scholarly journals Herbicidal activity of fluoroquinolone derivatives

Plant Direct ◽  
2021 ◽  
Vol 5 (9) ◽  
Author(s):  
Michael D. Wallace ◽  
Aleksandra W. Debowski ◽  
Kirill V. Sukhoverkov ◽  
Joshua S. Mylne ◽  
Keith A. Stubbs
Keyword(s):  
Herbicidal Activity ◽  
Fluoroquinolone Derivatives

scholarly journals Herbicidal activity of fluoroquinolone derivatives

2021 ◽  
Author(s):  
Michael D Wallace ◽  
Aleksandra W Debowski ◽  
Kirill V Sukhoverkov ◽  
Joshua S Mylne ◽  
Keith A Stubbs
Keyword(s):  
Antibacterial Activity ◽  
Dna Gyrase ◽  
Herbicidal Activity ◽  
Amino Group ◽  
Gram Negative Bacteria ◽  
Gram Negative ◽  
Structural Modifications ◽  
Weak Antibacterial Activity ◽  
Insight Into ◽  
Fluoroquinolone Derivatives

Development of herbicides with novel modes of action are crucial for weed control and to hinder herbicide resistance. An attractive novel herbicidal target is plant DNA gyrase, which has been demonstrated to be effectively inhibited by the known antimicrobial ciprofloxacin. Despite this good herbicidal activity ciprofloxacin is not suitable as a herbicide due to its antimicrobial activity, therefore, a diverse library of analogues was analysed to gain insight into the aspects required for herbicidal activity. This analysis revealed significant structural modifications were tolerated and that the fluoride at C-6 and a cyclic amino group at C-7 were not crucial for herbicidal activity. The analysis also revealed that these modifications also affected the antibacterial activity with one compound demonstrating good herbicidal activity and weak antibacterial activity, against both Gram-positive and Gram-negative bacteria.

Influence of Absolute Configuration of Indanofan on Herbicidal Activity

2001 ◽  
Vol 26 (4) ◽  
pp. 383-384 ◽  
Author(s):  
Akemi HOSOKAWA ◽  
Osamu IKEDA ◽  
Chizuko SASAKI ◽  
Yasuko T. OSANO ◽  
Tetsuo JIKIHARA
Keyword(s):  
Absolute Configuration ◽  
Herbicidal Activity

Chemical structure and herbicidal activity of .ALPHA.,.ALPHA.-dialkylbenzyl containing thiolcarbamate compounds.

1989 ◽  
Vol 34 (1) ◽  
pp. 27-36
Author(s):  
Kaoru IKEDA ◽  
Kiyoshi SUGAYA
Keyword(s):  
Chemical Structure ◽  
Herbicidal Activity

Toxicity, Uptake, and Distribution of Simazine in Canna hybrida `King Humbert': Implications for Phytoremediation

HortScience ◽  
1998 ◽  
Vol 33 (3) ◽  
pp. 484e-485
Author(s):  
Patrick C. Wilson ◽  
Ted Whitwell ◽  
Steven J. Klaine
Keyword(s):  
Mass Production ◽  
Photosynthetic Efficiency ◽  
Liquid Scintillation ◽  
Herbicidal Activity ◽  
Fresh Mass ◽  
Contaminated Water ◽  
Golf Courses ◽  
Plant Tolerance ◽  
Nutrient Media ◽  
Potential Use

This research focuses on the potential use of Canna hybrida `King Humbert' for removing simazine from contaminated water generated at golf courses and ornamental nurseries. Because of simazine's herbicidal activity, it is important for levels in solution not to exceed plant tolerance levels. Tolerance levels for C. hybrida were determined by dosing plants for 7 d with 0, 0.01, 0.03, 0.1, 0.3, 1.0, or 3.0 mg simazine/L nutrient media. Measurements of 7-d fresh mass production and photosynthetic efficiency (Fv/Fm) were taken. Simazine uptake and distribution within the plant was determined by dosing plants with 2.03 mCi 14C-simazine (0.243 mg/L) for 1, 3, 5, or 7 d. Plant tissues were analyzed by combustion and liquid scintillation counting. Fresh mass production was reduced 66% and 78% for plants exposed to 1.0 and 3.0 mg/L, respectively. Likewise, photosynthetic efficiency was reduced to 66% and 40% of the controls at the same respective concentrations. Plant uptake of simazine accounted for 13%, 34%, 48%, and 65% of the original simazine in the dosing solution after 1-, 3-, 5-, and 7-d exposure, respectively. This simazine was distributed primarily between roots and leaves.

