Synthesis, Structure–Activity Relationships and In Vitro Toxicity Profile of Lactose-Based Fatty Acid Monoesters as Possible Drug Permeability Enhancers

Pharmaceutics ◽

10.3390/pharmaceutics10030081 ◽

2018 ◽

Vol 10 (3) ◽

pp. 81 ◽

Author(s):

Simone Lucarini ◽

Laura Fagioli ◽

Robert Cavanagh ◽

Wanling Liang ◽

Diego Perinelli ◽

...

Keyword(s):

In Vitro Toxicity ◽

Toxicity Profile ◽

Drug Permeability ◽

Structure Activity Relationships ◽

Structure Activity ◽

Permeability Enhancers

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In vitro toxicity of several dithiocarbamates and structure-activity relationships

Journal of Applied Toxicology ◽

10.1002/jat.868 ◽

2002 ◽

Vol 22 (6) ◽

pp. 353-357 ◽

Author(s):

N. Segovia ◽

G. Crovetto ◽

P. Lardelli ◽

M. Espigares

Keyword(s):

In Vitro Toxicity ◽

Structure Activity Relationships ◽

Structure Activity

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Risk Assessment of High-Energy Chemicals by in Vitro Toxicity Screening and Quantitative Structure-Activity Relationships

Toxicological Sciences ◽

10.1093/toxsci/68.2.498 ◽

2002 ◽

Vol 68 (2) ◽

pp. 498-507 ◽

Author(s):

S. Trohalaki

Keyword(s):

Risk Assessment ◽

High Energy ◽

In Vitro Toxicity ◽

Toxicity Screening ◽

Quantitative Structure ◽

Structure Activity Relationships ◽

Structure Activity ◽

Quantitative Structure Activity Relationships

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Graphene-Based Materials In Vitro Toxicity and Their Structure–Activity Relationships: A Systematic Literature Review

Chemical Research in Toxicology ◽

10.1021/acs.chemrestox.1c00243 ◽

2021 ◽

Vol 34 (9) ◽

pp. 2003-2018

Author(s):

Salma Achawi ◽

Jérémie Pourchez ◽

Bruno Feneon ◽

Valérie Forest

Keyword(s):

Literature Review ◽

Systematic Literature Review ◽

In Vitro Toxicity ◽

Structure Activity Relationships ◽

Structure Activity

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Synthesis and structure-activity relationships of pyrimidine derivatives as potent and orally active FGFR3 inhibitors with both increased systemic exposure and enhanced in vitro potency

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2021.116019 ◽

2021 ◽

Vol 33 ◽

pp. 116019

Author(s):

Ikumi Kuriwaki ◽

Minoru Kameda ◽

Kazuhiko Iikubo ◽

Hiroyuki Hisamichi ◽

Yuichiro Kawamoto ◽

...

Keyword(s):

Systemic Exposure ◽

Pyrimidine Derivatives ◽

Structure Activity Relationships ◽

Structure Activity ◽

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Aqua mediated synthesis of 2-amino-6-benzothiazol-2-ylsulfanyl-chromenes and its in vitro study, explanation of the structure–activity relationships (SARs) as antibacterial agent

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2010.08.010 ◽

2010 ◽

Vol 45 (11) ◽

pp. 5031-5038 ◽

Author(s):

Mazaahir Kidwai ◽

Roona Poddar ◽

Saurav Bhardwaj ◽

Satendra Singh ◽

Pratibha Mehta Luthra

Keyword(s):

Antibacterial Agent ◽

In Vitro Study ◽

Vitro Study ◽

Structure Activity Relationships ◽

Structure Activity

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Structure-activity relationships of steroids in inducing germinal vesicle breakdown of Atlantic croaker oocytes in vitro

General and Comparative Endocrinology ◽

10.1016/0016-6480(88)90259-6 ◽

1988 ◽

Vol 71 (2) ◽

pp. 307-317 ◽

Author(s):

John M. Trant ◽

Peter Thomas

Keyword(s):

Germinal Vesicle ◽

Atlantic Croaker ◽

Germinal Vesicle Breakdown ◽

Structure Activity Relationships ◽

Structure Activity

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Structure-activity relationships and inhibitory effects of various purine derivatives on the in vitro growth of Plasmodium falciparum11Abbreviations: CDK, cyclin-dependent kinase; CDK1, cyclin-dependent kinase 1; and PfPK, Plasmodium falciparum protein kinase.

Biochemical Pharmacology ◽

10.1016/s0006-2952(01)00644-x ◽

2001 ◽

Vol 62 (3) ◽

pp. 341-348 ◽

Author(s):

Leonie Harmse ◽

Robyn van Zyl ◽

Nathanael Gray ◽

Peter Schultz ◽

Sophie Leclerc ◽

...

Keyword(s):

Plasmodium Falciparum ◽

Protein Kinase ◽

In Vitro Growth ◽

Cyclin Dependent Kinase ◽

Purine Derivatives ◽

Inhibitory Effects ◽

Structure Activity Relationships ◽

Structure Activity ◽

Falciparum Protein

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Structure-Activity Relationships of Acrylate Esters: Reactivity Towards Glutathione and Hydrolysis by Carboxylesterase in Vitro

Advances in Experimental Medicine and Biology - Biological Reactive Intermediates IV ◽

10.1007/978-1-4684-5877-0_42 ◽

1991 ◽

pp. 333-335 ◽

Author(s):

T. J. McCarthy ◽

G. Witz

Keyword(s):

Structure Activity Relationships ◽

Structure Activity ◽

Acrylate Esters

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Structure-activity relationships of cysteine esters and their effects on thiol levels in rat lung in vitro

Biochemical Pharmacology ◽

10.1016/0006-2952(93)90301-c ◽

1993 ◽

Vol 45 (8) ◽

pp. 1605-1612 ◽

Author(s):

M.J. Hobbs ◽

M. Butterworth ◽

G.M. Cohen ◽

D.G. Upshall

Keyword(s):

Rat Lung ◽

Structure Activity Relationships ◽

Structure Activity

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Structure-activity relationships of tetramethylpiperidine-substituted phenazines against Mycobacterium leprae in vitro.

Antimicrobial Agents and Chemotherapy ◽

10.1128/aac.33.11.2004 ◽

1989 ◽

Vol 33 (11) ◽

pp. 2004-2005 ◽

Author(s):

S G Franzblau ◽

K E White ◽

J F O'Sullivan

Keyword(s):

Mycobacterium Leprae ◽

Structure Activity Relationships ◽

Structure Activity

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