Probing the origin of estrogen receptor alpha inhibition via large-scale QSAR study

RSC Advances ◽

10.1039/c7ra10979b ◽

2018 ◽

Vol 8 (21) ◽

pp. 11344-11356 ◽

Author(s):

Naravut Suvannang ◽

Likit Preeyanon ◽

Aijaz Ahmad Malik ◽

Nalini Schaduangrat ◽

Watshara Shoombuatong ◽

...

Keyword(s):

Estrogen Receptor ◽

Inhibitory Activity ◽

Large Scale ◽

Estrogen Receptor Alpha ◽

Qsar Modeling ◽

This study compiles a large, non-redundant set of compounds tested for ERα inhibitory activity and applies QSAR modeling for unveiling the privileged substructures governing the activity.

Download Full-text

In silico approach for revealing the anti-breast cancer and estrogen receptor alpha inhibitory activity of Artocarpus altilis

10.1063/1.5062801 ◽

2018 ◽

Author(s):

Aida Fitriah ◽

Kholifah Holil ◽

Umaiyatus Syarifah ◽

Fitriyah ◽

Didik Huswo Utomo

Keyword(s):

Breast Cancer ◽

Estrogen Receptor ◽

Inhibitory Activity ◽

In Silico ◽

Estrogen Receptor Alpha ◽

Artocarpus Altilis ◽

Download Full-text

QSAR modeling, docking, ADME and reactivity of indazole derivatives as antagonizes of estrogen receptor alpha (ER-α) positive in breast cancer

Journal of Molecular Structure ◽

10.1016/j.molstruc.2020.128442 ◽

2020 ◽

Vol 1217 ◽

pp. 128442 ◽

Author(s):

Afaf Zekri ◽

Dalal Harkati ◽

Samir Kenouche ◽

Basil A. Saleh

Keyword(s):

Breast Cancer ◽

Estrogen Receptor ◽

Estrogen Receptor Alpha ◽

Qsar Modeling ◽

Download Full-text

Author response for "Estrogen receptor alpha, g‐protein coupled receptor 1, and aromatase: developmental, sex, and region‐specific differences across the rat caudate‐putamen, nucleus accumbens core and shell"

10.1002/cne.24978/v4/response1 ◽

2020 ◽

Author(s):

Amanda A. Krentzel ◽

Jaime A. Willett ◽

Ashlyn G. Johnson ◽

John Meitzen

Keyword(s):

Estrogen Receptor ◽

Nucleus Accumbens ◽

G Protein ◽

Estrogen Receptor Alpha ◽

Author Response ◽

G Protein Coupled Receptor ◽

Nucleus Accumbens Core ◽

Caudate Putamen ◽

Receptor Alpha ◽

G Protein Coupled

Download Full-text

Author response for "Estrogen receptor alpha, g‐protein coupled receptor 1, and aromatase: developmental, sex, and region‐specific differences across the rat caudate‐putamen, nucleus accumbens core and shell"

10.1002/cne.24978/v3/response1 ◽

2020 ◽

Author(s):

Amanda A. Krentzel ◽

Jaime A. Willett ◽

Ashlyn G. Johnson ◽

John Meitzen

Keyword(s):

Estrogen Receptor ◽

Nucleus Accumbens ◽

G Protein ◽

Estrogen Receptor Alpha ◽

Author Response ◽

G Protein Coupled Receptor ◽

Nucleus Accumbens Core ◽

Caudate Putamen ◽

Receptor Alpha ◽

G Protein Coupled

Download Full-text

Die Kaffee-vermittelte Induktion von UDP-Glukuronosyltransferasen wird durch den Estrogen-Receptor-alpha (ESR-1) geschlechtspezifisch reguliert

Zeitschrift für Gastroenterologie ◽

10.1055/s-0031-1285168 ◽

2011 ◽

Vol 49 (08) ◽

Author(s):

S Kalthoff ◽

A Winkler ◽

N Freiberg ◽

M Manns ◽

C Strassburg

Keyword(s):

Estrogen Receptor ◽

Estrogen Receptor Alpha ◽

Download Full-text

Mice lacking estrogen receptor [alpha] in hypothalamic POMC neurons display enhanced estrogenic response on cortical bone mass

Bone Abstracts ◽

10.1530/boneabs.5.ht2 ◽

2016 ◽

Author(s):

Helen Farman ◽

Sara Windahl ◽

Deborah Clegg ◽

Shang Kui Xie ◽

Lars Westberg ◽

...

Keyword(s):

Estrogen Receptor ◽

Bone Mass ◽

Cortical Bone ◽

Estrogen Receptor Alpha ◽

Receptor Alpha ◽

Cortical Bone Mass

Download Full-text

Faculty Opinions recommendation of Spontaneous airway hyperresponsiveness in estrogen receptor-alpha-deficient mice.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1049341.501250 ◽

2006 ◽

Author(s):

Charles Irvin

Keyword(s):

Estrogen Receptor ◽

Airway Hyperresponsiveness ◽

Estrogen Receptor Alpha ◽

Receptor Alpha ◽

Download Full-text

Faculty Opinions recommendation of Silencing of estrogen receptor alpha in the ventromedial nucleus of hypothalamus leads to metabolic syndrome.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1071026.551964 ◽

2007 ◽

Author(s):

Andrea Gore

Keyword(s):

Metabolic Syndrome ◽

Estrogen Receptor ◽

Estrogen Receptor Alpha ◽

Ventromedial Nucleus ◽

Download Full-text

Faculty Opinions recommendation of Amphiregulin is an essential mediator of estrogen receptor alpha function in mammary gland development.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1070943.523901 ◽

2007 ◽

Author(s):

Charles Streuli

Keyword(s):

Estrogen Receptor ◽

Mammary Gland ◽

Estrogen Receptor Alpha ◽

Mammary Gland Development ◽

Receptor Alpha ◽

Gland Development ◽

Download Full-text

Faculty Opinions recommendation of Estrogen prevents bone loss via estrogen receptor alpha and induction of Fas ligand in osteoclasts.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1091028.544409 ◽

2007 ◽

Author(s):

David Moore

Keyword(s):

Estrogen Receptor ◽

Bone Loss ◽

Estrogen Receptor Alpha ◽

Download Full-text