estrone sulfatase Latest Research Papers

Estrone Sulfatase Inhibitors as New Anticancer Agents

Chemistry and Biological Activity of Steroids ◽

10.5772/intechopen.85850 ◽

2020 ◽

Author(s):

Svetlana N. Morozkina ◽

Alexander G. Shavva

Keyword(s):

Anticancer Agents ◽

Estrone Sulfatase

Synthesis, Biological Evaluation and the Rationalisation of the Inhibitory Activity of a Range of Sulfonate Derivatives of Estrone (E1) in the Design of Reversible Inhibitors of Estrone Sulfatase (ES)

Letters in Drug Design & Discovery ◽

10.2174/1570180811666140226235116 ◽

2014 ◽

Vol 11 (8) ◽

pp. 985-992 ◽

Cited By ~ 1

Author(s):

Mohsen Akbarzadeh ◽

Timothy Cartledge ◽

Sabbir Ahmed

Keyword(s):

Inhibitory Activity ◽

Biological Evaluation ◽

Reversible Inhibitors ◽

Estrone Sulfatase ◽

Derivatives Of

Synthesis, In Vitro Activity and Rationalisation of a Series of Dialkyl Esters of 5-Aminosulfonylisophthanoate as Potential Estrone Sulfatase (ES) Inhibitors

Letters in Drug Design & Discovery ◽

10.2174/15701808113106660081 ◽

2014 ◽

Vol 11 (4) ◽

pp. 437-443

Author(s):

Sabbir Ahmed ◽

Chirag Patel

Keyword(s):

Vitro Activity ◽

In Vitro Activity ◽

Estrone Sulfatase

SYNTHESIS, BIOCHEMICAL EVALUATION AND RATIONALISATION OF A RANGE OF NOVEL THIOSEMICARBAZONE-BASED COMPOUNDS AS POTENTIALLY NEW CLASS OF DUAL INHIBITORS OF ESTRONE SULFATASE (ES) AND THE CYTOCHROME P-450 ENZYME AROMATASE (AR)

Letters in Drug Design & Discovery ◽

10.2174/15701808113109990047 ◽

2013 ◽

Vol 999 (999) ◽

pp. 13-18

Author(s):

Balkrishna Bhamare ◽

Sukriti Singh ◽

Bhanu C. Rudra ◽

Amit Kumar ◽

Sabbir Ahmed

Keyword(s):

Estrone Sulfatase ◽

New Class ◽

Biochemical Evaluation ◽

Dual Inhibitors ◽

Cytochrome P 450

Molecular Modelling, Design, Synthesis and Biochemical Evaluation of a Range of Non-Steroidal Thiosemicarbazone-Based Inhibitors of Estrone Sulfatase (ES) - A Potential Insight into the Action of a Range of Allosteric Inhibitors of ES

Letters in Drug Design & Discovery ◽

10.2174/157018011797200821 ◽

2011 ◽

Vol 8 (9) ◽

pp. 889-896

Author(s):

Amit Kumar ◽

Sukriti Singh ◽

Balkrishna Bhamare ◽

Kruti Shah ◽

Pallav S. Shah ◽

...

Keyword(s):

Molecular Modelling ◽

Allosteric Inhibitors ◽

Design Synthesis ◽

Estrone Sulfatase ◽

Biochemical Evaluation ◽

Insight Into

Aromatase, estrone sulfatase, and 17β-hydroxysteroid dehydrogenase: Structure–function studies and inhibitor development

Molecular and Cellular Endocrinology ◽

10.1016/j.mce.2010.09.012 ◽

2011 ◽

Vol 340 (2) ◽

pp. 120-126 ◽

Cited By ~ 17

Author(s):

Yanyan Hong ◽

Shiuan Chen

Keyword(s):

Structure Function ◽

Hydroxysteroid Dehydrogenase ◽

Inhibitor Development ◽

Estrone Sulfatase

Synthesis and Biological Evaluation of a Range of Thiosemicarbazone - Based Compounds as Potential Inhibitors of Estrone Sulfatase (ES)

Letters in Drug Design & Discovery ◽

10.2174/157018011794578231 ◽

2011 ◽

Vol 8 (3) ◽

pp. 241-245 ◽

Cited By ~ 3

Author(s):

Amit Kumar ◽

Sukriti Singh ◽

Hadi Bordbar ◽

Timothy Cartledge ◽

Sabbir Ahmed

Keyword(s):

Biological Evaluation ◽

Estrone Sulfatase ◽

Potential Inhibitors ◽

Synthesis And Biological Evaluation

Effect of tibolone and its principal metabolites (3α- and 3β-hydroxy, 3α-sulfate, and 4-ene derivatives) on estrone sulfatase activity in normal and cancerous human breast tissue

Hormone Molecular Biology and Clinical Investigation ◽

10.1515/hmbci.2011.121 ◽

2011 ◽

Vol 8 (3) ◽

Author(s):

Gérard S. Chetrite ◽

Joaquin Cortes-Prieto ◽

Jorge R. Pasqualini

Keyword(s):

Active Substance ◽

Breast Tissue ◽

Inhibitory Effect ◽

Human Breast ◽

Human Breast Tissue ◽

Estrone Sulfatase ◽

Significant Inhibitory Effect ◽

Sulfatase Activity

AbstractTibolone (Org-OD14) is the active substance of LivialTissue minces were incubated with physiological concentrations of [The sulfatase activity was significantly higher in cancerous breast but strongly inhibited by tibolone and the different metabolites, whereas 3α- and 3β-hydroxy derivatives were the most potent inhibitors.This very significant inhibitory effect of tibolone and its principal metabolites on the enzyme involved in E

