Synthesis and Pharmacological Characterization of Visabron, a Backbone Cyclic Peptide Dual Antagonist of α4β1 (VLA-4)/α9β1 Integrin for Therapy of Multiple Sclerosis

Development and Pharmacological Characterization of Selective Blockers of 2-Arachidonoyl Glycerol Degradation with Efficacy in Rodent Models of Multiple Sclerosis and Pain

Journal of Medicinal Chemistry ◽

10.1021/acs.jmedchem.5b01812 ◽

2016 ◽

Vol 59 (6) ◽

pp. 2612-2632 ◽

Cited By ~ 39

Author(s):

Margherita Brindisi ◽

Samuele Maramai ◽

Sandra Gemma ◽

Simone Brogi ◽

Alessandro Grillo ◽

...

Keyword(s):

Multiple Sclerosis ◽

Rodent Models ◽

Arachidonoyl Glycerol

A High-Throughput Assay for the Pancreatic Islet Beta-Cell Potassium Channel: Use in the Pharmacological Characterization of Insulin Secretagogues Identified from Phenotypic Screening

Assay and Drug Development Technologies ◽

10.1089/adt.2020.1011 ◽

2020 ◽

Author(s):

Luyan Song ◽

David G. Barrett ◽

Karen L. Cox ◽

Alexander M. Efanov ◽

Samreen K. Syed ◽

...

Keyword(s):

Beta Cell ◽

Potassium Channel ◽

Pancreatic Islet ◽

High Throughput ◽

Phenotypic Screening ◽

Insulin Secretagogues ◽

High Throughput Assay ◽

Pancreatic Islet Beta Cell

Pharmacological characterization of a novel, orally available GluN2B antagonist JNJ‐63612445

The FASEB Journal ◽

10.1096/fasebj.2020.34.s1.02535 ◽

2020 ◽

Vol 34 (S1) ◽

pp. 1-1

Author(s):

Bartosz Balana ◽

Jeffrey Schoellerman ◽

Brian Lord ◽

Ryan Wyatt ◽

Jose Matta ◽

...

Keyword(s):

Pharmacological characterization of the beta-adrenoceptor coupled to cyclic AMP formation, expressed by rat mesenteric artery vascular smooth muscle cells in culture

Journal of Hypertension ◽

10.1097/00004872-199112000-00032 ◽

1991 ◽

Vol 9 (6) ◽

pp. S98

Author(s):

Alistair S. Hall ◽

Susan E. Bryson ◽

Stephen G. Ball ◽

Anthony J. Balmforth

Keyword(s):

Smooth Muscle ◽

Cyclic Amp ◽

Vascular Smooth Muscle ◽

Smooth Muscle Cells ◽

Vascular Smooth Muscle Cells ◽

Mesenteric Artery ◽

Beta Adrenoceptor ◽

Rat Mesenteric Artery

Multiple sclerosis and periodic fever syndromes: Characterization of clinical symptoms

Neuropediatrics ◽

10.1055/s-0032-1307064 ◽

2012 ◽

Vol 43 (02) ◽

Author(s):

A Blaschek ◽

P Lohse ◽

F Heinen ◽

W Müller-Felber

Keyword(s):

Multiple Sclerosis ◽

Clinical Symptoms ◽

Periodic Fever ◽

Periodic Fever Syndromes ◽

Fever Syndromes

Structure-based design, synthesis and pharmacological characterization of estrogen receptor isotype selective ligands

Experimental and Clinical Endocrinology & Diabetes ◽

10.1055/s-2004-819048 ◽

2004 ◽

Vol 112 (S 1) ◽

Author(s):

A Hillisch ◽

O Peters ◽

D Kosemund ◽

G Müller ◽

C Hegele-Hartung ◽

...

Keyword(s):

Estrogen Receptor ◽

Design Synthesis ◽

Selective Ligands

Pharmacological characterization of α1-adrenoceptors In rabbit thoracic aorta

The Japanese Journal of Pharmacology ◽

10.1016/s0021-5198(19)49290-1 ◽

1992 ◽

Vol 58 ◽

pp. 265

Author(s):

Masafumi Oshita ◽

Manabu Takita ◽

Sigeru Klgoshi ◽

Ikunobu Muramatsu

Keyword(s):

Thoracic Aorta ◽

Pharmacological Characterization Of The Late Phase Reduction In Forced Vital Capacity (FVC) In Allergen-Challenged Brown Norway Rats: Correlations With Lung Edema

10.1164/ajrccm-conference.2011.183.1_meetingabstracts.a2880 ◽

2011 ◽

Author(s):

Peter Mauser ◽

Richard Chapman ◽

Howard Jones ◽

Aileen House ◽

Craig Correll

Keyword(s):

Forced Vital Capacity ◽

Vital Capacity ◽

Late Phase ◽

Brown Norway ◽

Lung Edema ◽

Phase Reduction ◽

Norway Rats

Pharmacological characterization of a novel 5-HT4 receptor agonist, TS-951 in vitro.

The Japanese Journal of Pharmacology ◽

10.1016/s0021-5198(19)34836-x ◽

1999 ◽

Vol 79 ◽

pp. 206

Author(s):

Sumiyo Kajita ◽

Chika Ito ◽

Yoshihiko Isobe ◽

Kiyomi Fukushima

Keyword(s):

Receptor Agonist ◽

Pharmacological Characterization of Mouse Hind Paw Edema Induced by Parachartergus fraternus Venom

Inflammation ◽

10.1007/s10753-019-01062-6 ◽

2019 ◽

Vol 42 (6) ◽

pp. 2011-2019 ◽

Cited By ~ 1

Author(s):

Jéssica de Araujo Isaias Muller ◽

Márcia Renata Mortari ◽

Iluska Senna Bonfá Moslaves ◽

Mônica Cristina Toffoli-Kadri

Keyword(s):

Paw Edema ◽