Brønsted Acid Catalyzed Domino Aza-Piancatelli Rearrangement/Michael Reaction: Construction of 1,4-Benzodiazepin-5-ones in One Pot

2017 ◽  
Vol 2017 (37) ◽  
pp. 5671-5678 ◽  
Author(s):  
Kiranmai Nayani ◽  
Radhika Cinsani ◽  
Anwar Hussaini SD ◽  
Prathama S. Mainkar ◽  
Srivari Chandrasekhar
ARKIVOC ◽  
2017 ◽  
Vol 2018 (2) ◽  
pp. 81-89
Author(s):  
Abhijeet Srivastava ◽  
Gaurav Shukla ◽  
Dhananjay Yadav ◽  
Maya Shankar Singh

Author(s):  
Xue-Jiao Lv ◽  
Yong-Chao Ming ◽  
Hui-Chun Wu ◽  
Yankai Liu

A Brønsted acid-catalyzed cascade acyclic N,O-hemiaminal formation/oxa-Michael reaction is developed for the synthesis of cis-2,6-disubstituted tetrahydropyrans bearing an exo amide group, that is, cyclic N,O-aminals. By using TsOH, various different...


2012 ◽  
Vol 67 (10) ◽  
pp. 1021-1029 ◽  
Author(s):  
Magnus Rueping ◽  
Stefan A. Moreth ◽  
Michael Bolte

The enantioselective synthesis of 2-aryl-substituted 2,3-dihydroquinolin-4-ones, a class of heterocyclic compounds with interesting biological activities, has been achieved through a Brønsted acidcatalyzed enantioselective intramolecular Michael addition. The products are available in moderate to high yields and with good enantioselectivities.


Synthesis ◽  
2007 ◽  
Vol 2007 (20) ◽  
pp. 3252-3256 ◽  
Author(s):  
Roberto Sanz ◽  
Félix Rodríguez ◽  
Alberto Martínez ◽  
Delia Miguel ◽  
Julia Álvarez-Gutiérrez

2015 ◽  
Vol 26 (20) ◽  
pp. 1180-1188 ◽  
Author(s):  
Margherita Barbero ◽  
Silvano Cadamuro ◽  
Stefano Dughera

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