Biased agonism at histamine H1 receptor: Desensitization, internalization and MAPK activation triggered by antihistamines

2021 ◽  
Vol 896 ◽  
pp. 173913
Author(s):  
Valeria Burghi ◽  
Emiliana B. Echeverría ◽  
Carlos D. Zappia ◽  
Antonela Díaz Nebreda ◽  
Sonia Ripoll ◽  
...  
Keyword(s):  
Receptor Desensitization ◽  
H1 Receptor ◽  
Mapk Activation ◽  
Histamine H1 Receptor ◽  
Biased Agonism

scholarly journals Protein kinase C-mediated histamine H1 receptor desensitization through direct phosphorylation of the receptor

1998 ◽  
Vol 76 ◽  
pp. 107
Author(s):  
Katsumi Fujimoto ◽  
Kazumi Ohta ◽  
Kenji Kangawa ◽  
Ushio Kikkawa ◽  
Satoshi Ogino ◽  
...  
Keyword(s):  
Protein Kinase C ◽  
Protein Kinase ◽  
Receptor Desensitization ◽  
H1 Receptor ◽  
Histamine H1 Receptor ◽  
Kinase C

Is Protein Kinase C Involved in Histamine H1-receptor Desensitization ?

1991 ◽  
pp. 393-402 ◽  
Author(s):  
R. Leurs ◽  
M. J. Smit ◽  
M. M. Brozius ◽  
W. Jansen ◽  
A. Bast ◽  
...  
Keyword(s):  
Protein Kinase C ◽  
Protein Kinase ◽  
Receptor Desensitization ◽  
H1 Receptor ◽  
Histamine H1 Receptor ◽  
Kinase C

scholarly journals Design of Phthalazinone Amide Histamine H1 Receptor Antagonists for Use in Rhinitis

2017 ◽  
Vol 8 (5) ◽  
pp. 577-581 ◽  
Author(s):  
Panayiotis A. Procopiou ◽  
Alison J. Ford ◽  
Paul M. Gore ◽  
Brian E. Looker ◽  
Simon T. Hodgson ◽  
...  
Keyword(s):  
H1 Receptor ◽  
Receptor Antagonists ◽  
Histamine H1 Receptor

Histamine H1 receptor ligands

Il Farmaco ◽  
1999 ◽  
Vol 54 (8) ◽  
pp. 533-541 ◽  
Author(s):  
K. Walczyński ◽  
H. Timmerman ◽  
O.P. Zuiderveld ◽  
M.Q. Zhang ◽  
R. Glinka
Keyword(s):  
Receptor Ligands ◽  
H1 Receptor ◽  
Histamine H1 Receptor
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