scholarly journals Modulation of Opioid Receptor Ligand Affinity and Efficacy Using Active and Inactive State Receptor Models

2012 ◽  
Vol 80 (5) ◽  
pp. 763-770 ◽  
Author(s):  
Jessica P. Anand ◽  
Lauren C. Purington ◽  
Irina D. Pogozheva ◽  
John R. Traynor ◽  
Henry I. Mosberg
Keyword(s):  
Opioid Receptor ◽  
Receptor Ligand ◽  
Ligand Affinity ◽  
Inactive State ◽  
Receptor Models

scholarly journals Effects of the novel, selective and low-efficacy mu opioid receptor ligand NAQ on intracranial self-stimulation in rats

2014 ◽  
Vol 232 (4) ◽  
pp. 815-824 ◽  
Author(s):  
Ahmad A. Altarifi ◽  
Yunyun Yuan ◽  
Yan Zhang ◽  
Dana E. Selley ◽  
S. Stevens Negus
Keyword(s):  
Opioid Receptor ◽  
Mu Opioid Receptor ◽  
The Novel ◽  
Receptor Ligand ◽  
Mu Opioid ◽  
Self Stimulation

Structure of the cannabinoid receptor 1: homology modeling of its inactive state and enrichment study based on CB1 antagonist docking

MedChemComm ◽  
2014 ◽  
Vol 5 (9) ◽  
pp. 1297-1302 ◽  
Author(s):  
Haining Liu ◽  
Ronak Y. Patel ◽  
Robert J. Doerksen
Keyword(s):  
Homology Modeling ◽  
Cannabinoid Receptor ◽  
Cannabinoid Receptor 1 ◽  
Inactive State ◽  
Receptor Models ◽  
Cannabinoid 1 Receptor ◽  
Cb1 Antagonist

Multiple cannabinoid 1 receptor models were prepared and the best one was selected based on the models' performance in selecting known ligands from a pool of competitors.

[125I][D-Ala2]deltorphin-I: A high affinity, delta-selective opioid receptor ligand

Peptides ◽  
1991 ◽  
Vol 12 (4) ◽  
pp. 825-830 ◽  
Author(s):  
Sylvie Dupin ◽  
Jean-Andre M. Tafani ◽  
Honoré Mazarguil ◽  
Jean-Marie Zajac
Keyword(s):  
Opioid Receptor ◽  
Receptor Ligand ◽  
High Affinity

scholarly journals Oncolytic potency of HER-2 retargeted VSV-FH hybrid viruses: the role of receptor ligand affinity

2015 ◽  
Vol 2 ◽  
pp. 15012 ◽  
Author(s):  
Camilo Ayala Breton ◽  
Nitwara Wikan ◽  
Arinda Abbuhl ◽  
Duncan R Smith ◽  
Stephen J Russell ◽  
...  
Keyword(s):  
Receptor Ligand ◽  
Ligand Affinity ◽  
Her 2

scholarly journals Homology modeling of opioid receptor-ligand complexes using experimental constraints

2005 ◽  
Vol 7 (2) ◽  
pp. E434-E448 ◽  
Author(s):  
Irina D. Pogozheva ◽  
Magdalena J. Przydzial ◽  
Henry I. Mosberg
Keyword(s):  
Homology Modeling ◽  
Opioid Receptor ◽  
Receptor Ligand
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