Design, Synthesis, Biological Evaluation, and Structure−Activity Relationship (SAR) Discussion of Dipeptidyl Boronate Proteasome Inhibitors, Part I: Comprehensive Understanding of the SAR of α-Amino Acid Boronates

2009 ◽  
Vol 52 (14) ◽  
pp. 4192-4199 ◽  
Author(s):  
Yongqiang Zhu ◽  
Xin Zhao ◽  
Xinrong Zhu ◽  
Gang Wu ◽  
Yuejie Li ◽  
...  
Keyword(s):  
Amino Acid ◽  
Proteasome Inhibitors ◽  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Activity Relationship ◽  
Comprehensive Understanding ◽  
Design Synthesis ◽  
Structure Activity

Design, synthesis and biological evaluation of novel peptide MC2 analogues from Momordica charantia as potential anti-diabetic agents

2015 ◽  
Vol 13 (15) ◽  
pp. 4551-4561 ◽  
Author(s):  
Baowei Yang ◽  
Xue Li ◽  
Chenyu Zhang ◽  
Sijia Yan ◽  
Wei Wei ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Momordica Charantia ◽  
Activity Relationship ◽  
Design Synthesis ◽  
Structure Activity ◽  
Oxidative Effects ◽  
Relationship Of ◽  
Synthesis And Biological Evaluation

The structure–activity relationship of peptide MC2 resulted in the development of compoundIII-3, which exhibited potent anti-hyperglycaemic and anti-oxidative effects.

Benzo[d]thiazole-2-carbanilides as new anti-TB chemotypes: Design, synthesis, biological evaluation, and structure-activity relationship

2018 ◽  
Vol 155 ◽  
pp. 364-380 ◽  
Author(s):  
Tejas M. Dhameliya ◽  
Rishu Tiwari ◽  
Arkaprabha Banerjee ◽  
Sahaj Pancholia ◽  
Dharmarajan Sriram ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Biological Evaluation ◽  
Activity Relationship ◽  
Design Synthesis ◽  
Structure Activity
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