From Structure to Clinical Development: Allosteric Modulation of G Protein-Coupled Receptors - Advances in Pharmacology

Preface

From Structure to Clinical Development: Allosteric Modulation of G Protein-Coupled Receptors - Advances in Pharmacology ◽

10.1016/s1054-3589(20)30037-5 ◽

2020 ◽

pp. xiii-xvii

Author(s):

Christopher J. Langmead

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Copyright

From Structure to Clinical Development: Allosteric Modulation of G Protein-Coupled Receptors - Advances in Pharmacology ◽

10.1016/s1054-3589(20)30034-x ◽

2020 ◽

pp. iv

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Structure-based discovery and development of metabotropic glutamate receptor 5 negative allosteric modulators

From Structure to Clinical Development: Allosteric Modulation of G Protein-Coupled Receptors - Advances in Pharmacology ◽

10.1016/bs.apha.2020.03.001 ◽

2020 ◽

pp. 35-58

Author(s):

Kirstie A. Bennett ◽

John A. Christopher ◽

Benjamin G. Tehan

Keyword(s):

Glutamate Receptor ◽

Metabotropic Glutamate Receptor ◽

Allosteric Modulators ◽

Metabotropic Glutamate Receptor 5 ◽

Metabotropic Glutamate

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Strategies and considerations of G-protein-coupled receptor photopharmacology

From Structure to Clinical Development: Allosteric Modulation of G Protein-Coupled Receptors - Advances in Pharmacology ◽

10.1016/bs.apha.2019.12.001 ◽

2020 ◽

pp. 143-172 ◽

Cited By ~ 1

Author(s):

Alice E. Berizzi ◽

Cyril Goudet

Keyword(s):

G Protein ◽

G Protein Coupled Receptor ◽

G Protein Coupled

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Discovery and pharmacology of the covalent GLP-1 receptor (GLP-1R) allosteric modulator BETP: A novel tool to probe GLP-1R pharmacology

From Structure to Clinical Development: Allosteric Modulation of G Protein-Coupled Receptors - Advances in Pharmacology ◽

10.1016/bs.apha.2020.02.001 ◽

2020 ◽

pp. 173-191

Author(s):

Francis S. Willard ◽

Joseph D. Ho ◽

Kyle W. Sloop

Keyword(s):

Allosteric Modulator

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M1 muscarinic acetylcholine receptors: A therapeutic strategy for symptomatic and disease-modifying effects in Alzheimer's disease?

From Structure to Clinical Development: Allosteric Modulation of G Protein-Coupled Receptors - Advances in Pharmacology ◽

10.1016/bs.apha.2019.12.003 ◽

2020 ◽

pp. 277-310

Author(s):

Miriam Scarpa ◽

Sarah Hesse ◽

Sophie J. Bradley

Keyword(s):

Alzheimer’S Disease ◽

Alzheimer's Disease ◽

Acetylcholine Receptors ◽

Therapeutic Strategy ◽

Muscarinic Acetylcholine Receptors ◽

Muscarinic Acetylcholine ◽

Disease Modifying ◽

M1 Muscarinic

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The function and allosteric control of the human sweet taste receptor

From Structure to Clinical Development: Allosteric Modulation of G Protein-Coupled Receptors - Advances in Pharmacology ◽

10.1016/bs.apha.2020.01.002 ◽

2020 ◽

pp. 59-82

Author(s):

Guy Servant ◽

Terry Kenakin ◽

Lan Zhang ◽

Mark Williams ◽

Nicole Servant

Keyword(s):

Taste Receptor ◽

Sweet Taste ◽

Allosteric Control ◽

Sweet Taste Receptor

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Allosteric modulation of muscarinic receptors in alcohol and substance use disorders

From Structure to Clinical Development: Allosteric Modulation of G Protein-Coupled Receptors - Advances in Pharmacology ◽

10.1016/bs.apha.2020.01.003 ◽

2020 ◽

pp. 233-275

Author(s):

Leigh C. Walker ◽

Andrew J. Lawrence

Keyword(s):

Substance Use ◽

Substance Use Disorders ◽

Muscarinic Receptors ◽

Allosteric Modulation

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RAMPs as allosteric modulators of the calcitonin and calcitonin-like class B G protein-coupled receptors

From Structure to Clinical Development: Allosteric Modulation of G Protein-Coupled Receptors - Advances in Pharmacology ◽

10.1016/bs.apha.2020.01.001 ◽

2020 ◽

pp. 115-141 ◽

Cited By ~ 2

Author(s):

Augen A. Pioszak ◽

Debbie L. Hay

Keyword(s):

G Protein ◽

G Protein Coupled Receptors ◽

Allosteric Modulators ◽

Class B ◽

G Protein Coupled

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Allosteric modulation of metabotropic glutamate receptors in alcohol use disorder: Insights from preclinical investigations

From Structure to Clinical Development: Allosteric Modulation of G Protein-Coupled Receptors - Advances in Pharmacology ◽

10.1016/bs.apha.2020.02.002 ◽

2020 ◽

pp. 193-232

Author(s):

Kari A. Johnson ◽

David M. Lovinger

Keyword(s):

Alcohol Use ◽

Glutamate Receptors ◽

Alcohol Use Disorder ◽

Metabotropic Glutamate Receptors ◽

Allosteric Modulation ◽

Metabotropic Glutamate

Download Full-text

From Structure to Clinical Development: Allosteric Modulation of G Protein-Coupled Receptors - Advances in Pharmacology
Latest Publications

TOTAL DOCUMENTS

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Published By Elsevier

Preface

Copyright

Structure-based discovery and development of metabotropic glutamate receptor 5 negative allosteric modulators

Strategies and considerations of G-protein-coupled receptor photopharmacology

Discovery and pharmacology of the covalent GLP-1 receptor (GLP-1R) allosteric modulator BETP: A novel tool to probe GLP-1R pharmacology

M1 muscarinic acetylcholine receptors: A therapeutic strategy for symptomatic and disease-modifying effects in Alzheimer's disease?

The function and allosteric control of the human sweet taste receptor

Allosteric modulation of muscarinic receptors in alcohol and substance use disorders

RAMPs as allosteric modulators of the calcitonin and calcitonin-like class B G protein-coupled receptors

Allosteric modulation of metabotropic glutamate receptors in alcohol use disorder: Insights from preclinical investigations

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From Structure to Clinical Development: Allosteric Modulation of G Protein-Coupled Receptors - Advances in PharmacologyLatest Publications

TOTAL DOCUMENTS

H-INDEX

Published By Elsevier

Preface

Copyright

Structure-based discovery and development of metabotropic glutamate receptor 5 negative allosteric modulators

Strategies and considerations of G-protein-coupled receptor photopharmacology

Discovery and pharmacology of the covalent GLP-1 receptor (GLP-1R) allosteric modulator BETP: A novel tool to probe GLP-1R pharmacology

M1 muscarinic acetylcholine receptors: A therapeutic strategy for symptomatic and disease-modifying effects in Alzheimer's disease?

The function and allosteric control of the human sweet taste receptor

Allosteric modulation of muscarinic receptors in alcohol and substance use disorders

RAMPs as allosteric modulators of the calcitonin and calcitonin-like class B G protein-coupled receptors

Allosteric modulation of metabotropic glutamate receptors in alcohol use disorder: Insights from preclinical investigations

From Structure to Clinical Development: Allosteric Modulation of G Protein-Coupled Receptors - Advances in Pharmacology
Latest Publications