Structure-activity relationship study of a series of caspase inhibitors containing γ-amino acid moiety for treatment of cholestatic liver disease

Activity Relationship ◽

Cholestatic Liver Disease ◽

Acid Moiety ◽

Caspase Inhibitors ◽

Structure Activity ◽

Amino Acid Moiety ◽

Isolation of 8′-Phosphate Ester Derivatives of Amicoumacins: Structure-activity Relationship of Hydroxy Amino Acid Moiety

The Journal of Antibiotics ◽

10.1038/ja.2007.99 ◽

2007 ◽

Vol 60 (12) ◽

pp. 752-756 ◽

Cited By ~ 20

Author(s):

Makoto Hashimoto ◽

Takaaki Taguchi ◽

Satoshi Nishida ◽

Kouji Ueno ◽

Kaio Koizumi ◽

...

Keyword(s):

Amino Acid ◽

Activity Relationship ◽

Phosphate Ester ◽

Acid Moiety ◽

Hydroxy Amino Acid ◽

Structure Activity ◽

Amino Acid Moiety ◽

Relationship Of ◽

Derivatives Of

ChemInform Abstract: Isolation of 8′-Phosphate Ester Derivatives of Amicoumacins: Structure-Activity Relationship of Hydroxy Amino Acid Moiety.

ChemInform ◽

10.1002/chin.200826218 ◽

2008 ◽

Vol 39 (26) ◽

Author(s):

Makoto Hashimoto ◽

Takaaki Taguchi ◽

Satoshi Nishida ◽

Kouji Ueno ◽

Kaio Koizumi ◽

...

Keyword(s):

Amino Acid ◽

Activity Relationship ◽

Phosphate Ester ◽

Acid Moiety ◽

Hydroxy Amino Acid ◽

Structure Activity ◽

Amino Acid Moiety ◽

Relationship Of ◽

Derivatives Of

Identification and Structure–Activity Relationship Study of Imidazo[1,2-a]pyridine-3-amines as First Selective Inhibitors of Excitatory Amino Acid Transporter Subtype 3 (EAAT3)

ACS Chemical Neuroscience ◽

10.1021/acschemneuro.9b00447 ◽

2019 ◽

Vol 10 (10) ◽

pp. 4414-4429

Author(s):

Peng Wu ◽

Walden E. Bjørn-Yoshimoto ◽

Markus Staudt ◽

Anders A. Jensen ◽

Lennart Bunch

Keyword(s):

Amino Acid ◽

Excitatory Amino Acid ◽

Amino Acid Transporter ◽

Activity Relationship ◽

Selective Inhibitors ◽

Excitatory Amino Acid Transporter ◽

Structure Activity ◽

Relationship Study ◽

Subtype 3

Structure-activity-relationship study of N-acyl-N-phenylpiperazines as potential inhibitors of the Excitatory Amino Acid Transporters (EAATs): improving the potency of a micromolar screening Hit is not truism

SpringerPlus ◽

10.1186/2193-1801-2-112 ◽

2013 ◽

Vol 2 (1) ◽

pp. 112

Author(s):

Tri HV Huynh ◽

Charles S Demmer ◽

Bjarke Abrahamsen ◽

Emil Marcher ◽

Mikael Frykman ◽

...

Keyword(s):

Amino Acid ◽

Excitatory Amino Acid ◽

Activity Relationship ◽

Amino Acid Transporters ◽

Excitatory Amino Acid Transporters ◽

Structure Activity ◽

Relationship Study ◽

Potential Inhibitors

Structure–activity relationship study of compounds binding to large amino acid transporter 1 (LAT1) based on pharmacophore modeling and in situ rat brain perfusion

European Journal of Pharmaceutical Sciences ◽

10.1016/j.ejps.2012.11.014 ◽

2013 ◽

Vol 48 (3) ◽

pp. 523-531 ◽

Cited By ~ 26

Author(s):

Henna Ylikangas ◽

Lauri Peura ◽

Kalle Malmioja ◽

Jukka Leppänen ◽

Krista Laine ◽

...

