Design, synthesis and evaluation of small molecule imidazo[2,1-b][1,3,4]thiadiazoles as inhibitors of transforming growth factor-β type-I receptor kinase (ALK5)

2015 ◽  
Vol 93 ◽  
pp. 599-613 ◽  
Author(s):  
Harun M. Patel ◽  
Baljeet Sing ◽  
Varun Bhardwaj ◽  
Mahesh Palkar ◽  
Mahamadhanif S. Shaikh ◽  
...  
Keyword(s):  
Growth Factor ◽  
Small Molecule ◽  
Transforming Growth Factor ◽  
Transforming Growth Factor Β ◽  
Type I ◽  
Receptor Kinase ◽  
Design Synthesis

Design, synthesis, and evaluation of novel 4-thiazolylimidazoles as inhibitors of transforming growth factor-β type I receptor kinase

2012 ◽  
Vol 22 (5) ◽  
pp. 2024-2029 ◽  
Author(s):  
Hideaki Amada ◽  
Yoshinori Sekiguchi ◽  
Naoya Ono ◽  
Yuko Matsunaga ◽  
Takeshi Koami ◽  
...  
Keyword(s):  
Growth Factor ◽  
Transforming Growth Factor ◽  
Transforming Growth Factor Β ◽  
Type I ◽  
Receptor Kinase ◽  
Design Synthesis

scholarly journals Inhibition of Pulmonary and Skeletal Metastasis by a Transforming Growth Factor-β Type I Receptor Kinase Inhibitor

2006 ◽  
Vol 66 (13) ◽  
pp. 6714-6721 ◽  
Author(s):  
Abhik Bandyopadhyay ◽  
Joseph K. Agyin ◽  
Long Wang ◽  
Yuping Tang ◽  
Xiufen Lei ◽  
...  
Keyword(s):  
Growth Factor ◽  
Transforming Growth Factor ◽  
Kinase Inhibitor ◽  
Skeletal Metastasis ◽  
Transforming Growth Factor Β ◽  
Type I ◽  
Receptor Kinase
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