Design, Synthesis, and Biological Evaluation of Novel Deguelin-Based Heat Shock Protein 90 (HSP90) Inhibitors Targeting Proliferation and Angiogenesis

2012 ◽  
Vol 55 (24) ◽  
pp. 10863-10884 ◽  
Author(s):  
Dong-Jo Chang ◽  
Hongchan An ◽  
Kyoung-suk Kim ◽  
Hyun Ho Kim ◽  
Jinkyung Jung ◽  
...  
Keyword(s):  
Heat Shock ◽  
Heat Shock Protein ◽  
Heat Shock Protein 90 ◽  
Biological Evaluation ◽  
Hsp90 Inhibitors ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation

Synthesis and biological evaluation of C-ring truncated deguelin derivatives as heat shock protein 90 (HSP90) inhibitors

2016 ◽  
Vol 24 (22) ◽  
pp. 6082-6093 ◽  
Author(s):  
Ho Shin Kim ◽  
Mannkyu Hong ◽  
Jihyae Ann ◽  
Suyoung Yoon ◽  
Cong-Truong Nguyen ◽  
...  
Keyword(s):  
Heat Shock ◽  
Heat Shock Protein ◽  
Heat Shock Protein 90 ◽  
Biological Evaluation ◽  
Hsp90 Inhibitors ◽  
Synthesis And Biological Evaluation

Synthesis and biological evaluation of 2,4-diaminoquinazoline derivatives as novel heat shock protein 90 inhibitors

2011 ◽  
Vol 21 (6) ◽  
pp. 1593-1597 ◽  
Author(s):  
Dhanaji Achyutrao Thorat ◽  
Munikumar Reddy Doddareddy ◽  
Seon Hee Seo ◽  
Tae-Joon Hong ◽  
Yong Seo Cho ◽  
...  
Keyword(s):  
Heat Shock ◽  
Heat Shock Protein ◽  
Heat Shock Protein 90 ◽  
Biological Evaluation ◽  
Synthesis And Biological Evaluation

Synthesis and biological evaluation of novobiocin analogues as potential heat shock protein 90 inhibitors

2013 ◽  
Vol 21 (17) ◽  
pp. 5118-5129 ◽  
Author(s):  
G.M. Kamal B. Gunaherath ◽  
Marilyn T. Marron ◽  
E.M. Kithsiri Wijeratne ◽  
Luke Whitesell ◽  
A.A. Leslie Gunatilaka
Keyword(s):  
Heat Shock ◽  
Heat Shock Protein ◽  
Heat Shock Protein 90 ◽  
Biological Evaluation ◽  
Synthesis And Biological Evaluation

Design, Synthesis, and Evaluation of Heat Shock Protein 90 Inhibitors in Human Breast Cancer and Its Metastasis

2016 ◽  
Vol 17 (14) ◽  
pp. 1231-1245 ◽  
Author(s):  
Mehmet Gümus ◽  
Aykut Ozgur ◽  
Lutfi Tutar ◽  
Ali Disli ◽  
Irfan Koca ◽  
...  
Keyword(s):  
Breast Cancer ◽  
Heat Shock ◽  
Heat Shock Protein ◽  
Human Breast Cancer ◽  
Heat Shock Protein 90 ◽  
Human Breast ◽  
Design Synthesis

Ligand Desolvation Steers On-Rate and Impacts Drug Residence Time of Heat Shock Protein 90 (Hsp90) Inhibitors

2018 ◽  
Vol 61 (10) ◽  
pp. 4397-4411 ◽  
Author(s):  
Doris A. Schuetz ◽  
Lars Richter ◽  
Marta Amaral ◽  
Melanie Grandits ◽  
Ulrich Grädler ◽  
...  
Keyword(s):  
Heat Shock ◽  
Heat Shock Protein ◽  
Residence Time ◽  
Heat Shock Protein 90 ◽  
Hsp90 Inhibitors

Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach

2016 ◽  
Vol 22 (37) ◽  
pp. 13236-13250 ◽  
Author(s):  
Maria G. Chini ◽  
Nicola Malafronte ◽  
Maria C. Vaccaro ◽  
Maria J. Gualtieri ◽  
Antonio Vassallo ◽  
...  
Keyword(s):  
Heat Shock ◽  
Heat Shock Protein ◽  
Multidisciplinary Approach ◽  
Heat Shock Protein 90 ◽  
Hsp90 Inhibitors
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