Structure-based design and synthesis of conformationally constrained derivatives of methyl-piperidinopyrazole (MPP) with estrogen receptor (ER) antagonist activity

2021 ◽  
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Mahmoud A. Ragab ◽  
Mohamed Elagawany ◽  
Hoda Daabees ◽  
Al-Shaimaa F. Ahmed ◽  
Eman M. Awad ◽  
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Estrogen Receptor ◽  
Antagonist Activity ◽  
Conformationally Constrained ◽  
Design And Synthesis ◽  
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Design and Synthesis of Novel 20(S)-α-aminophosphonate Derivatives of Camptothecin as Potent Antitumor Agents

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pp. 105065
Author(s):  
Yu-Yuan Chen ◽  
Yin-Peng Bai ◽  
Bin Li ◽  
Xiao-Bo Zhao ◽  
Cheng-Jie Yang ◽  
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Antitumor Agents ◽  
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Design and synthesis of herboxidiene derivatives that potently inhibit in vitro splicing

2021 ◽  
Vol 19 (6) ◽  
pp. 1365-1377
Author(s):  
Arun K. Ghosh ◽  
Srinivasa Rao Allu ◽  
Guddeti Chandrashekar Reddy ◽  
Adriana Gamboa Lopez ◽  
Patricia Mendez ◽  
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Biological Evaluation ◽  
Design And Synthesis ◽  
In Vitro Splicing ◽  
Enantioselective Syntheses ◽  
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Enantioselective syntheses of C-6 modified derivatives of herboxidiene and their biological evaluation in splicing inhibitory assay.

Design and synthesis of carborane-containing estrogen receptor-beta (ERβ)-selective ligands

2015 ◽  
Vol 25 (19) ◽  
pp. 4174-4178 ◽  
Author(s):  
Kiminori Ohta ◽  
Takumi Ogawa ◽  
Akifumi Oda ◽  
Asako Kaise ◽  
Yasuyuki Endo
Keyword(s):  
Estrogen Receptor ◽  
Estrogen Receptor Beta ◽  
Design And Synthesis ◽  
Selective Ligands ◽  
Receptor Beta

ChemInform Abstract: Design and Synthesis of Conformationally Constrained Arginal Thrombin Inhibitors.

ChemInform ◽  
2010 ◽  
Vol 29 (1) ◽  
pp. no-no
Author(s):  
A. SALIMBENI ◽  
F. PALEARI ◽  
R. CANEVOTTI ◽  
M. CRISCUOLI ◽  
A. LIPPI ◽  
...  
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Thrombin Inhibitors ◽  
Conformationally Constrained ◽  
Design And Synthesis

Novel, Potent, and Orally Active Substance P Antagonists: Synthesis and Antagonist Activity of N-Benzylcarboxamide Derivatives of Pyrido[3,4-b]pyridine

1995 ◽  
Vol 38 (16) ◽  
pp. 3106-3120 ◽  
Author(s):  
Hideaki Natsugari ◽  
Yoshinori Ikeura ◽  
Yutaka Kiyota ◽  
Yuji Ishichi ◽  
Takenori Ishimaru ◽  
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Substance P ◽  
Active Substance ◽  
Antagonist Activity ◽  
Substance P Antagonists ◽  
Orally Active ◽  
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Design and synthesis of novel water-soluble amino acid derivatives of chlorin p6 ethers as photosensitizer

2019 ◽  
Vol 30 (1) ◽  
pp. 247-249 ◽  
Author(s):  
Xingjie Zhang ◽  
Zhi Meng ◽  
Zhiqiang Ma ◽  
Junhong Liu ◽  
Guiyan Han ◽  
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Keyword(s):  
Amino Acid ◽  
Water Soluble ◽  
Amino Acid Derivatives ◽  
Design And Synthesis ◽  
Derivatives Of ◽  
Chlorin P6
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