Enlargement of a Modular System—Synthesis and Characterization of an s-Triazine-Based Carboxylic Acid Ester Bearing a Galactopyranosyl Moiety and an Enormous Boron Load
Keyword(s):
The amount of boron accumulated in tumor tissue plays an important role regarding the success of the boron neutron capture therapy (BNCT). In this article, we report a modular system, combining readily available starting materials, like glycine, 1,3,5-triazine and the well-known 9-mercapto-1,7-dicarba-closo-dodecaborane(12), as well as α-d-galactopyranose for increased hydrophilicity, with a novel boron-rich tris-meta-carboranyl thiol.
2008 ◽
pp. 238-249
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1996 ◽
Vol 11
(4)
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pp. 263-285
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2017 ◽
Vol 107
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pp. 217-229
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2009 ◽
Vol 206
(6)
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pp. 1361-1364
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2010 ◽