An Insight into Patents of Fluoroquinolone Derivatives

2015 ◽  
Vol 12 (10) ◽  
pp. 844-855
Author(s):  
Prabodh Chander Sharma ◽  
Mona Piplani ◽  
Harish Rajak
Keyword(s):  
Insight Into ◽  
Fluoroquinolone Derivatives

Antibacterial Activity of Lipophilic Fluoroquinolone Derivatives

2009 ◽  
Vol 5 (5) ◽  
pp. 419-421 ◽  
Author(s):  
Camila de Almeida ◽  
Claudio Diniz ◽  
Vania Silva ◽  
Mauricio Saraiva ◽  
Mireille Le Hyaric ◽  
...  
Keyword(s):  
Antibacterial Activity ◽  
Fluoroquinolone Derivatives

Preliminary Screening of Isolated Mycoherbicidal Fungi for the Management of Noxious Weed Xanthiumstrumarium

2019 ◽  
Vol 6 (02) ◽  
Author(s):  
AJAY KUMAR SINGH ◽  
AKHILESH KUMAR PANDEY
Keyword(s):  
Culture Filtrate ◽  
Photosynthetic Pigment ◽  
Phytopathogenic Fungi ◽  
Herbicidal Activity ◽  
Preliminary Screening ◽  
Detached Leaf ◽  
Noxious Weed ◽  
Complete Collapse

Natural phytotoxins of fungi are great source for the discovery of new herbicide and its offer a benign and eco-friendly alternative to manage weed. Thus, this study aimed to select potential fungi with potent herbicidal activity for control ofweeds. In the present study, various phytopathogenic fungi were isolated from infected tissues of various weeds and evaluated againstXanthium strumarium, a problematic monocotyledonous weed of open lands, agriculture, horticulture and forests. Herbicidal potential of Cell Free Culture Filtrate (CFCF) of strains ofPhoma herbarum (FGCCW#18, FGCCW#43) Fusariummonilifromecoded as FGCCW#35 and Fusarium roseum coded as FGCCW#55againstXanthium strumariumwere evaluated by seedling and shoot cut bioassays. Maximum mortalities of shoots, seedlings and phytotoxic damage were obtainedfrom28 day sold cell free culture filtrate (CFCF) of FGCCW#18 at 100% concentration. Significant reduction in biological contents i.e. photosynthetic pigment and protein was observed in the host weed on treatment with the CFCF as determined by detached leaf bioassay. Phytotoxic damage such as severe wilting, chlorosis, necrosis and complete collapse of the entire parts of the weed were also noticed due to CFCF application.

scholarly journals Discovery, characterization and functional improvement of kumamonamide as a novel plant growth inhibitor that disturbs plant microtubules

2021 ◽  
Vol 11 (1) ◽  
Author(s):  
Takashi Ishida ◽  
Haruna Yoshimura ◽  
Masatsugu Takekawa ◽  
Takumi Higaki ◽  
Takashi Ideue ◽  
...  
Keyword(s):  
Plant Growth ◽  
Human Life ◽  
Growth Inhibitor ◽  
Herbicidal Activity ◽  
Functional Improvement ◽  
Microtubule Inhibitors ◽  
Plant Microtubules ◽  
Plant Growth Inhibitor ◽  
Derivatives Of ◽  
Synthetic Intermediate

AbstractThe discovery and useful application of natural products can help improve human life. Chemicals that inhibit plant growth are broadly utilized as herbicides to control weeds. As various types of herbicides are required, the identification of compounds with novel modes of action is desirable. In the present study, we discovered a novelN-alkoxypyrrole compound, kumamonamide fromStreptomyces werraensisMK493-CF1 and established a total synthesis procedure. Resulted in the bioactivity assays, we found that kumamonamic acid, a synthetic intermediate of kumamonamide, is a potential plant growth inhibitor. Further, we developed various derivatives of kumamonamic acid, including a kumamonamic acid nonyloxy derivative (KAND), which displayed high herbicidal activity without adverse effects on HeLa cell growth. We also detected that kumamonamic acid derivatives disturb plant microtubules; and additionally, that KAND affected actin filaments and induced cell death. These multifaceted effects differ from those of known microtubule inhibitors, suggesting a novel mode of action of kumamonamic acid, which represents an important lead for the development of new herbicides.

Synthesis, herbicidal activity study and molecular docking of novel pyrimidine thiourea

2020 ◽  
pp. 104766
Author(s):  
Jia-hui Li ◽  
Yan Wang ◽  
Yun-peng Wu ◽  
Ran-hong Li ◽  
Shuang Liang ◽  
...  
Keyword(s):  
Molecular Docking ◽  
Herbicidal Activity

Synthesis, Crystal Structure, Herbicidal Activity, and SAR Study of Novel N-(Arylmethoxy)-2-chloronicotinamides Derived from Nicotinic Acid

2021 ◽  
Author(s):  
Chen-Sheng Yu ◽  
Qiao Wang ◽  
Joanna Bajsa-Hirschel ◽  
Charles L. Cantrell ◽  
Stephen O. Duke ◽  
...  
Keyword(s):  
Crystal Structure ◽  
Nicotinic Acid ◽  
Herbicidal Activity ◽  
Sar Study
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