Structure-Activity Relationship of N17'-Substituted Norbinaltorphimine Congeners. Role of the N17' Basic Group in the Interaction with a Putative Address Subsite on the .kappa. Opioid Receptor

Kappa Opioid Receptor ◽

Activity Relationship ◽

Kappa Opioid ◽

Basic Group ◽

Structure Activity ◽

Relationship Of

Structure–Activity Relationship Studies of Functionally Selective Kappa Opioid Receptor Agonists that Modulate ERK 1/2 Phosphorylation While Preserving G Protein Over βArrestin2 Signaling Bias

ACS Chemical Neuroscience ◽

10.1021/acschemneuro.5b00092 ◽

2015 ◽

Vol 6 (8) ◽

pp. 1411-1419 ◽

Cited By ~ 36

Author(s):

Kimberly M. Lovell ◽

Kevin J. Frankowski ◽

Edward L. Stahl ◽

Stephen R. Slauson ◽

Euna Yoo ◽

...

Keyword(s):

G Protein ◽

Opioid Receptor ◽

Kappa Opioid Receptor ◽

Activity Relationship ◽

Kappa Opioid ◽

Receptor Agonists ◽

Structure Activity ◽

Design and Synthesis of a Piperidinone Scaffold as an Analgesic through Kappa-Opioid Receptor: Structure–Activity Relationship Study of Matrine Alkaloids

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.c15-00962 ◽

2016 ◽

Vol 64 (5) ◽

pp. 410-419 ◽

Cited By ~ 6

Author(s):

Hiroyoshi Teramoto ◽

Takayasu Yamauchi ◽

Yasushi Terado ◽

Sanae Odagiri ◽

Shigeru Sasaki ◽

...

Keyword(s):

Opioid Receptor ◽

Kappa Opioid Receptor ◽

Activity Relationship ◽

Kappa Opioid ◽

Design And Synthesis ◽

Receptor Structure ◽

Structure Activity ◽

Relationship Study

Structure–activity relationship investigation of triazole-based kappa opioid receptor agonists

Medicinal Chemistry Research ◽

10.1007/s00044-021-02746-1 ◽

2021 ◽

Author(s):

Kevin J. Frankowski ◽

Tarsis Brust ◽

Kimberly M. Lovell ◽

Euna Yoo ◽

Laura M. Bohn ◽

...

Keyword(s):

Opioid Receptor ◽

Kappa Opioid Receptor ◽

Activity Relationship ◽

Kappa Opioid ◽

Receptor Agonists ◽

Structure Activity ◽

Nascent structure–activity relationship study of a diastereomeric series of kappa opioid receptor antagonists derived from CJ-15,208

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2009.04.105 ◽

2009 ◽

Vol 19 (13) ◽

pp. 3647-3650 ◽

Cited By ~ 24

Author(s):

Roland E. Dolle ◽

Mathieu Michaut ◽

Blanca Martinez-Teipel ◽

Pamela R. Seida ◽

Christopher W. Ajello ◽

...

Keyword(s):

Opioid Receptor ◽

Kappa Opioid Receptor ◽

Activity Relationship ◽

Receptor Antagonists ◽

Kappa Opioid ◽

Structure Activity ◽

Opioid Receptor Antagonists ◽

Relationship Study

Structure-Activity Relationship Studies of Dynorphin A Analogs at the Kappa Opioid Receptor

Peptides 2015, Proceedings of the 24th American Peptide Symposium ◽

10.17952/24aps.2015.096 ◽

2015 ◽

Author(s):

Cyf N. Ramos Colon ◽

Yeon Sun Lee ◽

Sara M. Hall ◽

Josephine Lai ◽

Frank Porreca ◽

...

Keyword(s):

Opioid Receptor ◽

Kappa Opioid Receptor ◽

Activity Relationship ◽

Dynorphin A ◽

Kappa Opioid ◽

Structure Activity

Faculty Opinions recommendation of Structure-activity relationship studies of functionally selective kappa opioid receptor agonists that modulate ERK 1/2 phosphorylation while preserving G protein over βarrestin2 signaling bias.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.725444384.793506439 ◽

2015 ◽

Author(s):

John Lowe

Keyword(s):

G Protein ◽

Opioid Receptor ◽

Kappa Opioid Receptor ◽

Activity Relationship ◽

Kappa Opioid ◽

Receptor Agonists ◽

Structure Activity ◽

Correction to “Structure–Activity Relationship Studies of Functionally Selective Kappa Opioid Receptor Agonists that Modulate ERK 1/2 Phosphorylation While Preserving G Protein Over βArrestin2 Signaling Bias”

ACS Chemical Neuroscience ◽

10.1021/acschemneuro.7b00157 ◽

2017 ◽

Vol 8 (7) ◽

pp. 1628-1628

Author(s):

Kimberly M. Lovell ◽

Kevin J. Frankowski ◽

Edward L. Stahl ◽

Stephen R. Slauson ◽

Euna Yoo ◽

...

Keyword(s):

G Protein ◽

Opioid Receptor ◽

Kappa Opioid Receptor ◽

Activity Relationship ◽

Kappa Opioid ◽

Receptor Agonists ◽

Structure Activity ◽

Structure–Activity Relationship of the Antimicrobial Peptide Gomesin: The Role of Peptide Hydrophobicity in Its Interaction with Model Membranes

Langmuir ◽

10.1021/la500146j ◽

2014 ◽

Vol 30 (12) ◽

pp. 3513-3521 ◽

Cited By ~ 27

Author(s):

Bruno Mattei ◽

Antonio Miranda ◽

Katia R. Perez ◽

Karin A. Riske

Keyword(s):

Antimicrobial Peptide ◽

Model Membranes ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Of ◽

Peptide Hydrophobicity

The Role of Dimension in Multivalent Binding Events: Structure-Activity Relationship of Dendritic Polyglycerol Sulfate Binding to L -Selectin in Correlation with Size and Surface Charge Density

Macromolecular Bioscience ◽

10.1002/mabi.201100051 ◽

2011 ◽

Vol 11 (8) ◽

pp. 1088-1098 ◽

Cited By ~ 55

Author(s):

Marie Weinhart ◽

Dominic Gröger ◽

Sven Enders ◽

Sebastian B. Riese ◽

Jens Dernedde ◽

...

Keyword(s):

Charge Density ◽

Surface Charge ◽

Surface Charge Density ◽

Activity Relationship ◽

Structure Activity ◽

Multivalent Binding ◽

Relationship Of

Structure–activity relationship of antioxidant dipeptides: Dominant role of Tyr, Trp, Cys and Met residues

Journal of Functional Foods ◽

10.1016/j.jff.2015.12.003 ◽

2016 ◽

Vol 21 ◽

pp. 485-496 ◽

Cited By ~ 56

Author(s):

Lin Zheng ◽

Yijun Zhao ◽

Hongzhu Dong ◽

Guowan Su ◽

Mouming Zhao

Keyword(s):

Dominant Role ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Of