ChemInform Abstract: Facile One-Pot Synthesis of Novel 3-Substituted-1,6-dihydro-1,2,4-triazin-5-(2H)-ones from Fatty Acid Hydrazides and Their in vitro Antimicrobial Activity.

ChemInform ◽  
2011 ◽  
Vol 42 (31) ◽  
pp. no-no
Author(s):  
Nida Nayyar Farshori ◽  
Mudasir Rashid Banday ◽  
Anis Ahmad ◽  
Asad Ullah Khan ◽  
Abdul Rauf
Keyword(s):  
Antimicrobial Activity ◽  
Fatty Acid ◽  
One Pot ◽  
In Vitro Antimicrobial Activity ◽  
One Pot Synthesis

PTSA-Catalyzed One Pot Domino Synthesis of Dihydropyrido[2,3-d]pyrimidine Derivatives and their Antimicrobial Activity

2021 ◽  
Vol 6 (3) ◽  
pp. 222-227
Author(s):  
Krishna A. Bhensdadia ◽  
Prakash L. Kalavadiya ◽  
Nilam H. Lalavani ◽  
Shipra H. Baluja
Keyword(s):  
Antimicrobial Activity ◽  
Spectral Analysis ◽  
Pyrimidine Derivatives ◽  
One Pot ◽  
In Vitro Antimicrobial Activity ◽  
Aryl Aldehydes ◽  
Three Component Reaction ◽  
The One

A novel series of dihydropyrido[2,3-d]pyrimidine derivatives were synthesized by multicomponent domino cyclization via the one-pot three component reaction of 6-amino uracil, substituted aryl aldehydes and N-methyl-1-(methylthio)-2-nitroethenamine in the presence of PTSA 10 mol% as a catalyst. The structures of these synthesized compounds were characterized by spectral analysis. Further the synthesized compounds screened for in vitro antimicrobial activity. Among all the compounds, compound 4b containing flouro substitution exhibited good inhibition against the tested species.

scholarly journals Microwave Assisted One Pot Synthesis of Tetrazole Based 3-hydroxy-4H-chromen-4-ones by modified Algar-Flynn-Oyamada reaction and their Antimicrobial activity

2019 ◽  
Vol 63 (4) ◽  
Author(s):  
ASHOK DONGAMANTI ◽  
Nagaraju Nalaparaju ◽  
Sarasija Madderla ◽  
Vijaya Lakshmi Bommidi
Keyword(s):  
Escherichia Coli ◽  
Antimicrobial Activity ◽  
Klebsiella Pneumonia ◽  
Good Activity ◽  
One Pot ◽  
Microwave Assisted ◽  
One Pot Synthesis ◽  
Antimicrobial Studies ◽  
The One

In the present work, we report the one pot synthesis of tetrazole based 3-hydroxy-4H-chromen-4-ones 3(a-g) from  4-(1H-tetrazol-5-yl)benzaldehyde and 2-hydroxy acetophenone using KOH and H2O2 by modified Algar-Flynn-Oyamada reaction under conventional and microwave irradiation conditions. In this technique, flavonols are synthesized without isolating chalcones, in good yields. All the synthesized compounds were characterized by IR, NMR, MS and elemental. All newly synthesized compounds were screened for their in-vitro antimicrobial activity against strains such as Staphylococcus aurous, Bacillus subtilis, Klebsiella pneumonia, Escherichia coli, Aspergillus Niger, Aspergillus flavus, and Fusarium oxysporum. The results of antimicrobial studies revealed that most of the compounds exhibit good activity.

Synthesis and characterization of novel fatty acid analogs of cholesterol: In vitro antimicrobial activity

2010 ◽  
Vol 45 (4) ◽  
pp. 1459-1464 ◽  
Author(s):  
Mudasir R. Banday ◽  
Nida N. Farshori ◽  
Anis Ahmad ◽  
Asad U. Khan ◽  
Abdul Rauf
Keyword(s):  
Antimicrobial Activity ◽  
Fatty Acid ◽  
Synthesis And Characterization ◽  
In Vitro Antimicrobial Activity

Synthesis and evaluation of in vitro antimicrobial activity of novel 2,3-disubstituted-4-thiazolidinones from fatty acid hydrazides

2012 ◽  
Vol 22 (7) ◽  
pp. 3204-3212 ◽  
Author(s):  
Himani Varshney ◽  
Aiman Ahmad ◽  
Nida N. Farshori ◽  
Anis Ahmad ◽  
Asad U. Khan ◽  
...  
Keyword(s):  
Antimicrobial Activity ◽  
Fatty Acid ◽  
In Vitro Antimicrobial Activity

Synthesis of novel 1,4-disubstituted 1,2,3-triazolo-bosentan derivatives – evaluation of antimicrobial and anticancer activities and molecular docking

RSC Advances ◽  
2015 ◽  
Vol 5 (127) ◽  
pp. 105266-105278 ◽  
Author(s):  
K. Easwaramoorthi ◽  
A. Jeya Rajendran ◽  
K. Chennakesava Rao ◽  
Y. Arun ◽  
C. Balachandran ◽  
...  
Keyword(s):  
Antimicrobial Activity ◽  
Molecular Docking ◽  
Anticancer Activity ◽  
Cell Lines ◽  
Anticancer Activities ◽  
One Pot ◽  
One Pot Synthesis

One pot synthesis with good yields. Good antimicrobial activity against 4EMV receptor. Prominent anticancer activity against A549 and SKOV-3 cell lines. Significantin vitrocytotoxicity at 7.81 μg mL−1. Docking mode of1hwith 2XP2 receptor.

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