure–Activity Relationship (SAR) Optimization of 6-(Indol-2-yl)pyridine-3-sulfonamides: Identification of Potent, Selective, and Orally Bioavailable Small Molecules Targeting Hepatitis C (HCV) NS4B

Journal of Medicinal Chemistry ◽

10.1021/jm401621g ◽

2013 ◽

Vol 57 (5) ◽

pp. 2121-2135 ◽

Author(s):

Nanjing Zhang ◽

Xiaoyan Zhang ◽

Jin Zhu ◽

Anthony Turpoff ◽

Guangming Chen ◽

...

Keyword(s):

Hepatitis C ◽

Small Molecules ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity ◽

Orally Bioavailable

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Structure-activity relationship of (-) mammea A/BB derivatives against Leishmania amazonensis

Planta Medica ◽

10.1055/s-0028-1084781 ◽

2008 ◽

Vol 74 (09) ◽

Author(s):

MA Brenzan ◽

CV Nakamura ◽

BPD Filho ◽

T Ueda-Nakamura ◽

MCM Young ◽

...

Keyword(s):

Structure Activity Relationship ◽

Leishmania Amazonensis ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Of

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Structure-activity-relationship (SAR) for in vitro antileishmanial activity of maesabalide (PX-6518) analogue natural products

Planta Medica ◽

10.1055/s-2006-949761 ◽

2006 ◽

Vol 72 (11) ◽

Author(s):

L Maes ◽

K Kuypers ◽

M Vermeersch ◽

P Cos ◽

L Pieters ◽

...

Keyword(s):

Natural Products ◽

Structure Activity Relationship ◽

Antileishmanial Activity ◽

Activity Relationship ◽

Structure Activity

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Structure Activity Relationship of Kahalalide F and its Analogs Against Fusarium Spp

Planta Medica ◽

10.1055/s-2008-1075262 ◽

2008 ◽

Vol 74 (03) ◽

Author(s):

N Kasanah ◽

AG Shilabin ◽

DE Wedge ◽

MT Hamann

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Fusarium Spp ◽

Structure Activity ◽

Kahalalide F ◽

Relationship Of

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STRUCTURE-ACTIVITY RELATIONSHIP OF VARIOUS ANALOGUES OF β-CORTICOTRROPHIN DETERMINED BY REFERENCE TO VARIOUS PARAMETERS IN VITRO AND IN VIVO

Acta Endocrinologica ◽

10.1530/acta.0.061s029 ◽

1969 ◽

Vol 61 (1_Suppl) ◽

pp. S29

Author(s):

Pierre A. Desaulles ◽

René Maier ◽

Matthys Staehelin

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Of

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Structure-Activity Relationship of the Antifungal 1-Aryl-2-(azol-1-yl)ethane Derivatives

Acta Phytopathologica et Entomologica Hungarica ◽

10.1556/aphyt.41.2006.1-2.11 ◽

2006 ◽

Vol 41 (1-2) ◽

pp. 109-119

Author(s):

I. Bélai ◽

G. Oros

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Of

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