Synthesis and In Vitro Biochemical Evaluation of a Series of Alkyl 6- Aminosulfonyl Naphthanoates as Potential Inhibitors of Human Placental Estrone Sulfatase (ES)

Letters in Drug Design & Discovery ◽

10.2174/157018011793663967 ◽

2011 ◽

Vol 8 (1) ◽

pp. 26-31

Author(s):

Chirag K. Patel ◽

Sabbir Ahmed

Keyword(s):

Estrone Sulfatase ◽

Biochemical Evaluation ◽

Potential Inhibitors

ChemInform Abstract: 17α-Alkyl- or 17α-Substituted Benzyl-17β-estradiols: A New Family of Estrone-Sulfatase Inhibitors.

ChemInform ◽

10.1002/chin.199846215 ◽

2010 ◽

Vol 29 (46) ◽

pp. no-no ◽

Cited By ~ 1

Author(s):

D. POIRIER ◽

R. P. BOIVIN

Keyword(s):

Estrone Sulfatase ◽

New Family

estrone sulfatase
Recently Published Documents

TOTAL DOCUMENTS

H-INDEX

Estrone Sulfatase Inhibitors as New Anticancer Agents

Synthesis, Biological Evaluation and the Rationalisation of the Inhibitory Activity of a Range of Sulfonate Derivatives of Estrone (E1) in the Design of Reversible Inhibitors of Estrone Sulfatase (ES)

Synthesis, In Vitro Activity and Rationalisation of a Series of Dialkyl Esters of 5-Aminosulfonylisophthanoate as Potential Estrone Sulfatase (ES) Inhibitors

SYNTHESIS, BIOCHEMICAL EVALUATION AND RATIONALISATION OF A RANGE OF NOVEL THIOSEMICARBAZONE-BASED COMPOUNDS AS POTENTIALLY NEW CLASS OF DUAL INHIBITORS OF ESTRONE SULFATASE (ES) AND THE CYTOCHROME P-450 ENZYME AROMATASE (AR)

Molecular Modelling, Design, Synthesis and Biochemical Evaluation of a Range of Non-Steroidal Thiosemicarbazone-Based Inhibitors of Estrone Sulfatase (ES) - A Potential Insight into the Action of a Range of Allosteric Inhibitors of ES

Aromatase, estrone sulfatase, and 17β-hydroxysteroid dehydrogenase: Structure–function studies and inhibitor development

Synthesis and Biological Evaluation of a Range of Thiosemicarbazone - Based Compounds as Potential Inhibitors of Estrone Sulfatase (ES)

Effect of tibolone and its principal metabolites (3α- and 3β-hydroxy, 3α-sulfate, and 4-ene derivatives) on estrone sulfatase activity in normal and cancerous human breast tissue

Synthesis and In Vitro Biochemical Evaluation of a Series of Alkyl 6- Aminosulfonyl Naphthanoates as Potential Inhibitors of Human Placental Estrone Sulfatase (ES)

ChemInform Abstract: 17α-Alkyl- or 17α-Substituted Benzyl-17β-estradiols: A New Family of Estrone-Sulfatase Inhibitors.

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estrone sulfataseRecently Published Documents

TOTAL DOCUMENTS

H-INDEX

Estrone Sulfatase Inhibitors as New Anticancer Agents

Synthesis, Biological Evaluation and the Rationalisation of the Inhibitory Activity of a Range of Sulfonate Derivatives of Estrone (E1) in the Design of Reversible Inhibitors of Estrone Sulfatase (ES)

Synthesis, In Vitro Activity and Rationalisation of a Series of Dialkyl Esters of 5-Aminosulfonylisophthanoate as Potential Estrone Sulfatase (ES) Inhibitors

SYNTHESIS, BIOCHEMICAL EVALUATION AND RATIONALISATION OF A RANGE OF NOVEL THIOSEMICARBAZONE-BASED COMPOUNDS AS POTENTIALLY NEW CLASS OF DUAL INHIBITORS OF ESTRONE SULFATASE (ES) AND THE CYTOCHROME P-450 ENZYME AROMATASE (AR)

Molecular Modelling, Design, Synthesis and Biochemical Evaluation of a Range of Non-Steroidal Thiosemicarbazone-Based Inhibitors of Estrone Sulfatase (ES) - A Potential Insight into the Action of a Range of Allosteric Inhibitors of ES

Aromatase, estrone sulfatase, and 17β-hydroxysteroid dehydrogenase: Structure–function studies and inhibitor development

Synthesis and Biological Evaluation of a Range of Thiosemicarbazone - Based Compounds as Potential Inhibitors of Estrone Sulfatase (ES)

Effect of tibolone and its principal metabolites (3α- and 3β-hydroxy, 3α-sulfate, and 4-ene derivatives) on estrone sulfatase activity in normal and cancerous human breast tissue

Synthesis and In Vitro Biochemical Evaluation of a Series of Alkyl 6- Aminosulfonyl Naphthanoates as Potential Inhibitors of Human Placental Estrone Sulfatase (ES)

ChemInform Abstract: 17α-Alkyl- or 17α-Substituted Benzyl-17β-estradiols: A New Family of Estrone-Sulfatase Inhibitors.

estrone sulfatase
Recently Published Documents