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Inhibition of Gene Markers of Fibrosis with a Novel Inhibitor of Transforming Growth Factor-β Type I Receptor Kinase in Puromycin-Induced Nephritis
Journal of Pharmacology and Experimental Therapeutics
◽
10.1124/jpet.104.082099
◽
2005
◽
Vol 313
(3)
◽
pp. 943-951
◽
Cited By ~ 120
Author(s):
Eugene T. Grygielko
◽
William M. Martin
◽
Christopher Tweed
◽
Peter Thornton
◽
John Harling
◽
...
Keyword(s):
Growth Factor
◽
Transforming Growth Factor
◽
Transforming Growth Factor Β
◽
Type I
◽
Receptor Kinase
◽
Gene Markers
Download Full-text
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References
A Novel Small-Molecule Inhibitor of Transforming Growth Factor β Type I Receptor Kinase (SM16) Inhibits Murine Mesothelioma Tumor Growth In vivo and Prevents Tumor Recurrence after Surgical Resection
Cancer Research
◽
10.1158/0008-5472.can-06-2389
◽
2007
◽
Vol 67
(5)
◽
pp. 2351-2359
◽
Cited By ~ 72
Author(s):
Eiji Suzuki
◽
Samuel Kim
◽
H.-Kam Cheung
◽
Michael J. Corbley
◽
Xiamei Zhang
◽
...
Keyword(s):
Growth Factor
◽
Tumor Growth
◽
Small Molecule
◽
Tumor Recurrence
◽
Transforming Growth Factor
◽
Transforming Growth Factor Β
◽
Type I
◽
Receptor Kinase
◽
Molecule Inhibitor
Download Full-text
Inhibition of Pulmonary and Skeletal Metastasis by a Transforming Growth Factor-β Type I Receptor Kinase Inhibitor
Cancer Research
◽
10.1158/0008-5472.can-05-3565
◽
2006
◽
Vol 66
(13)
◽
pp. 6714-6721
◽
Cited By ~ 137
Author(s):
Abhik Bandyopadhyay
◽
Joseph K. Agyin
◽
Long Wang
◽
Yuping Tang
◽
Xiufen Lei
◽
...
Keyword(s):
Growth Factor
◽
Transforming Growth Factor
◽
Kinase Inhibitor
◽
Skeletal Metastasis
◽
Transforming Growth Factor Β
◽
Type I
◽
Receptor Kinase
Download Full-text
Small molecule inhibitor of type I transforming growth factor-β receptor kinase ameliorates the inhibitory milieu in injured brain and promotes regeneration of nigrostriatal dopaminergic axons
Journal of Neuroscience Research
◽
10.1002/jnr.22552
◽
2010
◽
Vol 89
(3)
◽
pp. 381-393
◽
Cited By ~ 20
Author(s):
Nozomu Yoshioka
◽
Junko Kimura-Kuroda
◽
Taro Saito
◽
Koki Kawamura
◽
Shin-ichi Hisanaga
◽
...
Keyword(s):
Growth Factor
◽
Small Molecule
◽
Transforming Growth Factor
◽
Transforming Growth Factor Β
◽
Small Molecule Inhibitor
◽
Type I
◽
Receptor Kinase
◽
Molecule Inhibitor
◽
Injured Brain
◽
Β Receptor
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Inhibition of Growth and Metastasis of Mouse Mammary Carcinoma by Selective Inhibitor of Transforming Growth Factor-β Type I Receptor Kinase In vivo
Clinical Cancer Research
◽
10.1158/1078-0432.ccr-06-0162
◽
2006
◽
Vol 12
(14)
◽
pp. 4315-4330
◽
Cited By ~ 102
Author(s):
Rongrong Ge
◽
Vaishali Rajeev
◽
Partha Ray
◽
Edmund Lattime
◽
Susan Rittling
◽
...