Keyword(s):

Amino Acid ◽

Rat Brain ◽

Brain Perfusion ◽

Amino Acid Transporter ◽

Pharmacophore Modeling ◽

Activity Relationship ◽

Structure Activity ◽

Structure-activity relationship study on artificial CXCR4 ligands possessing the cyclic pentapeptide scaffold: the exploration of amino acid residues of pentapeptides by substitutions of several aromatic amino acids

Organic & Biomolecular Chemistry ◽

10.1039/b908286g ◽

2009 ◽

Vol 7 (18) ◽

pp. 3805 ◽

Cited By ~ 12

Author(s):

Tomohiro Tanaka ◽

Wataru Nomura ◽

Tetsuo Narumi ◽

Ai Esaka ◽

Shinya Oishi ◽

...

Keyword(s):

Amino Acids ◽

Amino Acid ◽

Aromatic Amino Acids ◽

Activity Relationship ◽

Amino Acid Residues ◽

Structure Activity ◽

Structure−Activity Relationship Study of First Selective Inhibitor of Excitatory Amino Acid Transporter Subtype 1: 2-Amino-4-(4-methoxyphenyl)-7-(naphthalen-1-yl)-5-oxo-5,6,7,8-tetrahydro-4H-chromene-3-carbonitrile (UCPH-101)

Journal of Medicinal Chemistry ◽

10.1021/jm1009154 ◽

2010 ◽

Vol 53 (19) ◽

pp. 7180-7191 ◽

Cited By ~ 82

Author(s):

Mette N. Erichsen ◽

Tri H. V. Huynh ◽

Bjarke Abrahamsen ◽

Jesper F. Bastlund ◽

Christoffer Bundgaard ◽

...

Keyword(s):

Amino Acid ◽

Excitatory Amino Acid ◽

Amino Acid Transporter ◽

Selective Inhibitor ◽

Activity Relationship ◽

Excitatory Amino Acid Transporter ◽

Structure Activity ◽

Relationship Study ◽

Acid Transporter

Structure-activity relationship study of antioxidative peptides by QSAR modeling: the amino acid next to C -terminus affects the activity

Journal of Peptide Science ◽

10.1002/psc.1345 ◽

2011 ◽

Vol 17 (6) ◽

pp. 454-462 ◽

Cited By ~ 39

Author(s):

Yao-Wang Li ◽

Bo Li ◽

Jiguo He ◽

Ping Qian

Keyword(s):

Amino Acid ◽

Activity Relationship ◽

Qsar Modeling ◽

Structure Activity ◽

C Terminus ◽

Identification of a New Class of Selective Excitatory Amino Acid Transporter Subtype 1 (EAAT1) Inhibitors Followed by a Structure–Activity Relationship Study

Journal of Medicinal Chemistry ◽

10.1021/acs.jmedchem.6b01058 ◽

2016 ◽

Vol 59 (19) ◽

pp. 8757-8770 ◽

Cited By ~ 11

Author(s):

Stinne W. Hansen ◽

Mette N. Erichsen ◽

Bingru Fu ◽

Walden E. Bjørn-Yoshimoto ◽

Bjarke Abrahamsen ◽

...

Keyword(s):

Amino Acid ◽

Excitatory Amino Acid ◽

Amino Acid Transporter ◽

Activity Relationship ◽

Excitatory Amino Acid Transporter ◽

New Class ◽

Structure Activity ◽

Relationship Study ◽

Acid Transporter

Extensive Structure–Activity Relationship Study of Albicidin's C‐Terminal Dipeptidic p ‐Aminobenzoic Acid Moiety

Chemistry - A European Journal ◽

10.1002/chem.201904752 ◽

2019 ◽

Vol 25 (72) ◽

pp. 16538-16543 ◽

Cited By ~ 3

Author(s):

Iraj Behroz ◽

Patrick Durkin ◽

Stefan Grätz ◽

Maria Seidel ◽

Lida Rostock ◽

...

Keyword(s):

Activity Relationship ◽

Aminobenzoic Acid ◽

Acid Moiety ◽

Structure Activity ◽