estrone sulfatase Latest Research Papers

AbstractTibolone (Org-OD14) is the active substance of LivialTissue minces were incubated with physiological concentrations of [The sulfatase activity was significantly higher in cancerous breast but strongly inhibited by tibolone and the different metabolites, whereas 3α- and 3β-hydroxy derivatives were the most potent inhibitors.This very significant inhibitory effect of tibolone and its principal metabolites on the enzyme involved in E

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Synthesis and In Vitro Biochemical Evaluation of a Series of Alkyl 6- Aminosulfonyl Naphthanoates as Potential Inhibitors of Human Placental Estrone Sulfatase (ES)

Letters in Drug Design & Discovery ◽

10.2174/157018011793663967 ◽

2011 ◽

Vol 8 (1) ◽

pp. 26-31

Author(s):

Chirag K. Patel ◽

Sabbir Ahmed

Keyword(s):

Estrone Sulfatase ◽

Biochemical Evaluation ◽

Potential Inhibitors

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ChemInform Abstract: 17α-Alkyl- or 17α-Substituted Benzyl-17β-estradiols: A New Family of Estrone-Sulfatase Inhibitors.

ChemInform ◽

10.1002/chin.199846215 ◽

2010 ◽

Vol 29 (46) ◽

pp. no-no ◽

Cited By ~ 1

Author(s):

D. POIRIER ◽

R. P. BOIVIN

Keyword(s):

Estrone Sulfatase ◽

New Family

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estrone sulfatase
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Estrone Sulfatase Inhibitors as New Anticancer Agents

Synthesis, Biological Evaluation and the Rationalisation of the Inhibitory Activity of a Range of Sulfonate Derivatives of Estrone (E1) in the Design of Reversible Inhibitors of Estrone Sulfatase (ES)

Synthesis, In Vitro Activity and Rationalisation of a Series of Dialkyl Esters of 5-Aminosulfonylisophthanoate as Potential Estrone Sulfatase (ES) Inhibitors

SYNTHESIS, BIOCHEMICAL EVALUATION AND RATIONALISATION OF A RANGE OF NOVEL THIOSEMICARBAZONE-BASED COMPOUNDS AS POTENTIALLY NEW CLASS OF DUAL INHIBITORS OF ESTRONE SULFATASE (ES) AND THE CYTOCHROME P-450 ENZYME AROMATASE (AR)

Molecular Modelling, Design, Synthesis and Biochemical Evaluation of a Range of Non-Steroidal Thiosemicarbazone-Based Inhibitors of Estrone Sulfatase (ES) - A Potential Insight into the Action of a Range of Allosteric Inhibitors of ES

Aromatase, estrone sulfatase, and 17β-hydroxysteroid dehydrogenase: Structure–function studies and inhibitor development

Synthesis and Biological Evaluation of a Range of Thiosemicarbazone - Based Compounds as Potential Inhibitors of Estrone Sulfatase (ES)

Effect of tibolone and its principal metabolites (3α- and 3β-hydroxy, 3α-sulfate, and 4-ene derivatives) on estrone sulfatase activity in normal and cancerous human breast tissue

Synthesis and In Vitro Biochemical Evaluation of a Series of Alkyl 6- Aminosulfonyl Naphthanoates as Potential Inhibitors of Human Placental Estrone Sulfatase (ES)

ChemInform Abstract: 17α-Alkyl- or 17α-Substituted Benzyl-17β-estradiols: A New Family of Estrone-Sulfatase Inhibitors.

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estrone sulfataseRecently Published Documents

TOTAL DOCUMENTS

H-INDEX

Estrone Sulfatase Inhibitors as New Anticancer Agents

Synthesis, Biological Evaluation and the Rationalisation of the Inhibitory Activity of a Range of Sulfonate Derivatives of Estrone (E1) in the Design of Reversible Inhibitors of Estrone Sulfatase (ES)

Synthesis, In Vitro Activity and Rationalisation of a Series of Dialkyl Esters of 5-Aminosulfonylisophthanoate as Potential Estrone Sulfatase (ES) Inhibitors

SYNTHESIS, BIOCHEMICAL EVALUATION AND RATIONALISATION OF A RANGE OF NOVEL THIOSEMICARBAZONE-BASED COMPOUNDS AS POTENTIALLY NEW CLASS OF DUAL INHIBITORS OF ESTRONE SULFATASE (ES) AND THE CYTOCHROME P-450 ENZYME AROMATASE (AR)

Molecular Modelling, Design, Synthesis and Biochemical Evaluation of a Range of Non-Steroidal Thiosemicarbazone-Based Inhibitors of Estrone Sulfatase (ES) - A Potential Insight into the Action of a Range of Allosteric Inhibitors of ES

Aromatase, estrone sulfatase, and 17β-hydroxysteroid dehydrogenase: Structure–function studies and inhibitor development

Synthesis and Biological Evaluation of a Range of Thiosemicarbazone - Based Compounds as Potential Inhibitors of Estrone Sulfatase (ES)

Effect of tibolone and its principal metabolites (3α- and 3β-hydroxy, 3α-sulfate, and 4-ene derivatives) on estrone sulfatase activity in normal and cancerous human breast tissue

Synthesis and In Vitro Biochemical Evaluation of a Series of Alkyl 6- Aminosulfonyl Naphthanoates as Potential Inhibitors of Human Placental Estrone Sulfatase (ES)

ChemInform Abstract: 17α-Alkyl- or 17α-Substituted Benzyl-17β-estradiols: A New Family of Estrone-Sulfatase Inhibitors.

estrone sulfatase
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