Structure–Activity Relationship between the in Vivo Skin Sensitizing Potency of Analogues of Phenyl Glycidyl Ether and the Induction of Nrf2-Dependent Luciferase Activity in the KeratinoSens in Vitro Assay

In Vitro Assay ◽

Activity Relationship ◽

Phenyl Glycidyl Ether ◽

Vitro Assay ◽

STRUCTURE-ACTIVITY RELATIONSHIP OF VARIOUS ANALOGUES OF β-CORTICOTRROPHIN DETERMINED BY REFERENCE TO VARIOUS PARAMETERS IN VITRO AND IN VIVO

Acta Endocrinologica ◽

10.1530/acta.0.061s029 ◽

1969 ◽

Vol 61 (1_Suppl) ◽

pp. S29

Author(s):

Pierre A. Desaulles ◽

René Maier ◽

Matthys Staehelin

Keyword(s):

Activity Relationship ◽

Structure Activity ◽

Relationship Of

The selective 5-HT2A receptor agonist 25CN-NBOH: Structure-activity relationship, in vivo pharmacology, and in vitro and ex vivo binding characteristics of [3H]25CN-NBOH

Biochemical Pharmacology ◽

10.1016/j.bcp.2020.113979 ◽

2020 ◽

Vol 177 ◽

pp. 113979 ◽

Cited By ~ 3

Author(s):

Anders A. Jensen ◽

Adam L. Halberstadt ◽

Emil Märcher-Rørsted ◽

Anna U. Odland ◽

Muhammad Chatha ◽

...

Keyword(s):

Receptor Agonist ◽

Ex Vivo ◽

Activity Relationship ◽

Binding Characteristics ◽

Radiochemical Investigations of99mTc−N3S-X-BBN[7−14]NH2: An in Vitro/in Vivo Structure−Activity Relationship Study Where X = 0-, 3-, 5-, 8-, and 11-Carbon Tethering Moieties

Bioconjugate Chemistry ◽

10.1021/bc020034r ◽

2003 ◽

Vol 14 (1) ◽

pp. 93-102 ◽

Cited By ~ 63

Author(s):

C. Jeffrey Smith ◽

Hariprasad Gali ◽

Gary L. Sieckman ◽

Chris Higginbotham ◽

Wynn A. Volkert ◽

...

Keyword(s):

Activity Relationship ◽

Structure Activity ◽

Relationship Study

Discovery and Structure−Activity Relationship of Antagonists of B-Cell Lymphoma 2 Family Proteins with Chemopotentiation Activity in Vitro and in Vivo

10.1021/jm050754u ◽

2006 ◽

Vol 49 (3) ◽

pp. 1165-1181 ◽

Cited By ~ 94

Author(s):

Michael D. Wendt ◽

Wang Shen ◽

Aaron Kunzer ◽

William J. McClellan ◽

Milan Bruncko ◽

...

Keyword(s):

B Cell ◽

Cell Lymphoma ◽

B Cell Lymphoma ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Of

Synthesis, in Vitro and in Vivo Biological Evaluation, Docking Studies, and Structure−Activity Relationship (SAR) Discussion of Dipeptidyl Boronic Acid Proteasome Inhibitors Composed of β-Amino Acids

10.1021/jm901407s ◽

2010 ◽

Vol 53 (5) ◽

pp. 1990-1999 ◽

Cited By ~ 29

Author(s):

Yongqiang Zhu ◽

Xinrong Zhu ◽

Gang Wu ◽

Yuheng Ma ◽

Yuejie Li ◽

...

Keyword(s):

Amino Acids ◽

Boronic Acid ◽

Proteasome Inhibitors ◽

Docking Studies ◽

Biological Evaluation ◽

Activity Relationship ◽

Structure–Activity Relationship Studies of Pyrazolo[3,4-d]pyrimidine Derivatives Leading to the Discovery of a Novel Multikinase Inhibitor That Potently Inhibits FLT3 and VEGFR2 and Evaluation of Its Activity against Acute Myeloid Leukemia in Vitro and in Vivo

10.1021/jm301537p ◽

2013 ◽

Vol 56 (4) ◽

pp. 1641-1655 ◽

Cited By ~ 43

Author(s):

Ling-Ling Yang ◽

Guo-Bo Li ◽

Shuang Ma ◽

Chan Zou ◽

Shu Zhou ◽

...

Keyword(s):

Acute Myeloid Leukemia ◽

Myeloid Leukemia ◽

Activity Relationship ◽

Pyrimidine Derivatives ◽

Multikinase Inhibitor ◽

Structure Activity ◽

Acute Myeloid

Synthesis, in vitro structure–activity relationship, and in vivo studies of 2-arylthiazolidine-4-carboxylic acid amides as anticancer agents

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2009.12.020 ◽

2010 ◽

Vol 18 (2) ◽

pp. 477-495 ◽

Cited By ~ 19

Author(s):

Yan Lu ◽

Zhao Wang ◽

Chien-Ming Li ◽

Jianjun Chen ◽

James T. Dalton ◽

...

Keyword(s):

Carboxylic Acid ◽

Anticancer Agents ◽

In Vivo Studies ◽

Activity Relationship ◽

Structure Activity ◽

Carboxylic Acid Amides

Structure-activity relationship studies and in vitro and in vivo anticancer activity of novel 3-aroyl-1,4-diarylpyrroles against solid tumors and hematological malignancies

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2019.111828 ◽

2020 ◽

Vol 185 ◽

pp. 111828 ◽

Cited By ~ 1

Author(s):

Michela Puxeddu ◽

Hongliang Shen ◽

Ruoli Bai ◽

Antonio Coluccia ◽

Marianna Nalli ◽

...

Keyword(s):

Anticancer Activity ◽

Solid Tumors ◽

Hematological Malignancies ◽

Activity Relationship ◽

In Vitro Structure−Activity Relationship and in Vivo Studies for a Novel Class of Cyclooxygenase-2 Inhibitors: 5-Aryl-2,2-dialkyl-4-phenyl-3(2H)furanone Derivatives

10.1021/jm020545z ◽

2004 ◽

Vol 47 (4) ◽

pp. 792-804 ◽

Cited By ~ 56

Author(s):

Song Seok Shin ◽

Youngjoo Byun ◽

Kyung Min Lim ◽

Jin Kyu Choi ◽

Ki-Wha Lee ◽

...

Keyword(s):

Cyclooxygenase 2 ◽

In Vivo Studies ◽

Activity Relationship ◽

Structure Activity ◽

Cyclooxygenase 2 Inhibitors

Impact of a Heteroatom in a Structure−Activity Relationship Study on Analogues of Phenyl Glycidyl Ether (PGE) from Epoxy Resin Systems

Chemical Research in Toxicology ◽

10.1021/tx100417r ◽

2011 ◽

Vol 24 (4) ◽

pp. 542-548 ◽

Cited By ~ 13

Author(s):

Ida B. Niklasson ◽

Tamara Delaine ◽

Kristina Luthman ◽

Ann-Therese Karlberg

Keyword(s):

Epoxy Resin ◽

Glycidyl Ether ◽

Activity Relationship ◽

Phenyl Glycidyl Ether ◽

Structure Activity ◽

Relationship Study