Furans with basic side chains: synthesis and biological evaluation of a novel series of antagonists with selectivity for the estrogen receptor alpha

Deborah S. Mortensen; Alice L. Rodriguez; Jun Sun; Benita S. Katzenellenbogen; John A. Katzenellenbogen

doi:10.1016/s0960-894x(01)00488-7

Furans with basic side chains: synthesis and biological evaluation of a novel series of antagonists with selectivity for the estrogen receptor alpha

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(01)00488-7 ◽

2001 ◽

Vol 11 (18) ◽

pp. 2521-2524 ◽

Cited By ~ 33

Author(s):

Deborah S. Mortensen ◽

Alice L. Rodriguez ◽

Jun Sun ◽

Benita S. Katzenellenbogen ◽

John A. Katzenellenbogen

Keyword(s):

Estrogen Receptor ◽

Estrogen Receptor Alpha ◽

Biological Evaluation ◽

Side Chains ◽

Receptor Alpha ◽

Synthesis And Biological Evaluation

Download Full-text

ChemInform Abstract: Furans with Basic Side Chains: Synthesis and Biological Evaluation of a Novel Series of Antagonists with Selectivity for the Estrogen Receptor Alpha.

ChemInform ◽

10.1002/chin.200206112 ◽

2010 ◽

Vol 33 (6) ◽

pp. no-no

Author(s):

Deborah S. Mortensen ◽

Alice L. Rodriguez ◽

Jun Sun ◽

Benita S. Katzenellenbogen ◽

John A. Katzenellenbogen

Keyword(s):

Estrogen Receptor ◽

Estrogen Receptor Alpha ◽

Biological Evaluation ◽

Side Chains ◽

Receptor Alpha ◽

Synthesis And Biological Evaluation

Download Full-text

Design, synthesis and biological evaluation of novel indole-benzimidazole hybrids targeting estrogen receptor alpha (ER-α)

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2018.01.051 ◽

2018 ◽

Vol 146 ◽

pp. 206-219 ◽

Cited By ~ 13

Author(s):

Ramit Singla ◽

Kunj Bihari Gupta ◽

Shishir Upadhyay ◽

Monisha Dhiman ◽

Vikas Jaitak

Keyword(s):

Estrogen Receptor ◽

Estrogen Receptor Alpha ◽

Biological Evaluation ◽

Design Synthesis ◽

Receptor Alpha ◽

Synthesis And Biological Evaluation

Download Full-text

Physicochemical Characteristics and Preliminary in Vivo Biological Evaluation of Nanocapsules Loaded with siRNA Targeting Estrogen Receptor Alpha

Biomacromolecules ◽

10.1021/bm800664c ◽

2008 ◽

Vol 9 (10) ◽

pp. 2881-2890 ◽

Cited By ~ 31

Author(s):

Céline Bouclier ◽

Laurence Moine ◽

Hervé Hillaireau ◽

Véronique Marsaud ◽

Elisabeth Connault ◽

...

Keyword(s):

Estrogen Receptor ◽

Estrogen Receptor Alpha ◽

Physicochemical Characteristics ◽

Biological Evaluation ◽

Receptor Alpha

Download Full-text

Author response for "Estrogen receptor alpha, g‐protein coupled receptor 1, and aromatase: developmental, sex, and region‐specific differences across the rat caudate‐putamen, nucleus accumbens core and shell"

10.1002/cne.24978/v4/response1 ◽

2020 ◽

Author(s):

Amanda A. Krentzel ◽

Jaime A. Willett ◽

Ashlyn G. Johnson ◽

John Meitzen

Keyword(s):

Estrogen Receptor ◽

Nucleus Accumbens ◽

G Protein ◽

Estrogen Receptor Alpha ◽

Author Response ◽

G Protein Coupled Receptor ◽

Nucleus Accumbens Core ◽

Caudate Putamen ◽

Receptor Alpha ◽

G Protein Coupled

Download Full-text

Author response for "Estrogen receptor alpha, g‐protein coupled receptor 1, and aromatase: developmental, sex, and region‐specific differences across the rat caudate‐putamen, nucleus accumbens core and shell"

10.1002/cne.24978/v3/response1 ◽

2020 ◽

Author(s):

Amanda A. Krentzel ◽

Jaime A. Willett ◽

Ashlyn G. Johnson ◽

John Meitzen

Keyword(s):

Estrogen Receptor ◽

Nucleus Accumbens ◽

G Protein ◽

Estrogen Receptor Alpha ◽

Author Response ◽

G Protein Coupled Receptor ◽

Nucleus Accumbens Core ◽

Caudate Putamen ◽

Receptor Alpha ◽

G Protein Coupled

Download Full-text

Die Kaffee-vermittelte Induktion von UDP-Glukuronosyltransferasen wird durch den Estrogen-Receptor-alpha (ESR-1) geschlechtspezifisch reguliert

Zeitschrift für Gastroenterologie ◽

10.1055/s-0031-1285168 ◽

2011 ◽

Vol 49 (08) ◽

Author(s):

S Kalthoff ◽

A Winkler ◽

N Freiberg ◽

M Manns ◽

C Strassburg

Keyword(s):

Estrogen Receptor ◽

Estrogen Receptor Alpha ◽

Receptor Alpha

Download Full-text

Mice lacking estrogen receptor [alpha] in hypothalamic POMC neurons display enhanced estrogenic response on cortical bone mass

Bone Abstracts ◽

10.1530/boneabs.5.ht2 ◽

2016 ◽

Author(s):

Helen Farman ◽

Sara Windahl ◽

Deborah Clegg ◽

Shang Kui Xie ◽

Lars Westberg ◽

...

Keyword(s):

Estrogen Receptor ◽

Bone Mass ◽

Cortical Bone ◽

Estrogen Receptor Alpha ◽

Receptor Alpha ◽

Cortical Bone Mass

Download Full-text

Faculty Opinions recommendation of Spontaneous airway hyperresponsiveness in estrogen receptor-alpha-deficient mice.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1049341.501250 ◽

2006 ◽

Author(s):

Charles Irvin

Keyword(s):

Estrogen Receptor ◽

Airway Hyperresponsiveness ◽

Estrogen Receptor Alpha ◽

Receptor Alpha ◽

Deficient Mice

Download Full-text

Faculty Opinions recommendation of Silencing of estrogen receptor alpha in the ventromedial nucleus of hypothalamus leads to metabolic syndrome.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1071026.551964 ◽

2007 ◽

Author(s):

Andrea Gore

Keyword(s):

Metabolic Syndrome ◽

Estrogen Receptor ◽

Estrogen Receptor Alpha ◽

Ventromedial Nucleus ◽

Receptor Alpha

Download Full-text

Faculty Opinions recommendation of Amphiregulin is an essential mediator of estrogen receptor alpha function in mammary gland development.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1070943.523901 ◽

2007 ◽

Author(s):

Charles Streuli

Keyword(s):

Estrogen Receptor ◽

Mammary Gland ◽

Estrogen Receptor Alpha ◽

Mammary Gland Development ◽

Receptor Alpha ◽

Gland Development ◽

Alpha Function

Download Full-text