Arachidonylsulfonyl derivatives as cannabinoid CB1 receptor and fatty acid amide hydrolase inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(03)00721-2 ◽

2003 ◽

Vol 13 (19) ◽

pp. 3301-3303 ◽

Author(s):

Yoffi Segall ◽

Gary B. Quistad ◽

Daniel K. Nomura ◽

John E. Casida

Keyword(s):

Fatty Acid Amide Hydrolase ◽

Cb1 Receptor ◽

Cannabinoid Cb1 Receptor ◽

Amide Hydrolase ◽

Fatty Acid Amide

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Preservation of Striatal Cannabinoid CB1 Receptor Function Correlates with the Antianxiety Effects of Fatty Acid Amide Hydrolase Inhibition

Molecular Pharmacology ◽

10.1124/mol.110.064196 ◽

2010 ◽

Vol 78 (2) ◽

pp. 260-268 ◽

Author(s):

Silvia Rossi ◽

Valentina De Chiara ◽

Alessandra Musella ◽

Lucia Sacchetti ◽

Cristina Cantarella ◽

...

Keyword(s):

Fatty Acid Amide Hydrolase ◽

Cb1 Receptor ◽

Receptor Function ◽

Cannabinoid Cb1 Receptor ◽

Amide Hydrolase ◽

Fatty Acid Amide

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Immunocytochemical localization of cannabinoid CB1 receptor and fatty acid amide hydrolase in rat retina

The Journal of Comparative Neurology ◽

10.1002/(sici)1096-9861(19991206)415:1<80::aid-cne6>3.0.co;2-h ◽

1999 ◽

Vol 415 (1) ◽

pp. 80-90 ◽

Author(s):

Stephen Yazulla ◽

Keith M. Studholme ◽

Helen H. McIntosh ◽

Dale G. Deutsch

Keyword(s):

Fatty Acid Amide Hydrolase ◽

Cb1 Receptor ◽

Immunocytochemical Localization ◽

Cannabinoid Cb1 Receptor ◽

Amide Hydrolase ◽

Fatty Acid Amide

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Cannabinoid CB1 receptor; fatty acid amide hydrolase (FAAH); monoacylglycerol lipase (MAGL)

Science-Business eXchange ◽

10.1038/scibx.2008.806 ◽

2008 ◽

Vol 1 (33) ◽

pp. 806-806

Keyword(s):

Fatty Acid Amide Hydrolase ◽

Cb1 Receptor ◽

Monoacylglycerol Lipase ◽

Cannabinoid Cb1 Receptor ◽

Amide Hydrolase ◽

Fatty Acid Amide

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Involvement of Endocannabinoids in Alcohol “Binge” Drinking: Studies of Mice with Human Fatty Acid Amide Hydrolase Genetic Variation and After CB1 Receptor Antagonists

Alcoholism Clinical and Experimental Research ◽

10.1111/acer.12989 ◽

2016 ◽

Vol 40 (3) ◽

pp. 467-473 ◽

Author(s):

Yan Zhou ◽

Ted Huang ◽

Francis Lee ◽

Mary Jeanne Kreek

Keyword(s):

Genetic Variation ◽

Binge Drinking ◽

Fatty Acid Amide Hydrolase ◽

Cb1 Receptor ◽

Receptor Antagonists ◽

Amide Hydrolase ◽

Cb1 Receptor Antagonists ◽

Fatty Acid Amide

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Interference with acute nausea and anticipatory nausea in rats by fatty acid amide hydrolase (FAAH) inhibition through a PPARα and CB1 receptor mechanism, respectively: a double dissociation

Psychopharmacology ◽

10.1007/s00213-015-4050-7 ◽

2015 ◽

Vol 232 (20) ◽

pp. 3841-3848 ◽

Author(s):

Erin M. Rock ◽

Cheryl L. Limebeer ◽

Jordan M. Ward ◽

Arianne Cohen ◽

Katherine Grove ◽

...

Keyword(s):

Fatty Acid Amide Hydrolase ◽

Cb1 Receptor ◽

Anticipatory Nausea ◽

Acute Nausea ◽

Double Dissociation ◽

Faah Inhibition ◽

Amide Hydrolase ◽

Fatty Acid Amide

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Inhibition of fatty acid amide hydrolase reduces reinstatement of nicotine seeking but not break point for nicotine self-administration—comparison with CB1 receptor blockade

Psychopharmacology ◽

10.1007/s00213-009-1569-5 ◽

2009 ◽

Vol 205 (4) ◽

pp. 613-624 ◽

Author(s):

Benoit Forget ◽

Kathleen M. Coen ◽

Bernard Le Foll

Keyword(s):

Fatty Acid Amide Hydrolase ◽

Break Point ◽

Cb1 Receptor ◽

Receptor Blockade ◽

Self Administration ◽

Amide Hydrolase ◽

Fatty Acid Amide

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Inhibition of fatty-acid amide hydrolase and CB1 receptor antagonism differentially affect behavioural responses in normal and PCP-treated rats

The International Journal of Neuropsychopharmacology ◽

10.1017/s146114570999023x ◽

2009 ◽

Vol 13 (03) ◽

pp. 373 ◽

Author(s):

Alexandre Seillier ◽

Tushar Advani ◽

Tomasso Cassano ◽

Julie G. Hensler ◽

Andrea Giuffrida

Keyword(s):

Fatty Acid Amide Hydrolase ◽

Cb1 Receptor ◽

Receptor Antagonism ◽

Behavioural Responses ◽

Amide Hydrolase ◽

Fatty Acid Amide

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Fatty Acid Amide Hydrolase in Prostate Cancer: Association with Disease Severity and Outcome, CB1 Receptor Expression and Regulation by IL-4

PLoS ONE ◽

10.1371/journal.pone.0012275 ◽

2010 ◽

Vol 5 (8) ◽

pp. e12275 ◽

Author(s):

Lina Thors ◽

Anders Bergh ◽

Emma Persson ◽

Peter Hammarsten ◽

Pär Stattin ◽

...

Keyword(s):

Prostate Cancer ◽

Disease Severity ◽

Fatty Acid Amide Hydrolase ◽

Cb1 Receptor ◽

Receptor Expression ◽

Amide Hydrolase ◽

Fatty Acid Amide

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A new perspective on cannabinoid signalling: complimentary localization of fatty acid amide hydrolase and the CB1 receptor in rat brain.

Proceedings of The Royal Society B Biological Sciences ◽

10.1098/rspb.1998.0543 ◽

1998 ◽

Vol 265 (1410) ◽

pp. 2081-2085 ◽

Author(s):

M. Egertová ◽

D. K. Giang ◽

B. F. Cravatt ◽

M. R. Elphick

Keyword(s):

Rat Brain ◽

Fatty Acid Amide Hydrolase ◽

Cb1 Receptor ◽

Amide Hydrolase ◽

New Perspective ◽

Fatty Acid Amide

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Faculty Opinions recommendation of Inactivation of fatty acid amide hydrolase exacerbates experimental fibrosis by enhanced endocannabinoid-mediated activation of CB1.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.717956659.793461149 ◽

2012 ◽

Author(s):

Jaap van Laar ◽

Steven O'Reilly

Keyword(s):

Fatty Acid Amide Hydrolase ◽

Amide Hydrolase ◽

Fatty Acid Amide

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