ScienceGate
Advanced Search
Author Search
Journal Finder
Blog
Sign in / Sign up
ScienceGate
Search
Author Search
Journal Finder
Blog
Sign in / Sign up
Abstract 3239: Discovery and biological characterization of ON108600, a small molecule inhibitor of protein kinase CK2.
Mapping Intimacies
◽
10.1158/1538-7445.am2013-3239
◽
2013
◽
Author(s):
Amol Padgaonkar
◽
Olga Rechkoblit
◽
Stephen Cosenza
◽
Venkat R. Pallela
◽
Venkata Subbaiah DRC
◽
...
Keyword(s):
Protein Kinase
◽
Small Molecule
◽
Protein Kinase Ck2
◽
Small Molecule Inhibitor
◽
Biological Characterization
◽
Molecule Inhibitor
◽
Kinase Ck2
Download Full-text
Related Documents
Cited By
References
Effect of CX-4945, a selective bioavailable small molecule inhibitor of protein kinase CK2, on gemcitabine antitumor activity in A2780 ovarian cancer.
Journal of Clinical Oncology
◽
10.1200/jco.2010.28.15_suppl.e13522
◽
2010
◽
Vol 28
(15_suppl)
◽
pp. e13522-e13522
◽
Cited By ~ 3
Author(s):
K. L. Anderes
◽
N. Streiner
◽
M. Omori
◽
N. Huser
◽
C. Ho
◽
...
Keyword(s):
Ovarian Cancer
◽
Protein Kinase
◽
Antitumor Activity
◽
Small Molecule
◽
Protein Kinase Ck2
◽
Small Molecule Inhibitor
◽
Molecule Inhibitor
◽
Kinase Ck2
Download Full-text
Abstract C39: Phase I clinical trial of CX‐4945: A first‐in‐class orally administered small molecule inhibitor of protein kinase CK2
10.1158/1535-7163.targ-09-c39
◽
2009
◽
Cited By ~ 2
Author(s):
Robert F. Marschke
◽
Eleni Andreopoulou
◽
Daniel D. Von Hoff
◽
John K.C. Lim
◽
Claire S. Padgett
◽
...
Keyword(s):
Clinical Trial
◽
Protein Kinase
◽
Phase I
◽
Small Molecule
◽
Protein Kinase Ck2
◽
Small Molecule Inhibitor
◽
Phase I Clinical Trial
◽
Molecule Inhibitor
◽
Kinase Ck2
Download Full-text
Abstract 3765: Discovery and biological characterization of CX-8184, a potent inhibitor of protein kinase CK2
10.1158/1538-7445.am2012-3765
◽
2012
◽
Author(s):
Denis Drygin
◽
Joshua Bliesath
◽
Nanni Huser
◽
Chris Proffitt
◽
Adam Siddiqui-Jain
◽
...
Keyword(s):
Protein Kinase
◽
Protein Kinase Ck2
◽
Potent Inhibitor
◽
Biological Characterization
◽
Kinase Ck2
Download Full-text
Identification and Characterization of a Small-Molecule Inhibitor of Death-Associated Protein Kinase 1
ChemBioChem
◽
10.1002/cbic.201402512
◽
2014
◽
Vol 16
(1)
◽
pp. 59-63
◽
Cited By ~ 13
Author(s):
Theis S. Wilbek
◽
Tine Skovgaard
◽
Fiona J. Sorrell
◽
Stefan Knapp
◽
Jens Berthelsen
◽
...
Keyword(s):
Protein Kinase
◽
Small Molecule
◽
Small Molecule Inhibitor
◽
Molecule Inhibitor
◽
Death Associated Protein Kinase
◽
Identification And Characterization
Download Full-text
Faculty Opinions recommendation of Identification and characterization of a small molecule inhibitor of formin-mediated actin assembly.
Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature
◽
10.3410/f.1283961.751061
◽
2009
◽
Author(s):
Marie-France Carlier
Keyword(s):
Small Molecule
◽
Small Molecule Inhibitor
◽
Actin Assembly
◽
Molecule Inhibitor
◽
Identification And Characterization
Download Full-text
A Novel Small-Molecule Inhibitor of Protein Kinase D Blocks Pancreatic Cancer Growth In vitro and In vivo
Molecular Cancer Therapeutics
◽
10.1158/1535-7163.mct-09-1145
◽
2010
◽
Vol 9
(5)
◽
pp. 1136-1146
◽
Cited By ~ 95
Author(s):
Kuzhuvelil B. Harikumar
◽
Ajaikumar B. Kunnumakkara
◽
Nobuo Ochi
◽
Zhimin Tong
◽
Amit Deorukhkar
◽
...
Keyword(s):
Pancreatic Cancer
◽
Protein Kinase
◽
Small Molecule
◽
Small Molecule Inhibitor
◽
Cancer Growth
◽
Protein Kinase D
◽
Molecule Inhibitor
Download Full-text
Biological characterization of AT7519, a small-molecule inhibitor of cyclin-dependent kinases, in human tumor cell lines
Molecular Cancer Therapeutics
◽
10.1158/1535-7163.mct-08-0890
◽
2009
◽
Vol 8
(2)
◽
pp. 324-332
◽
Cited By ~ 84
Author(s):
Matthew S. Squires
◽
Ruth E. Feltell
◽
Nicola G. Wallis
◽
E. Jonathan Lewis
◽
Donna-Michelle Smith
◽
...
Keyword(s):
Tumor Cell
◽
Small Molecule
◽
Human Tumor
◽
Tumor Cell Lines
◽
Biological Characterization
◽
Human Tumor Cell
◽
Human Tumor Cell Lines
◽
Cyclin Dependent Kinases
◽
Molecule Inhibitor
Download Full-text
Abstract LB-209: Identification and characterization of small molecule inhibitor of Wnt canonical pathway in a glioma setting.
10.1158/1538-7445.am2012-lb-209
◽
2012
◽
Author(s):
Alessandra De Robertis
◽
Silvia Valensin
◽
Marco Rossi
◽
Margherita Verani
◽
Patrizia Tunici
◽
...
Keyword(s):
Small Molecule
◽
Small Molecule Inhibitor
◽
Canonical Pathway
◽
Molecule Inhibitor
◽
Identification And Characterization
Download Full-text
Abstract 3228: Characterization of a novel, orally bioavailable, potent and highly selective small molecule inhibitor of PERK: A tool to probe the biphasic concentration-dependent induction of ER stress in models of multiple myeloma and B-cell lymphoma
10.1158/1538-7445.am2014-3228
◽
2014
◽
Author(s):
Ian Stansfield
◽
Yannick Ligny
◽
Yvan Simonnet
◽
Christophe Demestre
◽
Nathalie Amblard
◽
...
Keyword(s):
Multiple Myeloma
◽
Er Stress
◽
B Cell
◽
Small Molecule
◽
Cell Lymphoma
◽
B Cell Lymphoma
◽
Small Molecule Inhibitor
◽
Molecule Inhibitor
◽
Orally Bioavailable
Download Full-text
Abstract 4484: Discovery and in vitro characterization of AMG 510–a potent and selective covalent small-molecule inhibitor of KRASG12C
10.1158/1538-7445.sabcs18-4484
◽
2019
◽
Cited By ~ 1
Author(s):
Anne Y. Saiki
◽
Kevin Gaida
◽
Karen Rex
◽
Pragathi Achanta
◽
Tisha San Miguel
◽
...
Keyword(s):
Small Molecule
◽
Small Molecule Inhibitor
◽
In Vitro Characterization
◽
Molecule Inhibitor
Download Full-text
Sign in / Sign up
Close
Export Citation Format
Close
Share Document
Close