Keyword(s):
Growth Factor
◽
Mammary Carcinoma
◽
Transforming Growth Factor
◽
Transforming Growth Factor Β
◽
Selective Inhibitor
◽
Type I
◽
Receptor Kinase
◽
Mouse Mammary Carcinoma
◽
Inhibition Of Growth
Download Full-text
IN-1130, a novel transforming growth factor-β type I receptor kinase (ALK5) inhibitor, suppresses renal fibrosis in obstructive nephropathy
Kidney International
◽
10.1038/sj.ki.5001775
◽
2006
◽
Vol 70
(7)
◽
pp. 1234-1243
◽
Cited By ~ 138
Author(s):
J.-A. Moon
◽
H.-T. Kim
◽
I.-S. Cho
◽
Y.Y. Sheen
◽
D.-K. Kim
Keyword(s):
Growth Factor
◽
Renal Fibrosis
◽
Transforming Growth Factor
◽
Transforming Growth Factor Β
◽
Obstructive Nephropathy
◽
Type I
◽
Receptor Kinase
◽
Alk5 Inhibitor
Download Full-text
Design, synthesis and evaluation of small molecule imidazo[2,1-b][1,3,4]thiadiazoles as inhibitors of transforming growth factor-β type-I receptor kinase (ALK5)
European Journal of Medicinal Chemistry
◽
10.1016/j.ejmech.2014.09.002
◽
2015
◽
Vol 93
◽
pp. 599-613
◽
Cited By ~ 29
Author(s):
Harun M. Patel
◽
Baljeet Sing
◽
Varun Bhardwaj
◽
Mahesh Palkar
◽
Mahamadhanif S. Shaikh
◽
...
Keyword(s):
Growth Factor
◽
Small Molecule
◽
Transforming Growth Factor
◽
Transforming Growth Factor Β
◽
Type I
◽
Receptor Kinase
◽
Design Synthesis
Download Full-text
EW-7197, an oral transforming growth factor β type I receptor kinase inhibitor, for preventing peritoneal adhesion formation in a rat model
Surgery
◽
10.1016/j.surg.2018.07.005
◽
2018
◽
Vol 164
(5)
◽
pp. 1100-1108
◽
Cited By ~ 4
Author(s):
Jiaywei Tsauo
◽
Ho-Young Song
◽
Eun Young Choi
◽
Dae-Kee Kim
◽
Kun Yung Kim
◽
...
Keyword(s):
Growth Factor
◽
Rat Model
◽
Transforming Growth Factor
◽
Kinase Inhibitor
◽
Adhesion Formation
◽
Transforming Growth Factor Β
◽
Type I
◽
Receptor Kinase
◽
Peritoneal Adhesion
◽
Peritoneal Adhesion Formation
Download Full-text
Synthesis and biological evaluation of 5-(fluoro-substituted-6-methylpyridin-2-yl)-4-([1,2,4]triazolo[1,5-a]pyridin-6-yl)imidazoles as inhibitors of transforming growth factor-β type I receptor kinase
Bioorganic & Medicinal Chemistry Letters
◽
10.1016/j.bmcl.2015.09.058
◽
2015
◽
Vol 25
(22)
◽
pp. 5228-5231
◽
Cited By ~ 9
Author(s):
Maddeboina Krishnaiah
◽
Cheng Hua Jin
◽
Yhun Yhong Sheen
◽
Dae-Kee Kim
Keyword(s):
Growth Factor
◽
Transforming Growth Factor
◽
Transforming Growth Factor Β
◽
Biological Evaluation
◽
Type I
◽
Receptor Kinase
◽
Synthesis And Biological Evaluation
Download Full-text
4-([1,2,4]Triazolo[1,5-a]pyridin-6-yl)-5(3)-(6-methylpyridin-2-yl)imidazole and -pyrazole derivatives as potent and selective inhibitors of transforming growth factor-β type I receptor kinase
Bioorganic & Medicinal Chemistry
◽
10.1016/j.bmc.2014.03.022
◽
2014
◽
Vol 22
(9)
◽
pp. 2724-2732
◽
Cited By ~ 12
Author(s):
Cheng Hua Jin
◽
Maddeboina Krishnaiah
◽
Domalapally Sreenu
◽
Vura Bala Subrahmanyam
◽
Hyun-Ju Park
◽
...
Keyword(s):
Growth Factor
◽
Transforming Growth Factor
◽
Transforming Growth Factor Β
◽
Type I
◽
Pyrazole Derivatives
◽
Receptor Kinase
◽
Selective Inhibitors
Download Full-text
Synthesis and activity of new aryl- and heteroaryl-substituted 5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole inhibitors of the transforming growth factor-β type I receptor kinase domain
Bioorganic & Medicinal Chemistry Letters
◽
10.1016/j.bmcl.2004.04.007
◽
2004
◽
Vol 14
(13)
◽
pp. 3581-3584
◽
Cited By ~ 101
Author(s):
J. Scott Sawyer
◽
Douglas W. Beight
◽
Karen S. Britt
◽
Bryan D. Anderson
◽
Robert M. Campbell
◽
...
Keyword(s):
Growth Factor
◽
Transforming Growth Factor
◽
Transforming Growth Factor Β
◽
Kinase Domain
◽
Type I
◽
Receptor Kinase
Download Full-text
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