Test No. 458: Stably Transfected Human Androgen Receptor Transcriptional Activation Assay for Detection of Androgenic Agonist and Antagonist Activity of Chemicals

Antagonist Activity ◽

Activation Assay ◽

Agonist And Antagonist ◽

Domains of the Human Androgen Receptor Involved in Steroid Binding, Transcriptional Activation, and Subcellular Localization

Molecular Endocrinology ◽

10.1210/mend-5-10-1396 ◽

1991 ◽

Vol 5 (10) ◽

pp. 1396-1404 ◽

Cited By ~ 336

Author(s):

Guido Jenster ◽

Hetty A. G. M. van der Korput ◽

Cor van Vroonhoven ◽

Theo H. van der Kwast ◽

Jan Trapman ◽

...

Keyword(s):

Androgen Receptor ◽

Subcellular Localization ◽

Steroid Binding ◽

Substitution of synthetic chimpanzee androgen receptor for human androgen receptor in competitive binding and transcriptional activation assays for EDC screening☆

Toxicology Letters ◽

10.1016/j.toxlet.2007.08.013 ◽

2007 ◽

Vol 174 (1-3) ◽

pp. 89-97 ◽

Cited By ~ 9

Author(s):

P HARTIG ◽

M CARDON ◽

C LAMBRIGHT ◽

K BOBSEINE ◽

L GRAYJR ◽

...

Keyword(s):

Androgen Receptor ◽

Competitive Binding ◽

Substitution of Cys-560 by Phe, Trp, Tyr, and Ser in the first zinc finger of human androgen receptor affects hormonal sensitivity and transcriptional activation.

Journal of Biological Chemistry ◽

10.1016/s0021-9258(19)62007-7 ◽

1994 ◽

Vol 269 (46) ◽

pp. 29016-29023

Author(s):

N Warriar ◽

C Yu ◽

N Pagé ◽

M V Govindan

Keyword(s):

Androgen Receptor ◽

Zinc Finger ◽

Agonist and antagonist switch DNA motifs recognized by human androgen receptor in prostate cancer

The EMBO Journal ◽

10.15252/embj.201490306 ◽

2014 ◽

Vol 34 (4) ◽

pp. 502-516 ◽

Cited By ~ 45

Author(s):

Zhong Chen ◽

Xun Lan ◽

Jennifer M Thomas‐Ahner ◽

Dayong Wu ◽

Xiangtao Liu ◽

...

Keyword(s):

Prostate Cancer ◽

Androgen Receptor ◽

Dna Motifs ◽

Agonist And Antagonist ◽

Evaluation of a rapid in vitro androgen receptor transcriptional activation assay using AR-EcoScreen™ cells

Toxicology in Vitro ◽

10.1016/j.tiv.2004.10.008 ◽

2005 ◽

Vol 19 (3) ◽

pp. 335-352 ◽

Cited By ~ 29

Author(s):

Naohiro Araki ◽

Ken Ohno ◽

Masahiro Takeyoshi ◽

Mitsuru Iida

Keyword(s):

Androgen Receptor ◽

Activation Assay

Transcriptional activation and nuclear targeting signals of the human androgen receptor.

Journal of Biological Chemistry ◽

10.1016/s0021-9258(18)52466-2 ◽

1991 ◽

Vol 266 (1) ◽

pp. 510-518 ◽

Cited By ~ 3

Author(s):

J A Simental ◽

M Sar ◽

M V Lane ◽

F S French ◽

E M Wilson

Keyword(s):

Androgen Receptor ◽

Nuclear Targeting ◽

Targeting Signals ◽

Metabolite Profiling and a Transcriptional Activation Assay Provide Direct Evidence of Androgen Receptor Antagonism by Bisphenol A in Fish

Environmental Science & Technology ◽

10.1021/es3014634 ◽

2012 ◽

Vol 46 (17) ◽

pp. 9673-9680 ◽

Cited By ~ 32

Author(s):

D. R. Ekman ◽

P. C. Hartig ◽

M. Cardon ◽

D. M. Skelton ◽

Q. Teng ◽

...

Keyword(s):

Androgen Receptor ◽

Bisphenol A ◽

Metabolite Profiling ◽

Direct Evidence ◽

Receptor Antagonism ◽

Activation Assay

Transcriptional activation and transient expression of the human androgen receptor

The Journal of Steroid Biochemistry and Molecular Biology ◽

10.1016/s0960-0760(96)00097-0 ◽

1996 ◽

Vol 59 (1) ◽

pp. 9-20 ◽

Cited By ~ 96

Author(s):

Tianshu Gao ◽

Marco Marcelli ◽

Michael J. McPhaul

Keyword(s):

Androgen Receptor ◽

Transient Expression ◽

Endocrine disrupting potential of veterinary drugs by in vitro stably transfected human androgen receptor transcriptional activation assays

Environmental Pollution ◽

10.1016/j.envpol.2021.117201 ◽

2021 ◽

pp. 117201

Author(s):

Yooheon Park ◽

Juhee Park ◽

Hee-Seok Lee

Keyword(s):

Androgen Receptor ◽

Veterinary Drugs ◽

Endocrine Disrupting ◽

417: The Human Androgen Receptor Gene is a Primary Target of the WNT Signaling Pathway

The Journal of Urology ◽

10.1016/s0022-5347(18)32673-9 ◽

2006 ◽

Vol 175 (4S) ◽

pp. 136-136

Author(s):

Ralph Buttyan ◽

Xuezhen Yang ◽

Min-Wei Chen ◽

Debra L. Bemis ◽

Mitchell C. Benson ◽

...

Keyword(s):

Androgen Receptor ◽

Wnt Signaling ◽

Signaling Pathway ◽

Receptor Gene ◽

Wnt Signaling Pathway ◽

Androgen Receptor Gene ◽

Primary Target ◽

Human Androgen Receptor Gene ◽