Design, synthesis, biological evaluation, structure-activity relationship, and toxicity of clinafloxacin-azole conjugates as novel antitubercular agents

2019 ◽  
Vol 27 (1) ◽  
pp. 175-187 ◽  
Author(s):  
Jie Liu ◽  
Zhenghong Ren ◽  
Li Fan ◽  
Jianyong Wei ◽  
Xuemei Tang ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Activity Relationship ◽  
Antitubercular Agents ◽  
Design Synthesis ◽  
Structure Activity

Novel 2-(2-phenalkyl)-1H-benzo[d]imidazoles as antitubercular agents. Synthesis, biological evaluation and structure–activity relationship

2015 ◽  
Vol 23 (9) ◽  
pp. 2112-2120 ◽  
Author(s):  
Katarzyna Gobis ◽  
Henryk Foks ◽  
Karolina Suchan ◽  
Ewa Augustynowicz-Kopeć ◽  
Agnieszka Napiórkowska ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Activity Relationship ◽  
Antitubercular Agents ◽  
Structure Activity

Design, synthesis and biological evaluation of novel peptide MC2 analogues from Momordica charantia as potential anti-diabetic agents

2015 ◽  
Vol 13 (15) ◽  
pp. 4551-4561 ◽  
Author(s):  
Baowei Yang ◽  
Xue Li ◽  
Chenyu Zhang ◽  
Sijia Yan ◽  
Wei Wei ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Momordica Charantia ◽  
Activity Relationship ◽  
Design Synthesis ◽  
Structure Activity ◽  
Oxidative Effects ◽  
Relationship Of ◽  
Synthesis And Biological Evaluation

The structure–activity relationship of peptide MC2 resulted in the development of compoundIII-3, which exhibited potent anti-hyperglycaemic and anti-oxidative effects.

Benzo[d]thiazole-2-carbanilides as new anti-TB chemotypes: Design, synthesis, biological evaluation, and structure-activity relationship

2018 ◽  
Vol 155 ◽  
pp. 364-380 ◽  
Author(s):  
Tejas M. Dhameliya ◽  
Rishu Tiwari ◽  
Arkaprabha Banerjee ◽  
Sahaj Pancholia ◽  
Dharmarajan Sriram ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Activity Relationship ◽  
Design Synthesis ◽  
Structure Activity

Design, Synthesis, and Structure–Activity Relationship Studies of Tryptanthrins As Antitubercular Agents

2013 ◽  
Vol 76 (3) ◽  
pp. 354-367 ◽  
Author(s):  
Jae-Min Hwang ◽  
Taegwon Oh ◽  
Takushi Kaneko ◽  
Anna M. Upton ◽  
Scott G. Franzblau ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Antitubercular Agents ◽  
Design Synthesis ◽  
Structure Activity
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