STRUCTURE-ACTIVITY RELATIONSHIP OF VARIOUS ANALOGUES OF β-CORTICOTRROPHIN DETERMINED BY REFERENCE TO VARIOUS PARAMETERS IN VITRO AND IN VIVO

1969 ◽  
Vol 61 (1_Suppl) ◽  
pp. S29
Author(s):  
Pierre A. Desaulles ◽  
René Maier ◽  
Matthys Staehelin
2006 ◽  
Vol 49 (3) ◽  
pp. 1165-1181 ◽  
Author(s):  
Michael D. Wendt ◽  
Wang Shen ◽  
Aaron Kunzer ◽  
William J. McClellan ◽  
Milan Bruncko ◽  
...  

1998 ◽  
Vol 41 (11) ◽  
pp. 1777-1788 ◽  
Author(s):  
Thomas C. Kühler ◽  
Marianne Swanson ◽  
Vladimir Shcherbuchin ◽  
Håkan Larsson ◽  
Björn Mellgård ◽  
...  

2014 ◽  
Vol 12 (32) ◽  
pp. 6094-6104 ◽  
Author(s):  
Michael P. Storz ◽  
Giuseppe Allegretta ◽  
Benjamin Kirsch ◽  
Martin Empting ◽  
Rolf W. Hartmann

More than 60 derivatives of (2-nitrophenyl)methanol were synthesized and evaluated regarding their potency to inhibit PqsD. In vitro and in cellulo structure–activity relationships were derived.


2012 ◽  
Vol 3 (10) ◽  
pp. 814-817 ◽  
Author(s):  
Sheo B. Singh ◽  
Weiguo Liu ◽  
Xiaohua Li ◽  
Tom Chen ◽  
Ali Shafiee ◽  
...  

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