Discovery and Structure−Activity Relationship of N-(Ureidoalkyl)-Benzyl-Piperidines As Potent Small Molecule CC Chemokine Receptor-3 (CCR3) Antagonists

2002 ◽  
Vol 45 (17) ◽  
pp. 3794-3804 ◽  
Author(s):  
George V. De Lucca ◽  
Ui T. Kim ◽  
Curt Johnson ◽  
Brian J. Vargo ◽  
Patricia K. Welch ◽  
...  
Keyword(s):  
Small Molecule ◽  
Chemokine Receptor ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Cc Chemokine ◽  
Structure Activity ◽  
Relationship Of

Synthesis and Structure−Activity Relationship of the First Nonpeptidergic Inverse Agonists for the Human Cytomegalovirus Encoded Chemokine Receptor US28

2005 ◽  
Vol 48 (20) ◽  
pp. 6461-6471 ◽  
Author(s):  
Janneke W. Hulshof ◽  
Paola Casarosa ◽  
Wiro M. P. B. Menge ◽  
Leena M. S. Kuusisto ◽  
Henk van der Goot ◽  
...  
Keyword(s):  
Human Cytomegalovirus ◽  
Chemokine Receptor ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Inverse Agonists ◽  
Structure Activity ◽  
Relationship Of

scholarly journals Discovery and Structure Activity Relationship of Small Molecule Inhibitors of Toxic β-Amyloid-42 Fibril Formation

2012 ◽  
Vol 287 (41) ◽  
pp. 34786-34800 ◽  
Author(s):  
Heiko Kroth ◽  
Annalisa Ansaloni ◽  
Yvan Varisco ◽  
Asad Jan ◽  
Nampally Sreenivasachary ◽  
...  
Keyword(s):  
Small Molecule ◽  
Small Molecule Inhibitors ◽  
Structure Activity Relationship ◽  
Fibril Formation ◽  
Activity Relationship ◽  
Structure Activity ◽  
Β Amyloid ◽  
Relationship Of

Synthesis and structure–activity relationship of 3-phenyl-3H-quinazolin-4-one derivatives as CXCR3 chemokine receptor antagonists

2005 ◽  
Vol 15 (11) ◽  
pp. 2910-2913 ◽  
Author(s):  
Stefania Storelli ◽  
Pauline Verdijk ◽  
Dennis Verzijl ◽  
Henk Timmerman ◽  
Andrea C. van de Stolpe ◽  
...  
Keyword(s):  
Chemokine Receptor ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Receptor Antagonists ◽  
Structure Activity ◽  
Relationship Of

A Small Molecule, Lys-Ala-7-amido-4-methylcoumarin, Facilitates RNA Dimer Maturation of a Stem−Loop 1 Transcript in Vitro: Structure−Activity Relationship of the Activator†

Biochemistry ◽  
2008 ◽  
Vol 47 (31) ◽  
pp. 8148-8156 ◽  
Author(s):  
Janet Chung ◽  
Anwer Mujeeb ◽  
Yongying Jiang ◽  
Christophe Guilbert ◽  
Mrunal Pendke ◽  
...  
Keyword(s):  
Small Molecule ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Stem Loop ◽  
Structure Activity ◽  
Rna Dimer ◽  
Relationship Of

Modification and structure–activity relationship of a small molecule HIV-1 inhibitor targeting the viral envelope glycoprotein gp120

2005 ◽  
Vol 3 (9) ◽  
pp. 1781 ◽  
Author(s):  
Jingsong Wang ◽  
Nhut Le ◽  
Alonso Heredia ◽  
Haijing Song ◽  
Robert Redfield ◽  
...  
Keyword(s):  
Small Molecule ◽  
Envelope Glycoprotein ◽  
Structure Activity Relationship ◽  
Viral Envelope ◽  
Activity Relationship ◽  
Viral Envelope Glycoprotein ◽  
Structure Activity ◽  
Glycoprotein Gp120 ◽  
Relationship Of ◽  
Hiv 1

Synthesis and structure–Activity relationship of 2-amino-3-heteroaryl-quinoxalines as non-peptide, small-Molecule antagonists for interleukin-8 receptor

2003 ◽  
Vol 11 (17) ◽  
pp. 3777-3790 ◽  
Author(s):  
Jie Jack Li ◽  
Kenneth G Carson ◽  
Bharat K Trivedi ◽  
Wen Song Yue ◽  
Qing Ye ◽  
...  
Keyword(s):  
Small Molecule ◽  
Structure Activity Relationship ◽  
Interleukin 8 ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of

Synthesis and Structure−Activity Relationship of Small-Molecule Malonyl Coenzyme A Decarboxylase Inhibitors

2006 ◽  
Vol 49 (5) ◽  
pp. 1517-1525 ◽  
Author(s):  
Jie-Fei Cheng ◽  
Mi Chen ◽  
David Wallace ◽  
Souvothy Tith ◽  
Masayuki Haramura ◽  
...  
Keyword(s):  
Small Molecule ◽  
Coenzyme A ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity ◽  
Decarboxylase Inhibitors ◽  
Relationship Of

Logical synthetic strategies and structure-activity relationship of indolin-2-one hybrids as small molecule anticancer agents: An overview

2022 ◽  
Vol 1247 ◽  
pp. 131280
Author(s):  
Prashant Chaudhari ◽  
Sanjaykumar Bari ◽  
Sanjay Surana ◽  
Atul Shirkhedkar ◽  
Sharad Wakode ◽  
...  
Keyword(s):  
Small Molecule ◽  
Anticancer Agents ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of

Structure-activity relationship of (-) mammea A/BB derivatives against Leishmania amazonensis

Planta Medica ◽  
2008 ◽  
Vol 74 (09) ◽  
Author(s):  
MA Brenzan ◽  
CV Nakamura ◽  
BPD Filho ◽  
T Ueda-Nakamura ◽  
MCM Young ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Leishmania Amazonensis ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of
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