3′-Methoxy-4′-nitroflavone, a reported aryl hydrocarbon receptor antagonist, enhances Cyp1a1 transcription by a dioxin responsive element-dependent mechanism

Aryl Hydrocarbon ◽

Responsive Element ◽

Aryl Hydrocarbon Receptor Antagonist ◽

Dependent Mechanism

1057 Vemurafenib acts as an aryl hydrocarbon receptor antagonist

Journal of Investigative Dermatology ◽

10.1016/j.jid.2018.03.1070 ◽

2018 ◽

Vol 138 (5) ◽

pp. S179

Author(s):

H.C. Hawerkamp ◽

A. Kislat ◽

P. Gerber ◽

M. Pollet ◽

A.A. Soshilov ◽

...

Keyword(s):

Receptor Antagonist ◽

Aryl Hydrocarbon ◽

The aryl hydrocarbon receptor antagonist, 3′methoxy-4′nitroflavone, attenuates 2,3,7,8-tetrachlorodibenzo-p-dioxin-dependent regulation of growth factor signaling and apoptosis in the MCF-10A cell line

Toxicology and Applied Pharmacology ◽

10.1016/s0041-008x(03)00012-7 ◽

2003 ◽

Vol 188 (1) ◽

pp. 42-49 ◽

Cited By ~ 25

Author(s):

John W Davis ◽

Andrew D Burdick ◽

Fredine T Lauer ◽

Scott W Burchiel

Keyword(s):

Growth Factor ◽

Receptor Antagonist ◽

Cell Line ◽

Growth Factor Signaling ◽

Aryl Hydrocarbon ◽

Tetrachlorodibenzo P Dioxin ◽

Regulation Of Growth ◽

In Silico Identification of an Aryl Hydrocarbon Receptor Antagonist with Biological Activity In Vitro and In Vivo

Molecular Pharmacology ◽

10.1124/mol.114.093369 ◽

2014 ◽

Vol 86 (5) ◽

pp. 593-608 ◽

Cited By ~ 23

Author(s):

Ashley J. Parks ◽

Michael P. Pollastri ◽

Mark E. Hahn ◽

Elizabeth A. Stanford ◽

Olga Novikov ◽

...

Keyword(s):

Biological Activity ◽

Receptor Antagonist ◽

In Silico ◽

Aryl Hydrocarbon ◽

In Silico Identification ◽

The New Aryl Hydrocarbon Receptor Antagonist E/Z-2-Benzylindene-5,6-Dimethoxy-3,3-Dimethylindan-1-One Protects against UVB-Induced Signal Transduction

Journal of Investigative Dermatology ◽

10.1038/jid.2013.362 ◽

2014 ◽

Vol 134 (2) ◽

pp. 556-559 ◽

Cited By ~ 35

Author(s):

Julia Tigges ◽

Thomas Haarmann-Stemmann ◽

Christoph F.A. Vogel ◽

Annemarie Grindel ◽

Ulrike Hübenthal ◽

...

Keyword(s):

Signal Transduction ◽

Receptor Antagonist ◽

Aryl Hydrocarbon ◽

Induced Signal ◽

In vivoeffects of the pure aryl hydrocarbon receptor antagonist GNF-351 after oral administration are limited to the gastrointestinal tract

British Journal of Pharmacology ◽

10.1111/bph.12576 ◽

2014 ◽

Vol 171 (7) ◽

pp. 1735-1746 ◽

Cited By ~ 13

Author(s):

Zhong-Ze Fang ◽

Kristopher W Krausz ◽

Kenjiro Nagaoka ◽

Naoki Tanaka ◽

Krishne Gowda ◽

...

Keyword(s):

Gastrointestinal Tract ◽

Oral Administration ◽

Receptor Antagonist ◽

Aryl Hydrocarbon ◽

The Aryl Hydrocarbon Receptor Antagonist StemRegenin 1 Promotes Human Plasmacytoid and Myeloid Dendritic Cell Development from CD34+ Hematopoietic Progenitor Cells

Stem Cells and Development ◽

10.1089/scd.2013.0521 ◽

2014 ◽

Vol 23 (9) ◽

pp. 955-967 ◽

Cited By ~ 35

Author(s):

Soley Thordardottir ◽

Basav N. Hangalapura ◽

Tim Hutten ◽

Marta Cossu ◽

Jan Spanholtz ◽

...

Keyword(s):

Dendritic Cell ◽

Receptor Antagonist ◽

Progenitor Cells ◽

Cell Development ◽

Hematopoietic Progenitor Cells ◽

Myeloid Dendritic Cell ◽

Hematopoietic Progenitor ◽

Aryl Hydrocarbon ◽

Fluoranthene-Induced Cytotoxicity and Direct Effect of Aryl Hydrocarbon Receptor Antagonist on Hematopoietic Stem Cell Differentiation

Annals of Laboratory Medicine ◽

10.3343/alm.2019.39.6.580 ◽

2019 ◽

Vol 39 (6) ◽

pp. 580-583

Author(s):

Seung-Hyun Yang ◽

Min-Gu Kang ◽

Hye-Ran Kim ◽

Young Eun Lee ◽

Bo Ram Na ◽

...

Keyword(s):

Stem Cell ◽

Cell Differentiation ◽

Receptor Antagonist ◽

Direct Effect ◽

Stem Cell Differentiation ◽

Hematopoietic Stem ◽

Aryl Hydrocarbon ◽

Hematopoietic Stem Cell Differentiation ◽

Development of an Aryl Hydrocarbon Receptor Antagonist Using the Proteolysis-Targeting Chimeric Molecules Approach: A Potential Tool for Chemoprevention

Molecular Pharmacology ◽

10.1124/mol.107.040840 ◽

2008 ◽

Vol 73 (4) ◽

pp. 1064-1071 ◽

Cited By ~ 46

Author(s):

Dinesh Puppala ◽

Hyosung Lee ◽

Kyung Bo Kim ◽

Hollie I. Swanson

Keyword(s):

Receptor Antagonist ◽

Aryl Hydrocarbon ◽

Chimeric Molecules ◽

Potential Tool ◽

Mgta-456, Cord Blood CD34+ Cells Expanded with an Aryl Hydrocarbon Receptor Antagonist, Enhances Human Microglia Engraftment in the Brains of NSG Mice

Biology of Blood and Marrow Transplantation ◽

10.1016/j.bbmt.2017.12.031 ◽

2018 ◽

Vol 24 (3) ◽

pp. S115-S116

Author(s):

Kevin A. Goncalves ◽

Megan D. Hoban ◽

Jennifer L. Proctor ◽

Sharon L. Hyzy ◽

Katia S. George ◽

...

Keyword(s):

Cord Blood ◽

Receptor Antagonist ◽

Human Microglia ◽

Aryl Hydrocarbon ◽

Nsg Mice ◽

Cd34 Cells ◽

Cord Blood Cd34 ◽

Vemurafenib acts as an aryl hydrocarbon receptor antagonist: Implications for inflammatory cutaneous adverse events

Allergy ◽

10.1111/all.13972 ◽

2019 ◽

Vol 74 (12) ◽

pp. 2437-2448 ◽

Cited By ~ 5

Author(s):

Heike C. Hawerkamp ◽

Andreas Kislat ◽

Peter A. Gerber ◽

Marius Pollet ◽

Katharina M. Rolfes ◽

...

Keyword(s):

Adverse Events ◽

Receptor Antagonist ◽

Aryl Hydrocarbon ◽