Design, synthesis & structure–activity relationships of a new class of antihuman enterovirus D68 & A71 agents

Future Medicinal Chemistry ◽

10.4155/fmc-2017-0268 ◽

2018 ◽

Vol 10 (11) ◽

pp. 1333-1347

Author(s):

Bidyadhar Sethy ◽

Chung-Fan Hsieh ◽

Chieh Yeh ◽

Jim-Tong Horng ◽

Pei-Wen Hsieh

Keyword(s):

Design Synthesis ◽

Structure Activity Relationships ◽

New Class ◽

Structure Activity ◽

Enterovirus D68

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Design, Synthesis, and Structure−Activity Relationships of Alkylcarbamic Acid Aryl Esters, a New Class of Fatty Acid Amide Hydrolase Inhibitors

Journal of Medicinal Chemistry ◽

10.1021/jm021119g ◽

2003 ◽

Vol 46 (12) ◽

pp. 2352-2360 ◽

Author(s):

Giorgio Tarzia ◽

Andrea Duranti ◽

Andrea Tontini ◽

Giovanni Piersanti ◽

Marco Mor ◽

...

Keyword(s):

Fatty Acid Amide Hydrolase ◽

Design Synthesis ◽

Structure Activity Relationships ◽

New Class ◽

Structure Activity ◽

Amide Hydrolase ◽

Fatty Acid Amide

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Design, synthesis and structure-activity relationships of novel N11-, C12- and C13-substituted 15-membered homo-aza-clarithromycin derivatives against various resistant bacteria

Bioorganic Chemistry ◽

10.1016/j.bioorg.2021.104992 ◽

2021 ◽

pp. 104992

Author(s):

Yinhui Qin ◽

Di Song ◽

Yuetai Teng ◽

Xingbang Liu ◽

Panpan Zhang ◽

...

Keyword(s):

Resistant Bacteria ◽

Design Synthesis ◽

Structure Activity Relationships ◽

Structure Activity

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ChemInform Abstract: The Synthesis and Structure-Activity Relationships of 1,3-Diaryl 1,2,4-(4H)-Triazol-5-ones: A New Class of Calcium-Dependent, Large Conductance, Potassium (Maxi-K) Channel Opener Targeted for Urge Urinary Incontinence.

10.1002/chin.200230166 ◽

2010 ◽

Vol 33 (30) ◽

pp. no-no

Author(s):

Piyasena Hewawasam ◽

Matthew Erway ◽

George Thalody ◽

Harvey Weiner ◽

Christopher G. Boissard ◽

...

Keyword(s):

Urinary Incontinence ◽

Urge Urinary Incontinence ◽

K Channel ◽

Structure Activity Relationships ◽

Calcium Dependent ◽

New Class ◽

Structure Activity ◽

Channel Opener ◽

K Channel Opener

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Discovery of small-molecule nonpeptide antagonists of nociceptin/orphanin FQ receptor: The studies of design, synthesis, and structure–activity relationships for (4-arylpiperidine substituted-methyl)-[bicyclic (hetero)cycloalkanobenzene] derivatives

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2016.02.014 ◽

2016 ◽

Vol 114 ◽

pp. 345-364 ◽

Author(s):

Shigeo Hayashi ◽

Katsuyo Ohashi ◽

Sachiko Mihara ◽

Eriko Nakata ◽

Chie Emoto ◽

...

Keyword(s):

Small Molecule ◽

Orphanin Fq ◽

Design Synthesis ◽

Structure Activity Relationships ◽

Structure Activity

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Nicotinamide Derivatives as a New Class of Gastric H+/K+-ATPase Inhibitors. 1. Synthesis and Structure−Activity Relationships ofN-Substituted 2-(Benzhydryl- and benzylsulfinyl)nicotinamides

Journal of Medicinal Chemistry ◽

10.1021/jm9605593 ◽

1997 ◽

Vol 40 (3) ◽

pp. 313-321 ◽

Author(s):

Hideo Terauchi ◽

Akihiko Tanitame ◽

Keiko Tada ◽

Keiji Nakamura ◽

Yasuhiro Seto ◽

...

Keyword(s):

Structure Activity Relationships ◽

New Class ◽

Structure Activity ◽

Atpase Inhibitors ◽

Nicotinamide Derivatives

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Structure-Activity Relationships of MDMA and Related Compounds: A New Class of Psychoactive Agents?

Topics in the Neurosciences - Ecstasy: The Clinical, Pharmacological and Neurotoxicological Effects of the Drug MDMA ◽

10.1007/978-1-4613-1485-1_7 ◽

1990 ◽

pp. 105-131 ◽

Author(s):

David F. Nichols ◽

Robert Oberlender

Keyword(s):

Structure Activity Relationships ◽

New Class ◽

Structure Activity ◽

Related Compounds

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Design, synthesis and structure-activity relationships of novel 15-membered macrolides: Quinolone/quinoline-containing sidechains tethered to the C-6 position of azithromycin acylides

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2020.112222 ◽

2020 ◽

Vol 193 ◽

pp. 112222 ◽

Author(s):

Bing-Zhi Fan ◽

Hiroshi Hiasa ◽

Wei Lv ◽

Scott Brody ◽

Zhao-Yong Yang ◽

...

Keyword(s):

Design Synthesis ◽

Structure Activity Relationships ◽

Structure Activity

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Design, synthesis and structure–activity relationships of new phosphinate inhibitors of MurD

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2005.09.086 ◽

2006 ◽

Vol 16 (2) ◽

pp. 343-348 ◽

Author(s):

Katja Štrancar ◽

Didier Blanot ◽

Stanislav Gobec

Keyword(s):

Design Synthesis ◽

Structure Activity Relationships ◽

Structure Activity

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Design, Synthesis, and Structure−Activity Relationships of Benzophenone-Based Tetraamides as Novel Antibacterial Agents

Journal of Medicinal Chemistry ◽

10.1021/jm900519b ◽

2009 ◽

Vol 52 (16) ◽

pp. 5020-5031 ◽

Author(s):

Sunil K. Vooturi ◽

Chrissy M. Cheung ◽

Michael J. Rybak ◽

Steven M. Firestine

Keyword(s):

Antibacterial Agents ◽

Design Synthesis ◽

Structure Activity Relationships ◽

Structure Activity

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Application of “Hydrogen-Bonding Interaction” in Drug Design. Part 2: Design, Synthesis, and Structure–Activity Relationships of Thiophosphoramide Derivatives as Novel Antiviral and Antifungal Agents

Journal of Agricultural and Food Chemistry ◽

10.1021/acs.jafc.5b02676 ◽

2015 ◽

Vol 63 (43) ◽

pp. 9435-9440 ◽

Author(s):

Aidang Lu ◽

Yuanyuan Ma ◽

Ziwen Wang ◽

Zhenghong Zhou ◽

Qingmin Wang

Keyword(s):

Hydrogen Bonding ◽

Drug Design ◽

Antifungal Agents ◽

Hydrogen Bonding Interaction ◽

Design Synthesis ◽

Structure Activity Relationships ◽

Structure Activity ◽

Bonding Interaction

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